SK8132001A3 - Sulphonyloxazolamines as therapeutic active ingredients - Google Patents
Sulphonyloxazolamines as therapeutic active ingredients Download PDFInfo
- Publication number
- SK8132001A3 SK8132001A3 SK813-2001A SK8132001A SK8132001A3 SK 8132001 A3 SK8132001 A3 SK 8132001A3 SK 8132001 A SK8132001 A SK 8132001A SK 8132001 A3 SK8132001 A3 SK 8132001A3
- Authority
- SK
- Slovakia
- Prior art keywords
- formula
- oxazol
- compounds
- amine
- benzenesulfonyl
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
- C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
- C07D263/30—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D263/34—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D263/48—Nitrogen atoms not forming part of a nitro radical
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- General Chemical & Material Sciences (AREA)
- Psychiatry (AREA)
- Psychology (AREA)
- Pain & Pain Management (AREA)
- Hospice & Palliative Care (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE19858593A DE19858593A1 (de) | 1998-12-18 | 1998-12-18 | Sulfonyloxazolamine als therapeutische Wirkstoffe |
| PCT/EP1999/009335 WO2000037452A1 (de) | 1998-12-18 | 1999-12-01 | Sulfonyloxazolamine als therapeutische wirkstoffe |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| SK8132001A3 true SK8132001A3 (en) | 2002-02-05 |
Family
ID=7891645
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| SK813-2001A SK8132001A3 (en) | 1998-12-18 | 1999-12-01 | Sulphonyloxazolamines as therapeutic active ingredients |
Country Status (19)
| Country | Link |
|---|---|
| US (1) | US6441013B1 (id) |
| EP (1) | EP1140875A1 (id) |
| JP (1) | JP2002533332A (id) |
| CN (1) | CN1146549C (id) |
| AR (1) | AR021896A1 (id) |
| AU (1) | AU763070B2 (id) |
| BR (1) | BR9916310A (id) |
| CA (1) | CA2356134A1 (id) |
| CZ (1) | CZ20012144A3 (id) |
| DE (1) | DE19858593A1 (id) |
| HK (1) | HK1043125A1 (id) |
| HU (1) | HUP0104834A3 (id) |
| ID (1) | ID29966A (id) |
| NO (1) | NO20012965D0 (id) |
| PL (1) | PL349393A1 (id) |
| RU (1) | RU2232757C2 (id) |
| SK (1) | SK8132001A3 (id) |
| WO (1) | WO2000037452A1 (id) |
| ZA (1) | ZA200105881B (id) |
Families Citing this family (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE19956791A1 (de) * | 1999-11-25 | 2001-05-31 | Merck Patent Gmbh | Neue Sulfonyloxazolamine |
| DE10129940A1 (de) * | 2001-06-13 | 2002-12-19 | Merck Patent Gmbh | Sulfonyloxazolamine als therapeutische Wirkstoffe |
| US6875771B2 (en) * | 2002-07-26 | 2005-04-05 | Bristol-Myers Squibb Company | Pyridopyrimidine derivatives as 5-HT6 antagonists |
| FR2854632B1 (fr) * | 2003-05-07 | 2005-06-17 | Centre Nat Rech Scient | Synthese de composes heterocycliques substitues |
| DK1831159T3 (da) * | 2004-12-21 | 2010-03-22 | Hoffmann La Roche | Tetralin og indanderivater samt anvendelser deraf |
| SG172738A1 (en) * | 2005-07-29 | 2011-07-28 | 4Sc Ag | Novel heterocyclic nf-kb inhibitors |
| WO2008061248A2 (en) * | 2006-11-16 | 2008-05-22 | The Regents Of The University Of California | Phenylsulfoxyoxazole compound inhibitors of urea transporters |
| KR101174191B1 (ko) * | 2007-02-02 | 2012-08-14 | 에프. 호프만-라 로슈 아게 | 중추 신경계 장애의 치료용 ｔａａｒ1 리간드로서 2-아미노옥사졸린 |
| WO2008098857A1 (en) * | 2007-02-15 | 2008-08-21 | F. Hoffmann-La Roche Ag | 2-aminooxazolines as taar1 ligands |
| RU2443697C1 (ru) | 2010-12-21 | 2012-02-27 | Александр Васильевич Иващенко | Замещенные метил-амины, антагонисты серотониновых 5-ht6 рецепторов, способы получения и применения |
| CN109789129B (zh) * | 2016-07-12 | 2022-04-29 | 延世大学校产学协力团 | 自噬改良材料及其用途 |
| KR102533605B1 (ko) * | 2018-01-10 | 2023-05-17 | 주식회사 라이조테크 | 신규한 페닐설포닐 옥사졸 유도체 및 이의 용도 |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| HUP0002351A3 (en) | 1996-02-20 | 2001-10-29 | Bristol Myers Squibb Co | Methods for the preparation of biphenyl isoxazole sulfonamides, intermediates and process for preparing them |
-
1998
- 1998-12-18 DE DE19858593A patent/DE19858593A1/de not_active Withdrawn
-
1999
- 1999-12-01 JP JP2000589524A patent/JP2002533332A/ja active Pending
- 1999-12-01 AU AU18612/00A patent/AU763070B2/en not_active Ceased
- 1999-12-01 ID IDW00200101555A patent/ID29966A/id unknown
- 1999-12-01 SK SK813-2001A patent/SK8132001A3/sk unknown
- 1999-12-01 US US09/868,097 patent/US6441013B1/en not_active Expired - Fee Related
- 1999-12-01 EP EP99962190A patent/EP1140875A1/de not_active Withdrawn
- 1999-12-01 CN CNB998147281A patent/CN1146549C/zh not_active Expired - Fee Related
- 1999-12-01 BR BR9916310-1A patent/BR9916310A/pt not_active IP Right Cessation
- 1999-12-01 PL PL99349393A patent/PL349393A1/xx unknown
- 1999-12-01 HU HU0104834A patent/HUP0104834A3/hu unknown
- 1999-12-01 WO PCT/EP1999/009335 patent/WO2000037452A1/de not_active Application Discontinuation
- 1999-12-01 RU RU2001119273/04A patent/RU2232757C2/ru not_active IP Right Cessation
- 1999-12-01 CZ CZ20012144A patent/CZ20012144A3/cs unknown
- 1999-12-01 CA CA002356134A patent/CA2356134A1/en not_active Abandoned
- 1999-12-17 AR ARP990106528A patent/AR021896A1/es not_active Application Discontinuation
-
2001
- 2001-06-15 NO NO20012965A patent/NO20012965D0/no not_active Application Discontinuation
- 2001-07-17 ZA ZA200105881A patent/ZA200105881B/en unknown
-
2002
- 2002-07-02 HK HK02104944.7A patent/HK1043125A1/zh unknown
Also Published As
| Publication number | Publication date |
|---|---|
| ID29966A (id) | 2001-10-25 |
| BR9916310A (pt) | 2001-11-06 |
| EP1140875A1 (de) | 2001-10-10 |
| ZA200105881B (en) | 2002-10-17 |
| HUP0104834A3 (en) | 2005-06-28 |
| JP2002533332A (ja) | 2002-10-08 |
| HK1043125A1 (zh) | 2002-09-06 |
| US6441013B1 (en) | 2002-08-27 |
| DE19858593A1 (de) | 2000-06-21 |
| AR021896A1 (es) | 2002-08-07 |
| WO2000037452A1 (de) | 2000-06-29 |
| HUP0104834A2 (hu) | 2002-07-29 |
| NO20012965L (no) | 2001-06-15 |
| RU2232757C2 (ru) | 2004-07-20 |
| NO20012965D0 (no) | 2001-06-15 |
| CA2356134A1 (en) | 2000-06-29 |
| PL349393A1 (en) | 2002-07-15 |
| CN1146549C (zh) | 2004-04-21 |
| AU1861200A (en) | 2000-07-12 |
| CN1331684A (zh) | 2002-01-16 |
| AU763070B2 (en) | 2003-07-10 |
| CZ20012144A3 (cs) | 2002-01-16 |
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