SK4972003A3 - 5-spiro-pyrimidine-2,4,6-trione metalloproteinase inhibitors - Google Patents

5-spiro-pyrimidine-2,4,6-trione metalloproteinase inhibitors Download PDF

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Publication number
SK4972003A3
SK4972003A3 SK497-2003A SK4972003A SK4972003A3 SK 4972003 A3 SK4972003 A3 SK 4972003A3 SK 4972003 A SK4972003 A SK 4972003A SK 4972003 A3 SK4972003 A3 SK 4972003A3
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SK
Slovakia
Prior art keywords
group
alkyl
pyridin
triazaspiro
compounds
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Application number
SK497-2003A
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English (en)
Slovak (sk)
Inventor
Brian Scott Bronk
Mark Carl Noe
Martin James Wythes
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Pfizer Prod Inc
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Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Publication of SK4972003A3 publication Critical patent/SK4972003A3/sk

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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/10Spiro-condensed systems
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  • Chemical Kinetics & Catalysis (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
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  • Endocrinology (AREA)
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  • Dermatology (AREA)
  • Communicable Diseases (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Pain & Pain Management (AREA)
  • Pulmonology (AREA)
  • Diabetes (AREA)
  • Gynecology & Obstetrics (AREA)
  • Cardiology (AREA)
  • Virology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Pregnancy & Childbirth (AREA)
  • Hematology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Psychiatry (AREA)
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SK497-2003A 2000-10-26 2001-10-23 5-spiro-pyrimidine-2,4,6-trione metalloproteinase inhibitors SK4972003A3 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US24338900P 2000-10-26 2000-10-26
PCT/IB2001/001986 WO2002034753A2 (en) 2000-10-26 2001-10-23 Spiro-pyrimidine-2,4,6-trione metalloproteinase inhibitors

Publications (1)

Publication Number Publication Date
SK4972003A3 true SK4972003A3 (en) 2004-05-04

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Application Number Title Priority Date Filing Date
SK497-2003A SK4972003A3 (en) 2000-10-26 2001-10-23 5-spiro-pyrimidine-2,4,6-trione metalloproteinase inhibitors

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EP (1) EP1332146A2 (es)
JP (1) JP2004518635A (es)
KR (1) KR20040004412A (es)
CN (1) CN1501937A (es)
AP (1) AP2001002318A0 (es)
AR (1) AR035069A1 (es)
AU (1) AU2002210813A1 (es)
BG (1) BG107653A (es)
BR (1) BR0114913A (es)
CA (1) CA2425283A1 (es)
CZ (1) CZ20031083A3 (es)
EA (1) EA005762B1 (es)
EC (1) ECSP034567A (es)
EE (1) EE200300196A (es)
GT (1) GT200100213A (es)
HN (1) HN2001000244A (es)
HR (1) HRP20030332A2 (es)
HU (1) HUP0301577A3 (es)
IL (1) IL154948A0 (es)
IS (1) IS6762A (es)
MA (1) MA26957A1 (es)
MX (1) MXPA03003735A (es)
NO (1) NO20031853L (es)
OA (1) OA12529A (es)
PA (1) PA8531401A1 (es)
PE (1) PE20020589A1 (es)
PL (1) PL366201A1 (es)
SK (1) SK4972003A3 (es)
SV (1) SV2003000705A (es)
TN (1) TNSN01149A1 (es)
WO (1) WO2002034753A2 (es)
ZA (1) ZA200302190B (es)

Families Citing this family (36)

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MXPA03004920A (es) 2001-02-14 2003-09-05 Warner Lambert Co Pirimidinas inhibidoras de metaloproteinasas de matriz.
DOP2002000333A (es) 2001-02-14 2002-09-30 Warner Lambert Co Derivados de acido isoftalico como inhibidores de metaloproteinasas de la matriz
DOP2002000332A (es) 2001-02-14 2002-08-30 Warner Lambert Co Inhibidores de piridina de metaloproteinasas de la matriz
PA8539501A1 (es) 2001-02-14 2002-09-30 Warner Lambert Co Compuestos triazolo como inhibidores de mmp
JP2004518726A (ja) 2001-02-14 2004-06-24 ワーナー−ランバート・カンパニー、リミテッド、ライアビリティ、カンパニー ベンゾチアジアジンマトリックスメタロプロテイナーゼ阻害剤
US6924276B2 (en) 2001-09-10 2005-08-02 Warner-Lambert Company Diacid-substituted heteroaryl derivatives as matrix metalloproteinase inhibitors
US6962922B2 (en) 2001-10-12 2005-11-08 Warner-Lambert Company Llc Alkynylated quinazoline compounds
CA2462442A1 (en) 2001-10-12 2003-04-24 Warner-Lambert Company Llc Alkyne matrix metalloproteinase inhibitors
US6894057B2 (en) 2002-03-08 2005-05-17 Warner-Lambert Company Oxo-azabicyclic compounds
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