SK287477B6 - Spôsob prípravy 2-[5-(fluórfenyl)-3-pyridylmetylaminometyl]- chrománu - Google Patents

Spôsob prípravy 2-[5-(fluórfenyl)-3-pyridylmetylaminometyl]- chrománu Download PDF

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Publication number
SK287477B6
SK287477B6 SK1433-2003A SK14332003A SK287477B6 SK 287477 B6 SK287477 B6 SK 287477B6 SK 14332003 A SK14332003 A SK 14332003A SK 287477 B6 SK287477 B6 SK 287477B6
Authority
SK
Slovakia
Prior art keywords
fluorophenyl
aminomethylchroman
pyridylmethylaminomethyl
formula
salts
Prior art date
Application number
SK1433-2003A
Other languages
English (en)
Slovak (sk)
Other versions
SK14332003A3 (sk
Inventor
Heinz-Hermann Bokel
Steffen Neunfeld
Ludwig Gantzert
Ralf Knierieme
Elke Simon
Ralf Devant
Udo Helm
Helmut Reubold
Original Assignee
Merck Patent Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck Patent Gmbh filed Critical Merck Patent Gmbh
Publication of SK14332003A3 publication Critical patent/SK14332003A3/sk
Publication of SK287477B6 publication Critical patent/SK287477B6/sk

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D311/00—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings
    • C07D311/02—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D311/04—Benzo[b]pyrans, not hydrogenated in the carbocyclic ring
    • C07D311/58—Benzo[b]pyrans, not hydrogenated in the carbocyclic ring other than with oxygen or sulphur atoms in position 2 or 4

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pyridine Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
SK1433-2003A 2001-04-26 2002-04-08 Spôsob prípravy 2-[5-(fluórfenyl)-3-pyridylmetylaminometyl]- chrománu SK287477B6 (sk)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE10120619A DE10120619A1 (de) 2001-04-26 2001-04-26 2-(5-(4-Fluorphenyl)-3-pyridylmethylaminomethyl-chroman
PCT/EP2002/003857 WO2002088117A2 (de) 2001-04-26 2002-04-08 Verfahren zur herstellung von 2-[-5-(4-fluorphenyl)-3-pyridylmethylaminomethyl]-chroman

Publications (2)

Publication Number Publication Date
SK14332003A3 SK14332003A3 (sk) 2004-04-06
SK287477B6 true SK287477B6 (sk) 2010-11-08

Family

ID=7682908

Family Applications (1)

Application Number Title Priority Date Filing Date
SK1433-2003A SK287477B6 (sk) 2001-04-26 2002-04-08 Spôsob prípravy 2-[5-(fluórfenyl)-3-pyridylmetylaminometyl]- chrománu

Country Status (24)

Country Link
US (1) US7045629B2 (cs)
EP (1) EP1383763B1 (cs)
JP (1) JP2004526797A (cs)
KR (1) KR100839168B1 (cs)
CN (1) CN100430391C (cs)
AR (1) AR033262A1 (cs)
AT (1) ATE306485T1 (cs)
AU (1) AU2002257763B2 (cs)
BR (1) BR0209179A (cs)
CA (1) CA2445207C (cs)
CZ (1) CZ301615B6 (cs)
DE (2) DE10120619A1 (cs)
DK (1) DK1383763T3 (cs)
ES (1) ES2250647T3 (cs)
HK (1) HK1077302A1 (cs)
HU (1) HU229151B1 (cs)
MX (1) MXPA03009684A (cs)
MY (1) MY130616A (cs)
PL (1) PL208705B1 (cs)
RU (1) RU2288229C2 (cs)
SI (1) SI1383763T1 (cs)
SK (1) SK287477B6 (cs)
WO (1) WO2002088117A2 (cs)
ZA (1) ZA200309164B (cs)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP4896518B2 (ja) * 2002-12-13 2012-03-14 ワイエム・バイオサイエンシズ・オーストラリア・ピーティーワイ・リミテッド ニコチンアミド系キナーゼ阻害薬
BRPI0608353A2 (pt) * 2005-02-17 2009-12-01 Wyeth Corp derivados de indol, benzotiofeno, benzofurano e indeno cicloalquilfundidos
AU2006239937A1 (en) * 2005-04-22 2006-11-02 Wyeth Chromane and chromene derivatives and uses thereof
MX2007015359A (es) * 2005-06-21 2008-02-15 Merck Patent Gmbh Preparacion farmaceutica solida que contiene (r)-(-)-2-[5-(4- fluorofenil)-3-piridilmetilaminometil]-cromano.
EP2012778A4 (en) * 2006-04-18 2011-08-10 Abbott Lab VANILLOID RECEPTOR (VR1) SUBType 1 ANTAGONISTS AND USES THEREOF
BR112013001257A2 (pt) * 2010-07-20 2016-05-17 Glaxo Group Ltd processo.

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE4135474A1 (de) * 1991-10-28 1993-04-29 Bayer Ag 2-aminomethyl-chromane
FR2701479B1 (fr) 1993-02-11 1995-05-12 Pf Medicament Nouveaux dérivés hétérocycliques de l'aminométhyl-4 pipéridine, leur préparation et leur application en thérapeutique.
US5824682A (en) * 1993-08-18 1998-10-20 Janssen Pharmaceutica, N.V. Vasoconstrictive dihydrobenzopyran derivatives
GB9318431D0 (en) * 1993-09-06 1993-10-20 Boots Co Plc Therapeutic agents
EP1123933A1 (en) * 1994-10-14 2001-08-16 MERCK PATENT GmbH 2-[5-(4-fluorophenyl)-3-pyridylmethylaminomethyl]chromane as CNS active agent
DE10005150A1 (de) 2000-02-07 2001-08-09 Merck Patent Gmbh Verfahren zur Herstellung von 5-Arylnicotinaldehyden

Also Published As

Publication number Publication date
KR20040010616A (ko) 2004-01-31
WO2002088117A2 (de) 2002-11-07
CZ20033214A3 (cs) 2004-02-18
US7045629B2 (en) 2006-05-16
CA2445207A1 (en) 2002-11-07
MXPA03009684A (es) 2004-02-12
DE50204535D1 (de) 2006-02-23
DE10120619A1 (de) 2002-10-31
RU2288229C2 (ru) 2006-11-27
AR033262A1 (es) 2003-12-10
EP1383763A2 (de) 2004-01-28
MY130616A (en) 2007-07-31
HU229151B1 (hu) 2013-09-30
HUP0303969A2 (hu) 2004-04-28
CA2445207C (en) 2010-03-02
WO2002088117A3 (de) 2002-12-27
BR0209179A (pt) 2004-08-03
ZA200309164B (en) 2004-09-29
CZ301615B6 (cs) 2010-05-05
SK14332003A3 (sk) 2004-04-06
ES2250647T3 (es) 2006-04-16
ATE306485T1 (de) 2005-10-15
DK1383763T3 (da) 2006-02-06
CN100430391C (zh) 2008-11-05
EP1383763B1 (de) 2005-10-12
HK1077302A1 (en) 2006-02-10
HUP0303969A3 (en) 2011-02-28
SI1383763T1 (sl) 2006-04-30
US20040138266A1 (en) 2004-07-15
PL208705B1 (pl) 2011-05-31
KR100839168B1 (ko) 2008-06-17
CN1622944A (zh) 2005-06-01
RU2003132433A (ru) 2005-04-20
PL363281A1 (en) 2004-11-15
AU2002257763B2 (en) 2007-03-15
JP2004526797A (ja) 2004-09-02

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Legal Events

Date Code Title Description
MM4A Patent lapsed due to non-payment of maintenance fees

Effective date: 20120408