FR2701479B1 - Nouveaux dérivés hétérocycliques de l'aminométhyl-4 pipéridine, leur préparation et leur application en thérapeutique. - Google Patents

Nouveaux dérivés hétérocycliques de l'aminométhyl-4 pipéridine, leur préparation et leur application en thérapeutique.

Info

Publication number
FR2701479B1
FR2701479B1 FR9301525A FR9301525A FR2701479B1 FR 2701479 B1 FR2701479 B1 FR 2701479B1 FR 9301525 A FR9301525 A FR 9301525A FR 9301525 A FR9301525 A FR 9301525A FR 2701479 B1 FR2701479 B1 FR 2701479B1
Authority
FR
France
Prior art keywords
preparation
therapeutic use
heterocyclic derivatives
new heterocyclic
aminomethyl piperidine
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
FR9301525A
Other languages
English (en)
Other versions
FR2701479A1 (fr
Inventor
Dennis Bigg
Florence Castan
Wouter Koek
Bernard Bonnaud
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pierre Fabre Medicament SA
Original Assignee
Pierre Fabre Medicament SA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority to FR9301525A priority Critical patent/FR2701479B1/fr
Application filed by Pierre Fabre Medicament SA filed Critical Pierre Fabre Medicament SA
Priority to ZA94910A priority patent/ZA94910B/xx
Priority to PCT/FR1994/000152 priority patent/WO1994018193A1/fr
Priority to EP94906261A priority patent/EP0683775A1/fr
Priority to CA002155849A priority patent/CA2155849A1/fr
Priority to NZ261331A priority patent/NZ261331A/en
Priority to AU60033/94A priority patent/AU6003394A/en
Priority to JP6517735A priority patent/JPH08506334A/ja
Publication of FR2701479A1 publication Critical patent/FR2701479A1/fr
Application granted granted Critical
Publication of FR2701479B1 publication Critical patent/FR2701479B1/fr
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/20Hypnotics; Sedatives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/26Psychostimulants, e.g. nicotine, cocaine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/04Anorexiants; Antiobesity agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D411/00Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen and sulfur atoms as the only ring hetero atoms
    • C07D411/02Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen and sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D411/12Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen and sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
FR9301525A 1993-02-11 1993-02-11 Nouveaux dérivés hétérocycliques de l'aminométhyl-4 pipéridine, leur préparation et leur application en thérapeutique. Expired - Fee Related FR2701479B1 (fr)

Priority Applications (8)

Application Number Priority Date Filing Date Title
FR9301525A FR2701479B1 (fr) 1993-02-11 1993-02-11 Nouveaux dérivés hétérocycliques de l'aminométhyl-4 pipéridine, leur préparation et leur application en thérapeutique.
PCT/FR1994/000152 WO1994018193A1 (fr) 1993-02-11 1994-02-10 Nouveaux derives heterocycliques de l'aminomethyl-4 piperidine, leur preparation et leur application en therapeutique
EP94906261A EP0683775A1 (fr) 1993-02-11 1994-02-10 Derives heterocycliques de l'aminomethyl-4 piperidine, leur preparation et leur application en therapeutique
CA002155849A CA2155849A1 (fr) 1993-02-11 1994-02-10 Nouveaux derives heterocycliques de l'aminomethyl-4 piperidine, leur preparation et leur application en therapeutique
ZA94910A ZA94910B (en) 1993-02-11 1994-02-10 New heterocyclic 4-(aminomethyl) piperidine derivatives preparations thereof and application thereof in therapeutics
NZ261331A NZ261331A (en) 1993-02-11 1994-02-10 Heterocyclically-substituted 4-aminomethylpiperidines and pharmaceutical compositions
AU60033/94A AU6003394A (en) 1993-02-11 1994-02-10 Novel heterocyclic aminomethyl-4 piperidine derivatives, their preparation and application in therapy
JP6517735A JPH08506334A (ja) 1993-02-11 1994-02-10 新規な複素環式アミノメチル‐4 ピペリジン誘導体、その調製および治療への使用

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR9301525A FR2701479B1 (fr) 1993-02-11 1993-02-11 Nouveaux dérivés hétérocycliques de l'aminométhyl-4 pipéridine, leur préparation et leur application en thérapeutique.

Publications (2)

Publication Number Publication Date
FR2701479A1 FR2701479A1 (fr) 1994-08-19
FR2701479B1 true FR2701479B1 (fr) 1995-05-12

Family

ID=9443949

Family Applications (1)

Application Number Title Priority Date Filing Date
FR9301525A Expired - Fee Related FR2701479B1 (fr) 1993-02-11 1993-02-11 Nouveaux dérivés hétérocycliques de l'aminométhyl-4 pipéridine, leur préparation et leur application en thérapeutique.

Country Status (8)

Country Link
EP (1) EP0683775A1 (fr)
JP (1) JPH08506334A (fr)
AU (1) AU6003394A (fr)
CA (1) CA2155849A1 (fr)
FR (1) FR2701479B1 (fr)
NZ (1) NZ261331A (fr)
WO (1) WO1994018193A1 (fr)
ZA (1) ZA94910B (fr)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2725989B1 (fr) * 1994-10-20 1997-01-10 Pf Medicament Nouvelles 2-(1-(omega-phenoxyalcoylpiperidin-4-yl) aminomethylene)-2h-benzofuran-3-ones substituees, leur preparation et leur application en therapeutique
GB9627006D0 (en) * 1996-12-27 1997-02-12 Knoll Ag Therapeutic agents
GB9811879D0 (en) * 1998-06-03 1998-07-29 Knoll Ag Therapeutic agents
DE10120619A1 (de) 2001-04-26 2002-10-31 Merck Patent Gmbh 2-(5-(4-Fluorphenyl)-3-pyridylmethylaminomethyl-chroman
US7728155B2 (en) 2003-10-24 2010-06-01 Wyeth Llc Dihydrobenzofuranyl alkanamines and methods for using same as cns agents
WO2008052078A2 (fr) * 2006-10-24 2008-05-02 Wyeth Dérivés de benzoxathine et de benzoxathiole, et leurs utilisations

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4910302A (en) * 1988-12-19 1990-03-20 American Home Products Corporation Psychotropic polycyclic imides
FR2658823B1 (fr) * 1990-02-27 1992-04-30 Adir Nouveaux derives d'aminomethylpiperidine, leur procede de preparation et les compositions pharmaceutiques qui les contiennent .
FR2659323B1 (fr) * 1990-03-07 1992-06-12 Synthelabo Derives de 4-(aminomethyl) piperidine, leur preparation et leur application en therapeutique.
FR2660657B1 (fr) * 1990-04-09 1993-05-07 Adir Nouveaux derives du 3-aminochromane, leur procede de preparation et les compositions pharmaceutiques qui les contiennent.

Also Published As

Publication number Publication date
WO1994018193A1 (fr) 1994-08-18
EP0683775A1 (fr) 1995-11-29
FR2701479A1 (fr) 1994-08-19
AU6003394A (en) 1994-08-29
JPH08506334A (ja) 1996-07-09
ZA94910B (en) 1994-08-22
CA2155849A1 (fr) 1994-08-18
NZ261331A (en) 1996-05-28

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Legal Events

Date Code Title Description
ST Notification of lapse