SK287309B6 - Spôsob prípravy dibenzotiazepínových derivátov - Google Patents

Spôsob prípravy dibenzotiazepínových derivátov Download PDF

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Publication number
SK287309B6
SK287309B6 SK31-2002A SK312002A SK287309B6 SK 287309 B6 SK287309 B6 SK 287309B6 SK 312002 A SK312002 A SK 312002A SK 287309 B6 SK287309 B6 SK 287309B6
Authority
SK
Slovakia
Prior art keywords
carboxy
derivative
diphenylsulfide
group
general formula
Prior art date
Application number
SK31-2002A
Other languages
English (en)
Slovak (sk)
Other versions
SK312002A3 (en
Inventor
Katsumasa Harada
Shigeyoshi Nishino
Kiyotaka Yoshii
Original Assignee
Astrazeneca Uk Limited
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astrazeneca Uk Limited filed Critical Astrazeneca Uk Limited
Publication of SK312002A3 publication Critical patent/SK312002A3/sk
Publication of SK287309B6 publication Critical patent/SK287309B6/sk

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D281/00Heterocyclic compounds containing rings of more than six members having one nitrogen atom and one sulfur atom as the only ring hetero atoms
    • C07D281/02Seven-membered rings
    • C07D281/04Seven-membered rings having the hetero atoms in positions 1 and 4
    • C07D281/08Seven-membered rings having the hetero atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D281/12Seven-membered rings having the hetero atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems condensed with two six-membered rings
    • C07D281/14[b, e]-condensed
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C319/00Preparation of thiols, sulfides, hydropolysulfides or polysulfides
    • C07C319/14Preparation of thiols, sulfides, hydropolysulfides or polysulfides of sulfides
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C323/00Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups
    • C07C323/50Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton
    • C07C323/62Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton having the sulfur atom of at least one of the thio groups bound to a carbon atom of a six-membered aromatic ring of the carbon skeleton
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D281/00Heterocyclic compounds containing rings of more than six members having one nitrogen atom and one sulfur atom as the only ring hetero atoms
    • C07D281/02Seven-membered rings
    • C07D281/04Seven-membered rings having the hetero atoms in positions 1 and 4
    • C07D281/08Seven-membered rings having the hetero atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D281/12Seven-membered rings having the hetero atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems condensed with two six-membered rings
    • C07D281/16[b, f]-condensed

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Neurosurgery (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biomedical Technology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Psychiatry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Neurology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
SK31-2002A 1999-07-09 1999-07-09 Spôsob prípravy dibenzotiazepínových derivátov SK287309B6 (sk)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
PCT/JP1999/003719 WO2001004106A1 (fr) 1999-07-09 1999-07-09 Procede de production de derives de dibenzothiazepine

Publications (2)

Publication Number Publication Date
SK312002A3 SK312002A3 (en) 2002-06-04
SK287309B6 true SK287309B6 (sk) 2010-06-07

Family

ID=14236203

Family Applications (1)

Application Number Title Priority Date Filing Date
SK31-2002A SK287309B6 (sk) 1999-07-09 1999-07-09 Spôsob prípravy dibenzotiazepínových derivátov

Country Status (21)

Country Link
US (2) US7045621B1 (zh)
EP (1) EP1201663A4 (zh)
JP (1) JP4688383B2 (zh)
KR (1) KR100604690B1 (zh)
CN (1) CN1247556C (zh)
AU (1) AU782988B2 (zh)
BR (1) BR9917400A (zh)
CA (1) CA2379294C (zh)
CZ (1) CZ301061B6 (zh)
EE (1) EE05609B1 (zh)
HK (1) HK1047278B (zh)
HU (1) HUP0202247A3 (zh)
IL (3) IL147379A0 (zh)
MX (1) MXPA02000136A (zh)
NO (2) NO322420B1 (zh)
NZ (1) NZ516851A (zh)
PL (1) PL201699B1 (zh)
RU (1) RU2233275C2 (zh)
SK (1) SK287309B6 (zh)
TW (1) TWI265165B (zh)
WO (1) WO2001004106A1 (zh)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20030216376A1 (en) * 2002-03-20 2003-11-20 Revital Lifshitz-Liron Crystalline forms of quetiapine hemifumarate
KR100707050B1 (ko) * 2002-11-28 2007-04-13 에스케이 주식회사 10H-디벤조[b,f][1,4]티아제핀-11-온의 제조방법
US20060081361A1 (en) * 2004-09-13 2006-04-20 Gabbey Lawrence W Oil cooler with integral filter
EP1869007A1 (en) * 2005-04-14 2007-12-26 Teva Pharmaceutical Industries Ltd Process for preparing quetiapine fumarate
KR20080108468A (ko) * 2006-02-22 2008-12-15 아스트라제네카 유케이 리미티드 디벤조티아제핀 화합물의 제조 방법
EP2144892A2 (en) * 2007-03-29 2010-01-20 Teva Pharmaceutical Industries Ltd. Improved process for preparing quetiapine fumarate
JP2011126887A (ja) * 2011-01-11 2011-06-30 Ube Industries Ltd ジベンゾチアゼピン誘導体の製造法
GB201106520D0 (en) * 2011-04-18 2011-06-01 Numedicus Ltd Pharmaceutical compounds

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3560622A (en) * 1967-10-13 1971-02-02 American Cyanamid Co Trifluoromethyl oxazepines,thiazepines and diazepines as anti-inflammatory agents
JPS60202879A (ja) * 1984-02-06 1985-10-14 ワ−ナ−−ランバ−ト・コンパニ− 1,4−アミノアルキルアミノ−9h−チオキサンテン−9−オン
GB9109497D0 (en) 1991-05-02 1991-06-26 Wellcome Found Chemical compounds
GB9109557D0 (en) * 1991-05-02 1991-06-26 Wellcome Found Chemical compounds
US5180720A (en) * 1991-05-03 1993-01-19 G. D. Searle & Co. 2- and 3-alkoxy or hydroxy-8-substituted-dibenz[b,f]-[1,4]oxazepine-10(11H)-carboxylic acid, substituted hydrazides and methods for treating pain
SE9500998D0 (sv) * 1995-03-19 1995-03-19 Haakan Wilhelm Wikstroem New sulfone ester analogues of iso-clozapine and related structures: atypical neuroleptics
US6207837B1 (en) * 1997-07-18 2001-03-27 Nippon Suisan Kaisha, Ltd. Process for producing dibenzo[b,f]thiepine derivatives
JP3865096B2 (ja) 1998-01-09 2007-01-10 宇部興産株式会社 ジベンゾチアゼピン誘導体の製造方法

Also Published As

Publication number Publication date
TWI265165B (en) 2006-11-01
HUP0202247A1 (en) 2002-10-28
IL147379A (en) 2008-04-13
HUP0202247A3 (en) 2002-12-28
CA2379294C (en) 2009-10-20
NO20063661L (no) 2002-03-04
EP1201663A4 (en) 2005-02-16
BR9917400A (pt) 2004-01-06
NO20020059L (no) 2002-03-04
CZ200276A3 (cs) 2002-04-17
CA2379294A1 (en) 2001-01-18
CN1367782A (zh) 2002-09-04
HK1047278A1 (en) 2003-02-14
IL189161A0 (en) 2009-02-11
IL189161A (en) 2010-05-31
US7045621B1 (en) 2006-05-16
KR20020022767A (ko) 2002-03-27
KR100604690B1 (ko) 2006-07-25
US7314930B2 (en) 2008-01-01
IL147379A0 (en) 2002-08-14
NO322420B1 (no) 2006-10-02
CN1247556C (zh) 2006-03-29
RU2233275C2 (ru) 2004-07-27
CZ301061B6 (cs) 2009-10-29
HK1047278B (zh) 2006-09-29
AU4650699A (en) 2001-01-30
AU782988B2 (en) 2005-09-15
US20060173178A1 (en) 2006-08-03
JP4688383B2 (ja) 2011-05-25
EE05609B1 (et) 2012-12-17
PL201699B1 (pl) 2009-04-30
WO2001004106A1 (fr) 2001-01-18
NZ516851A (en) 2004-02-27
MXPA02000136A (es) 2002-07-02
EP1201663A1 (en) 2002-05-02
PL352928A1 (en) 2003-09-22
EE200200014A (et) 2003-04-15
NO20020059D0 (no) 2002-01-07
SK312002A3 (en) 2002-06-04

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Legal Events

Date Code Title Description
MM4A Patent lapsed due to non-payment of maintenance fees

Effective date: 20140709