SK284979B6 - Derivát tienopyrimidínu, jeho použitie a farmaceutický prostriedok, ktorý ho obsahuje - Google Patents

Derivát tienopyrimidínu, jeho použitie a farmaceutický prostriedok, ktorý ho obsahuje Download PDF

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Publication number
SK284979B6
SK284979B6 SK502-99A SK50299A SK284979B6 SK 284979 B6 SK284979 B6 SK 284979B6 SK 50299 A SK50299 A SK 50299A SK 284979 B6 SK284979 B6 SK 284979B6
Authority
SK
Slovakia
Prior art keywords
pyrimidin
chloro
benzoic acid
thieno
pyrimidine
Prior art date
Application number
SK502-99A
Other languages
English (en)
Slovak (sk)
Other versions
SK50299A3 (en
Inventor
Rochus Jonas
Pierre Schelling
Maria Christadler
Franz-Werner Kluxen
Original Assignee
Merck Patent Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck Patent Gmbh filed Critical Merck Patent Gmbh
Publication of SK50299A3 publication Critical patent/SK50299A3/sk
Publication of SK284979B6 publication Critical patent/SK284979B6/sk

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/10—Drugs for genital or sexual disorders; Contraceptives for impotence
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure

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  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Hospice & Palliative Care (AREA)
  • Gynecology & Obstetrics (AREA)
  • Endocrinology (AREA)
  • Reproductive Health (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
SK502-99A 1996-10-24 1997-10-08 Derivát tienopyrimidínu, jeho použitie a farmaceutický prostriedok, ktorý ho obsahuje SK284979B6 (sk)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE19644228A DE19644228A1 (de) 1996-10-24 1996-10-24 Thienopyrimidine
PCT/EP1997/005530 WO1998017668A1 (de) 1996-10-24 1997-10-08 Thienopyrimidine mit pde v inhibierender wirkung

Publications (2)

Publication Number Publication Date
SK50299A3 SK50299A3 (en) 2000-03-13
SK284979B6 true SK284979B6 (sk) 2006-03-02

Family

ID=7809880

Family Applications (1)

Application Number Title Priority Date Filing Date
SK502-99A SK284979B6 (sk) 1996-10-24 1997-10-08 Derivát tienopyrimidínu, jeho použitie a farmaceutický prostriedok, ktorý ho obsahuje

Country Status (24)

Country Link
US (1) US6130223A (ru)
EP (1) EP0934321B1 (ru)
JP (1) JP2001502342A (ru)
KR (1) KR100488429B1 (ru)
CN (1) CN1105116C (ru)
AR (1) AR008504A1 (ru)
AT (1) ATE246689T1 (ru)
AU (1) AU726639B2 (ru)
BR (1) BR9712652A (ru)
CA (1) CA2269815C (ru)
CZ (1) CZ294027B6 (ru)
DE (2) DE19644228A1 (ru)
DK (1) DK0934321T3 (ru)
ES (1) ES2201275T3 (ru)
HK (1) HK1024484A1 (ru)
HU (1) HUP9904680A3 (ru)
NO (1) NO991951L (ru)
PL (1) PL192163B1 (ru)
PT (1) PT934321E (ru)
RU (1) RU2197492C2 (ru)
SK (1) SK284979B6 (ru)
TW (1) TW457242B (ru)
WO (1) WO1998017668A1 (ru)
ZA (1) ZA979516B (ru)

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US6369092B1 (en) 1998-11-23 2002-04-09 Cell Pathways, Inc. Method for treating neoplasia by exposure to substituted benzimidazole derivatives
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US6077842A (en) * 1998-11-24 2000-06-20 Cell Pathways, Inc. Method of inhibiting neoplastic cells with pyrazolopyridylpyridazinone derivatives
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Also Published As

Publication number Publication date
DK0934321T3 (da) 2003-11-03
CA2269815A1 (en) 1998-04-30
JP2001502342A (ja) 2001-02-20
EP0934321B1 (de) 2003-08-06
DE59710547D1 (de) 2003-09-11
NO991951D0 (no) 1999-04-23
PT934321E (pt) 2003-12-31
AU4945097A (en) 1998-05-15
DE19644228A1 (de) 1998-04-30
NO991951L (no) 1999-06-17
KR100488429B1 (ko) 2005-05-10
CZ142299A3 (cs) 1999-07-14
BR9712652A (pt) 1999-10-26
AU726639B2 (en) 2000-11-16
HK1024484A1 (en) 2000-10-13
EP0934321A1 (de) 1999-08-11
HUP9904680A3 (en) 2001-11-28
WO1998017668A1 (de) 1998-04-30
ES2201275T3 (es) 2004-03-16
PL192163B1 (pl) 2006-09-29
SK50299A3 (en) 2000-03-13
CN1240450A (zh) 2000-01-05
PL332970A1 (en) 1999-10-25
ZA979516B (en) 1998-05-12
RU2197492C2 (ru) 2003-01-27
TW457242B (en) 2001-10-01
CN1105116C (zh) 2003-04-09
ATE246689T1 (de) 2003-08-15
KR20000052772A (ko) 2000-08-25
HUP9904680A2 (hu) 2000-05-28
CA2269815C (en) 2007-09-25
CZ294027B6 (cs) 2004-09-15
US6130223A (en) 2000-10-10
AR008504A1 (es) 2000-01-19

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