SK278567B6 - Pharmaceutical composition consists of the pellets containing tetracycline compound - Google Patents

Pharmaceutical composition consists of the pellets containing tetracycline compound Download PDF

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Publication number
SK278567B6
SK278567B6 SK6563-88A SK656388A SK278567B6 SK 278567 B6 SK278567 B6 SK 278567B6 SK 656388 A SK656388 A SK 656388A SK 278567 B6 SK278567 B6 SK 278567B6
Authority
SK
Slovakia
Prior art keywords
deoxy
demethyltetracycline
compound
alkylamino
carbon atoms
Prior art date
Application number
SK6563-88A
Other languages
English (en)
Slovak (sk)
Other versions
SK656388A3 (en
Inventor
Joseph J Valerose Jr
Raymond J Biehl
Nitin V Sheth
Walter A Strathy
Michael K Doelling
Original Assignee
Valerose Joseph J. Jr.
Biehl Raymond J.
Sheth Nitin V.
Strathy Walter A.
Doelling Michael K.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=22303124&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=SK278567(B6) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Valerose Joseph J. Jr., Biehl Raymond J., Sheth Nitin V., Strathy Walter A., Doelling Michael K. filed Critical Valerose Joseph J. Jr.
Publication of SK278567B6 publication Critical patent/SK278567B6/sk
Publication of SK656388A3 publication Critical patent/SK656388A3/sk

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/65—Tetracyclines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1605—Excipients; Inactive ingredients
    • A61K9/1629—Organic macromolecular compounds
    • A61K9/1652—Polysaccharides, e.g. alginate, cellulose derivatives; Cyclodextrin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5073—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings
    • A61K9/5078—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings with drug-free core
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Epidemiology (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
SK6563-88A 1987-10-06 1988-10-03 Pharmaceutical preparation consisting of granules with tetracycline compound SK656388A3 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US07/104,917 US4837030A (en) 1987-10-06 1987-10-06 Novel controlled release formulations of tetracycline compounds

Publications (2)

Publication Number Publication Date
SK278567B6 true SK278567B6 (en) 1997-10-08
SK656388A3 SK656388A3 (en) 1997-10-08

Family

ID=22303124

Family Applications (1)

Application Number Title Priority Date Filing Date
SK6563-88A SK656388A3 (en) 1987-10-06 1988-10-03 Pharmaceutical preparation consisting of granules with tetracycline compound

Country Status (24)

Country Link
US (1) US4837030A (ja)
EP (1) EP0310814B1 (ja)
JP (1) JP2771189B2 (ja)
KR (1) KR970007902B1 (ja)
AR (1) AR243077A1 (ja)
AT (1) ATE120957T1 (ja)
AU (1) AU609525B2 (ja)
CA (1) CA1338439C (ja)
CZ (1) CZ279809B6 (ja)
DE (1) DE3853566T2 (ja)
DK (1) DK175578B1 (ja)
ES (1) ES2070837T3 (ja)
FI (1) FI97862C (ja)
GR (1) GR3015767T3 (ja)
HK (1) HK1000313A1 (ja)
HU (1) HU202110B (ja)
IL (1) IL87699A (ja)
NO (1) NO175619C (ja)
NZ (1) NZ226396A (ja)
PH (1) PH27236A (ja)
PL (1) PL275089A1 (ja)
PT (1) PT88664B (ja)
SK (1) SK656388A3 (ja)
ZA (1) ZA887478B (ja)

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DE3887179T2 (de) * 1987-03-02 1994-06-16 Brocades Pharma Bv Pharmazeutische Zusammensetzung, pharmazeutisches Granulat und Verfahren zu ihrer Herstellung.
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US5277916A (en) * 1988-02-01 1994-01-11 F. H. Faulding & Co., Ltd. Tetracycline dosage form
DE68916983T2 (de) * 1988-02-25 1995-01-19 Yamanouchi Europ Bv Verfahren zur Herstellung eines pharmazeutischen Granulats.
EP0418596A3 (en) * 1989-09-21 1991-10-23 American Cyanamid Company Controlled release pharmaceutical compositions from spherical granules in tabletted oral dosage unit form
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US5460825A (en) * 1990-05-23 1995-10-24 Mcneil-Ppc, Inc. Taste mask coatings for preparing chewable pharmaceutical tablets
US5260072A (en) * 1990-08-30 1993-11-09 Mcneil-Ppc, Inc. Rotogranulations and taste masking coatings for preparation of chewable pharmaceutical tablets
USRE40183E1 (en) 1991-10-04 2008-03-25 Wyeth Holdings Corporation 7-Substituted-9-substituted amino-6-demethyl-6-deoxytetracyclines
US5494903A (en) 1991-10-04 1996-02-27 American Cyanamid Company 7-substituted-9-substituted amino-6-demethyl-6-deoxytetracyclines
DE69231499T2 (de) * 1991-12-30 2001-05-03 Fmc Corp Zusammensetzung auf der basis von mikrokristalliner zellulose für die herstellung von kugelförmigen teilchen
US5262173A (en) * 1992-03-02 1993-11-16 American Cyanamid Company Pulsatile once-a-day delivery systems for minocycline
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US20060068017A1 (en) * 1996-03-25 2006-03-30 Wyeth Extended release formulation
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AU2002256092C1 (en) * 2001-04-05 2009-10-15 Collagenex Pharmaceuticals, Inc. Controlled delivery of tetracycline compounds and tetracycline derivatives
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US6958161B2 (en) * 2002-04-12 2005-10-25 F H Faulding & Co Limited Modified release coated drug preparation
AUPS167602A0 (en) * 2002-04-12 2002-05-16 F.H. Faulding & Co. Limited An improved modified release preparation
AU2003213876B2 (en) * 2002-04-12 2006-10-12 Mayne Pharma International Pty Ltd An improved modified release preparation
MXPA05004648A (es) * 2002-10-30 2005-06-08 Pharmacia Corp Comprimidos orales de liberacion extendida y procedimientos de preparacion y uso de los mismos.
US20040158194A1 (en) * 2003-02-06 2004-08-12 Wolff Andy And Beiski Ben Z. Oral devices and methods for controlled drug release
DK1615622T3 (da) * 2003-04-07 2012-10-15 Supernus Pharmaceuticals Inc Doxycyclinpræparater til indgivelse én gang dagligt
GB2414668B (en) * 2004-06-03 2009-07-29 Dexcel Ltd Tetracycline modified release delivery system
SG158869A1 (en) * 2005-01-21 2010-02-26 Warner Chilcott Co Llc A tetracycline metal complex in a solid dosage form
CN101115409B (zh) * 2005-02-04 2013-03-27 菲利普莫里斯生产公司 具有纤维质滋味添加剂的香烟及过滤嘴
US20070106138A1 (en) * 2005-05-26 2007-05-10 Beiski Ben Z Intraoral apparatus for non-invasive blood and saliva monitoring & sensing
US7544373B2 (en) * 2007-04-02 2009-06-09 Medicis Pharmaceutical Corporation Minocycline oral dosage forms for the treatment of acne
US7919483B2 (en) * 2005-06-24 2011-04-05 Medicis Pharmaceutical Corporation Method for the treatment of acne
US8722650B1 (en) 2005-06-24 2014-05-13 Medicis Pharmaceutical Corporation Extended-release minocycline dosage forms
US20080242642A1 (en) * 2007-04-02 2008-10-02 Medicis Pharmaceutical Corporation Minocycline oral dosage forms for the treatment of acne
US20080241235A1 (en) * 2007-04-02 2008-10-02 Medicis Pharmaceutical Corporation Minocycline oral dosage forms for the treatment of acne
US7541347B2 (en) * 2007-04-02 2009-06-02 Medicis Pharmaceutical Coropration Minocycline oral dosage forms for the treatment of acne
US8252776B2 (en) 2007-04-02 2012-08-28 Medicis Pharmaceutical Corporation Minocycline oral dosage forms for the treatment of acne
EP1965770A2 (en) * 2005-12-22 2008-09-10 Wyeth a Corporation of the State of Delaware Oral formulations comprising tigecycline
US20070166273A1 (en) * 2006-01-19 2007-07-19 Krivulka Joseph J Skin treatment educational kit
JP5527921B2 (ja) * 2006-12-22 2014-06-25 エスエス製薬株式会社 苦味を隠蔽した経口固形組成物
ITMI20070022A1 (it) 2007-01-09 2008-07-10 I P S Internat Products & Services Srl Formulazione di prodotti solidi a rilascio controllato per uso orale in bustine monodose e relativo procedimento di preparazione
CN102688492A (zh) * 2007-03-23 2012-09-26 分子研究中心公司 包含四环素类的抗炎组合物及其用途
US20080241197A1 (en) * 2007-04-02 2008-10-02 Medicis Pharmaceutical Corporation Minocycline dosage forms for the treatment of acne
PT2271348T (pt) * 2008-03-28 2018-04-16 Paratek Pharm Innc Formulação de comprimido oral de composto de tetraciclina
WO2010017310A1 (en) * 2008-08-06 2010-02-11 Medicis Pharmaceutical Corporation Method for the treatment of acne and certain dosage forms thereof
US9561241B1 (en) 2011-06-28 2017-02-07 Medicis Pharmaceutical Corporation Gastroretentive dosage forms for minocycline
JP6077555B2 (ja) * 2012-02-15 2017-02-08 武田薬品工業株式会社 錠剤
AU2014227598B2 (en) 2013-03-15 2018-12-06 Braintree Laboratories, Inc. Dual use oral pharmaceutical composition tablets of sulfate salts and methods of use thereof
US20170182070A1 (en) 2014-10-08 2017-06-29 Mayne Pharma International Pty Ltd. Controlled Release Doxycycline
US11103517B2 (en) 2015-04-07 2021-08-31 Dr. Reddy's Laboratories Ltd. Pharmaceutical compositions for minocycline

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CH434240A (de) * 1965-12-30 1967-04-30 Chemical And Pharmaceutical Pa Verfahren zur Herstellung einer therapeutischen Tetracyclinzubereitung mit verlängerter therapeutischer Wirkung
CH434571A (de) * 1966-07-05 1967-04-30 Chemical And Pharmaceutical Pa Verfahren zur Herstellung von Antibiotika mit verlängerter therapeutischer Wirkung
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Also Published As

Publication number Publication date
KR890006242A (ko) 1989-06-12
PL275089A1 (en) 1989-07-10
NZ226396A (en) 1991-08-27
AU609525B2 (en) 1991-05-02
GR3015767T3 (en) 1995-07-31
IL87699A (en) 1994-06-24
ES2070837T3 (es) 1995-06-16
FI97862C (fi) 1997-03-10
HUT50046A (en) 1989-12-28
NO884408D0 (no) 1988-10-05
ATE120957T1 (de) 1995-04-15
HK1000313A1 (en) 1998-02-27
DE3853566D1 (de) 1995-05-18
NO884408L (no) 1989-04-07
DK556788A (da) 1989-04-07
KR970007902B1 (ko) 1997-05-17
FI884575A (fi) 1989-04-07
JPH01128929A (ja) 1989-05-22
HU202110B (en) 1991-02-28
ZA887478B (en) 1989-06-28
CZ279809B6 (cs) 1995-07-12
EP0310814A3 (en) 1989-05-03
NO175619C (no) 1994-11-09
EP0310814A2 (en) 1989-04-12
DK556788D0 (da) 1988-10-05
FI884575A0 (fi) 1988-10-05
AU2344488A (en) 1989-04-06
DK175578B1 (da) 2004-12-13
PT88664A (pt) 1989-07-31
US4837030A (en) 1989-06-06
NO175619B (ja) 1994-08-01
CA1338439C (en) 1996-07-09
PT88664B (pt) 2003-06-30
EP0310814B1 (en) 1995-04-12
DE3853566T2 (de) 1996-01-11
CZ656388A3 (en) 1995-02-15
AR243077A1 (es) 1993-07-30
PH27236A (en) 1993-05-04
IL87699A0 (en) 1989-02-28
SK656388A3 (en) 1997-10-08
FI97862B (fi) 1996-11-29
JP2771189B2 (ja) 1998-07-02

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