SK186599A3 - 2-substituted 4,5-diaryl imidazoles, process for their preparation, pharmaceutical composition containing them and their use - Google Patents

2-substituted 4,5-diaryl imidazoles, process for their preparation, pharmaceutical composition containing them and their use Download PDF

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Publication number
SK186599A3
SK186599A3 SK1865-99A SK186599A SK186599A3 SK 186599 A3 SK186599 A3 SK 186599A3 SK 186599 A SK186599 A SK 186599A SK 186599 A3 SK186599 A3 SK 186599A3
Authority
SK
Slovakia
Prior art keywords
group
carbon atoms
pyridyl
fluorophenyl
imidazole
Prior art date
Application number
SK1865-99A
Other languages
English (en)
Slovak (sk)
Inventor
Laszlo Revesz
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of SK186599A3 publication Critical patent/SK186599A3/sk

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D451/00—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof
    • C07D451/02—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
    • A61P19/10—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic System
    • C07F7/02—Silicon compounds
    • C07F7/08—Compounds having one or more C—Si linkages
    • C07F7/0803—Compounds with Si-C or Si-Si linkages
    • C07F7/081—Compounds with Si-C or Si-Si linkages comprising at least one atom selected from the elements N, O, halogen, S, Se or Te
    • C07F7/0812—Compounds with Si-C or Si-Si linkages comprising at least one atom selected from the elements N, O, halogen, S, Se or Te comprising a heterocyclic ring
SK1865-99A 1997-06-30 1998-06-26 2-substituted 4,5-diaryl imidazoles, process for their preparation, pharmaceutical composition containing them and their use SK186599A3 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB9713726.9A GB9713726D0 (en) 1997-06-30 1997-06-30 Organic compounds
PCT/EP1998/003930 WO1999001449A1 (en) 1997-06-30 1998-06-26 2-substituted 4,5-diaryl imidazoles

Publications (1)

Publication Number Publication Date
SK186599A3 true SK186599A3 (en) 2000-06-12

Family

ID=10815101

Family Applications (1)

Application Number Title Priority Date Filing Date
SK1865-99A SK186599A3 (en) 1997-06-30 1998-06-26 2-substituted 4,5-diaryl imidazoles, process for their preparation, pharmaceutical composition containing them and their use

Country Status (28)

Country Link
US (1) US6300347B1 (de)
EP (2) EP1396491A3 (de)
JP (1) JP3704362B2 (de)
KR (1) KR20010013215A (de)
CN (1) CN1261885A (de)
AR (1) AR014886A1 (de)
AT (1) ATE275557T1 (de)
AU (1) AU744411B2 (de)
BR (1) BR9810955A (de)
CA (1) CA2291758A1 (de)
CO (1) CO4940462A1 (de)
DE (1) DE69826127T2 (de)
ES (1) ES2226164T3 (de)
GB (1) GB9713726D0 (de)
HU (1) HUP0003351A3 (de)
ID (1) ID23385A (de)
IL (1) IL133034A0 (de)
NO (1) NO996429L (de)
NZ (1) NZ501275A (de)
PE (1) PE99999A1 (de)
PL (1) PL337057A1 (de)
PT (1) PT993456E (de)
RU (1) RU2214408C2 (de)
SK (1) SK186599A3 (de)
TR (1) TR199903278T2 (de)
TW (1) TW429258B (de)
WO (1) WO1999001449A1 (de)
ZA (1) ZA985656B (de)

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Also Published As

Publication number Publication date
EP0993456B1 (de) 2004-09-08
JP2001506280A (ja) 2001-05-15
HUP0003351A2 (hu) 2001-06-28
PE99999A1 (es) 1999-11-01
NO996429D0 (no) 1999-12-23
BR9810955A (pt) 2000-09-26
DE69826127T2 (de) 2005-09-29
EP1396491A2 (de) 2004-03-10
CN1261885A (zh) 2000-08-02
AU8801598A (en) 1999-01-25
ID23385A (id) 2000-04-20
RU2214408C2 (ru) 2003-10-20
ATE275557T1 (de) 2004-09-15
PL337057A1 (en) 2000-07-31
AU744411B2 (en) 2002-02-21
KR20010013215A (ko) 2001-02-26
EP1396491A3 (de) 2004-06-30
JP3704362B2 (ja) 2005-10-12
TR199903278T2 (en) 2000-07-21
CO4940462A1 (es) 2000-07-24
HUP0003351A3 (en) 2002-01-28
US6300347B1 (en) 2001-10-09
PT993456E (pt) 2005-01-31
IL133034A0 (en) 2001-03-19
AR014886A1 (es) 2001-04-11
GB9713726D0 (en) 1997-09-03
NO996429L (no) 1999-12-23
ZA985656B (en) 1998-12-30
NZ501275A (en) 2002-04-26
CA2291758A1 (en) 1999-01-14
ES2226164T3 (es) 2005-03-16
DE69826127D1 (de) 2004-10-14
WO1999001449A1 (en) 1999-01-14
EP0993456A1 (de) 2000-04-19
TW429258B (en) 2001-04-11

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