SK156995A3 - Method for preparation of oxazolidinecarboxylic acid useful for preparation therapeutically active taxoids - Google Patents

Method for preparation of oxazolidinecarboxylic acid useful for preparation therapeutically active taxoids Download PDF

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Publication number
SK156995A3
SK156995A3 SK1569-95A SK156995A SK156995A3 SK 156995 A3 SK156995 A3 SK 156995A3 SK 156995 A SK156995 A SK 156995A SK 156995 A3 SK156995 A3 SK 156995A3
Authority
SK
Slovakia
Prior art keywords
group
carbon atoms
tert
optionally substituted
alkyl
Prior art date
Application number
SK1569-95A
Other languages
English (en)
Slovak (sk)
Inventor
Jean-Dominique Bourzat
Alain Commercon
Original Assignee
Rhone Poulenc Rorer Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Rhone Poulenc Rorer Sa filed Critical Rhone Poulenc Rorer Sa
Publication of SK156995A3 publication Critical patent/SK156995A3/sk

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
    • C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
    • C07D263/04—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D305/00—Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms
    • C07D305/14—Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms condensed with carbocyclic rings or ring systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Epoxy Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
SK1569-95A 1993-06-16 1994-06-15 Method for preparation of oxazolidinecarboxylic acid useful for preparation therapeutically active taxoids SK156995A3 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR9307240A FR2706457B1 (fr) 1993-06-16 1993-06-16 Procédé de préparation d'un acide oxazolidinecarboxylique utile pour préparer des taxoïdes thérapeutiquement actifs.
PCT/FR1994/000713 WO1994029284A1 (fr) 1993-06-16 1994-06-15 Procede de preparation d'un acide oxazolidinecarboxylique utile pour preparer des taxoides therapeutiquement actifs

Publications (1)

Publication Number Publication Date
SK156995A3 true SK156995A3 (en) 1996-06-05

Family

ID=9448182

Family Applications (1)

Application Number Title Priority Date Filing Date
SK1569-95A SK156995A3 (en) 1993-06-16 1994-06-15 Method for preparation of oxazolidinecarboxylic acid useful for preparation therapeutically active taxoids

Country Status (23)

Country Link
US (2) US6444825B1 (de)
EP (1) EP0703907B1 (de)
JP (1) JPH09500370A (de)
KR (1) KR960703118A (de)
AT (1) ATE156819T1 (de)
AU (1) AU678585B2 (de)
CA (1) CA2165328A1 (de)
CZ (1) CZ284051B6 (de)
DE (1) DE69404991T2 (de)
DK (1) DK0703907T3 (de)
ES (1) ES2107237T3 (de)
FI (1) FI956025A (de)
FR (1) FR2706457B1 (de)
GR (1) GR3024534T3 (de)
HU (1) HUT73972A (de)
NO (1) NO955112L (de)
NZ (1) NZ268037A (de)
PL (1) PL312212A1 (de)
RU (1) RU2128652C1 (de)
SK (1) SK156995A3 (de)
WO (1) WO1994029284A1 (de)
YU (1) YU37594A (de)
ZA (1) ZA943994B (de)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5973160A (en) 1992-12-23 1999-10-26 Poss; Michael A. Methods for the preparation of novel sidechain-bearing taxanes
CA2170661A1 (en) 1995-03-22 1996-09-23 John K. Thottathil Novel methods for the preparation of taxanes using oaxzolidine intermediates
KR20000010861A (ko) * 1996-05-08 2000-02-25 로렌스 티. 마이젠헬더 탁솔의 제조 방법
KR100225535B1 (ko) * 1996-08-27 1999-10-15 정지석 파클리탁셀의 제조방법
CA2422964A1 (en) 2000-09-22 2002-03-28 Bristol Myers Squibb Company Method for reducing toxicity of combined chemotherapies
US8338617B2 (en) * 2004-11-19 2012-12-25 Dr. Reddy's Laboratories Limited Process for preparing oxazolidine derivatives
CA2599888C (en) 2005-03-31 2010-06-15 Bioxel Pharma Inc. Preparation of taxanes from 9-dihydro-13-acetylbaccatin iii

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4240987A (en) * 1979-10-29 1980-12-23 Xerox Corporation Chemical process
FR2629819B1 (fr) * 1988-04-06 1990-11-16 Rhone Poulenc Sante Procede de preparation de derives de la baccatine iii et de la desacetyl-10 baccatine iii
MX9102128A (es) * 1990-11-23 1992-07-08 Rhone Poulenc Rorer Sa Derivados de taxano,procedimiento para su preparacion y composicion farmaceutica que los contiene
FR2696460B1 (fr) * 1992-10-05 1994-11-25 Rhone Poulenc Rorer Sa Procédé de préparation de dérivés du taxane.
FR2696459B1 (fr) * 1992-10-05 1994-11-25 Rhone Poulenc Rorer Sa Procédé de préparation de dérivés du taxane.
FR2696458B1 (fr) * 1992-10-05 1994-11-10 Rhone Poulenc Rorer Sa Procédé de préparation de dérivés du taxane.
FR2698361B1 (fr) * 1992-11-20 1995-01-13 Rhone Poulenc Rorer Sa Procédé de préparation d'un acide oxazolidine-1,3 carboxylique-5.
FR2698871B1 (fr) * 1992-12-09 1995-02-24 Rhone Poulenc Rorer Sa Nouveau taxoïdes, leur préparation et les compositions pharmaceutiques qui les contiennent.
FR2702212B1 (fr) * 1993-03-02 1995-04-07 Rhone Poulenc Rorer Sa Nouveaux taxoïdes, leur préparation et les compositions pharmaceutiques qui les contiennent.

Also Published As

Publication number Publication date
NZ268037A (en) 1997-11-24
US6444825B1 (en) 2002-09-03
GR3024534T3 (en) 1997-12-31
FR2706457B1 (fr) 1995-07-28
NO955112D0 (no) 1995-12-15
HUT73972A (en) 1996-10-28
US6043375A (en) 2000-03-28
ES2107237T3 (es) 1997-11-16
JPH09500370A (ja) 1997-01-14
PL312212A1 (en) 1996-04-01
DK0703907T3 (da) 1998-03-23
DE69404991T2 (de) 1998-01-22
EP0703907A1 (de) 1996-04-03
RU2128652C1 (ru) 1999-04-10
ATE156819T1 (de) 1997-08-15
ZA943994B (en) 1995-02-03
CA2165328A1 (fr) 1994-12-22
KR960703118A (ko) 1996-06-19
NO955112L (no) 1995-12-15
FI956025A0 (fi) 1995-12-14
DE69404991D1 (de) 1997-09-18
FI956025A (fi) 1995-12-14
AU7076294A (en) 1995-01-03
AU678585B2 (en) 1997-06-05
CZ284051B6 (cs) 1998-07-15
WO1994029284A1 (fr) 1994-12-22
FR2706457A1 (fr) 1994-12-23
CZ329295A3 (en) 1996-03-13
YU37594A (sh) 1997-03-07
EP0703907B1 (de) 1997-08-13
HU9503611D0 (en) 1996-02-28

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