SK156995A3 - Method for preparation of oxazolidinecarboxylic acid useful for preparation therapeutically active taxoids - Google Patents
Method for preparation of oxazolidinecarboxylic acid useful for preparation therapeutically active taxoids Download PDFInfo
- Publication number
- SK156995A3 SK156995A3 SK1569-95A SK156995A SK156995A3 SK 156995 A3 SK156995 A3 SK 156995A3 SK 156995 A SK156995 A SK 156995A SK 156995 A3 SK156995 A3 SK 156995A3
- Authority
- SK
- Slovakia
- Prior art keywords
- group
- carbon atoms
- tert
- optionally substituted
- alkyl
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
- C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
- C07D263/04—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D305/00—Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms
- C07D305/14—Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms condensed with carbocyclic rings or ring systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Epoxy Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR9307240A FR2706457B1 (fr) | 1993-06-16 | 1993-06-16 | Procédé de préparation d'un acide oxazolidinecarboxylique utile pour préparer des taxoïdes thérapeutiquement actifs. |
| PCT/FR1994/000713 WO1994029284A1 (fr) | 1993-06-16 | 1994-06-15 | Procede de preparation d'un acide oxazolidinecarboxylique utile pour preparer des taxoides therapeutiquement actifs |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| SK156995A3 true SK156995A3 (en) | 1996-06-05 |
Family
ID=9448182
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| SK1569-95A SK156995A3 (en) | 1993-06-16 | 1994-06-15 | Method for preparation of oxazolidinecarboxylic acid useful for preparation therapeutically active taxoids |
Country Status (23)
| Country | Link |
|---|---|
| US (2) | US6444825B1 (de) |
| EP (1) | EP0703907B1 (de) |
| JP (1) | JPH09500370A (de) |
| KR (1) | KR960703118A (de) |
| AT (1) | ATE156819T1 (de) |
| AU (1) | AU678585B2 (de) |
| CA (1) | CA2165328A1 (de) |
| CZ (1) | CZ284051B6 (de) |
| DE (1) | DE69404991T2 (de) |
| DK (1) | DK0703907T3 (de) |
| ES (1) | ES2107237T3 (de) |
| FI (1) | FI956025A (de) |
| FR (1) | FR2706457B1 (de) |
| GR (1) | GR3024534T3 (de) |
| HU (1) | HUT73972A (de) |
| NO (1) | NO955112D0 (de) |
| NZ (1) | NZ268037A (de) |
| PL (1) | PL312212A1 (de) |
| RU (1) | RU2128652C1 (de) |
| SK (1) | SK156995A3 (de) |
| WO (1) | WO1994029284A1 (de) |
| YU (1) | YU37594A (de) |
| ZA (1) | ZA943994B (de) |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5973160A (en) | 1992-12-23 | 1999-10-26 | Poss; Michael A. | Methods for the preparation of novel sidechain-bearing taxanes |
| CA2170661A1 (en) * | 1995-03-22 | 1996-09-23 | John K. Thottathil | Novel methods for the preparation of taxanes using oaxzolidine intermediates |
| PT1114815E (pt) * | 1996-05-08 | 2005-01-31 | Upjohn Co | Processo para a preparacao de taxol |
| KR100225535B1 (ko) * | 1996-08-27 | 1999-10-15 | 정지석 | 파클리탁셀의 제조방법 |
| CZ2003837A3 (cs) | 2000-09-22 | 2004-12-15 | Bristol-Myers Squibb Company | Způsob pro snížení toxicity při kombinovaných chemoterapiích |
| US8338617B2 (en) * | 2004-11-19 | 2012-12-25 | Dr. Reddy's Laboratories Limited | Process for preparing oxazolidine derivatives |
| RS52438B (en) * | 2005-03-31 | 2013-02-28 | Accord Healthcare Inc. | PREPARATION OF 9-DIHYDRO-13-ACETYLBACCATINE TAXAN III |
Family Cites Families (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4240987A (en) * | 1979-10-29 | 1980-12-23 | Xerox Corporation | Chemical process |
| FR2629819B1 (fr) * | 1988-04-06 | 1990-11-16 | Rhone Poulenc Sante | Procede de preparation de derives de la baccatine iii et de la desacetyl-10 baccatine iii |
| MX9102128A (es) * | 1990-11-23 | 1992-07-08 | Rhone Poulenc Rorer Sa | Derivados de taxano,procedimiento para su preparacion y composicion farmaceutica que los contiene |
| FR2696460B1 (fr) * | 1992-10-05 | 1994-11-25 | Rhone Poulenc Rorer Sa | Procédé de préparation de dérivés du taxane. |
| FR2696458B1 (fr) * | 1992-10-05 | 1994-11-10 | Rhone Poulenc Rorer Sa | Procédé de préparation de dérivés du taxane. |
| FR2696459B1 (fr) * | 1992-10-05 | 1994-11-25 | Rhone Poulenc Rorer Sa | Procédé de préparation de dérivés du taxane. |
| FR2698361B1 (fr) * | 1992-11-20 | 1995-01-13 | Rhone Poulenc Rorer Sa | Procédé de préparation d'un acide oxazolidine-1,3 carboxylique-5. |
| FR2698871B1 (fr) * | 1992-12-09 | 1995-02-24 | Rhone Poulenc Rorer Sa | Nouveau taxoïdes, leur préparation et les compositions pharmaceutiques qui les contiennent. |
| FR2702212B1 (fr) * | 1993-03-02 | 1995-04-07 | Rhone Poulenc Rorer Sa | Nouveaux taxoïdes, leur préparation et les compositions pharmaceutiques qui les contiennent. |
-
1993
- 1993-06-16 FR FR9307240A patent/FR2706457B1/fr not_active Expired - Fee Related
-
1994
- 1994-06-07 ZA ZA943994A patent/ZA943994B/xx unknown
- 1994-06-15 CZ CZ953292A patent/CZ284051B6/cs unknown
- 1994-06-15 JP JP7501433A patent/JPH09500370A/ja active Pending
- 1994-06-15 CA CA002165328A patent/CA2165328A1/fr not_active Abandoned
- 1994-06-15 DK DK94919710.7T patent/DK0703907T3/da active
- 1994-06-15 HU HU9503611A patent/HUT73972A/hu unknown
- 1994-06-15 KR KR1019950705715A patent/KR960703118A/ko not_active Application Discontinuation
- 1994-06-15 US US08/564,345 patent/US6444825B1/en not_active Expired - Lifetime
- 1994-06-15 RU RU96101137A patent/RU2128652C1/ru active
- 1994-06-15 WO PCT/FR1994/000713 patent/WO1994029284A1/fr active IP Right Grant
- 1994-06-15 AU AU70762/94A patent/AU678585B2/en not_active Ceased
- 1994-06-15 ES ES94919710T patent/ES2107237T3/es not_active Expired - Lifetime
- 1994-06-15 EP EP94919710A patent/EP0703907B1/de not_active Expired - Lifetime
- 1994-06-15 PL PL94312212A patent/PL312212A1/xx unknown
- 1994-06-15 SK SK1569-95A patent/SK156995A3/sk unknown
- 1994-06-15 DE DE69404991T patent/DE69404991T2/de not_active Expired - Fee Related
- 1994-06-15 AT AT94919710T patent/ATE156819T1/de not_active IP Right Cessation
- 1994-06-15 NZ NZ268037A patent/NZ268037A/en unknown
- 1994-06-16 YU YU37594A patent/YU37594A/sh unknown
-
1995
- 1995-12-14 FI FI956025A patent/FI956025A/fi unknown
- 1995-12-15 NO NO955112A patent/NO955112D0/no unknown
-
1997
- 1997-08-26 GR GR970400040T patent/GR3024534T3/el unknown
-
1998
- 1998-04-02 US US09/053,486 patent/US6043375A/en not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| PL312212A1 (en) | 1996-04-01 |
| FI956025A0 (fi) | 1995-12-14 |
| ZA943994B (en) | 1995-02-03 |
| US6043375A (en) | 2000-03-28 |
| CZ284051B6 (cs) | 1998-07-15 |
| EP0703907A1 (de) | 1996-04-03 |
| KR960703118A (ko) | 1996-06-19 |
| NO955112L (no) | 1995-12-15 |
| WO1994029284A1 (fr) | 1994-12-22 |
| JPH09500370A (ja) | 1997-01-14 |
| ATE156819T1 (de) | 1997-08-15 |
| AU678585B2 (en) | 1997-06-05 |
| EP0703907B1 (de) | 1997-08-13 |
| CA2165328A1 (fr) | 1994-12-22 |
| NZ268037A (en) | 1997-11-24 |
| AU7076294A (en) | 1995-01-03 |
| NO955112D0 (no) | 1995-12-15 |
| HU9503611D0 (en) | 1996-02-28 |
| FR2706457B1 (fr) | 1995-07-28 |
| RU2128652C1 (ru) | 1999-04-10 |
| DK0703907T3 (da) | 1998-03-23 |
| FI956025A (fi) | 1995-12-14 |
| YU37594A (sh) | 1997-03-07 |
| ES2107237T3 (es) | 1997-11-16 |
| FR2706457A1 (fr) | 1994-12-23 |
| HUT73972A (en) | 1996-10-28 |
| DE69404991D1 (de) | 1997-09-18 |
| CZ329295A3 (en) | 1996-03-13 |
| GR3024534T3 (en) | 1997-12-31 |
| DE69404991T2 (de) | 1998-01-22 |
| US6444825B1 (en) | 2002-09-03 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| US5688977A (en) | Method for docetaxel synthesis | |
| JP3064419B2 (ja) | バッカチン▲ｉｉｉ▼及び１０−デアセチルバッカチン▲ｉｉｉ▼のエステル化のための新規な方法 | |
| RU2088578C1 (ru) | Способ получения производных баккатина iii или 10-дезацетилбаккатина iii и способ получения производных таксана | |
| JP3295879B2 (ja) | タキサン誘導体の製造方法 | |
| JPH0686441B2 (ja) | バカチン１１１および１０―デアセチルバカチン１１１の誘導体を調製する方法 | |
| JPH10291930A (ja) | 新規タキソイドを含む製薬学的組成物 | |
| IE65642B1 (en) | Process for preparing taxane derivatives new derivatives obtained and pharmaceutical compositions containing them | |
| CA2576231A1 (en) | One pot synthesis of taxane derivatives and their conversion to paclitaxel and docetaxel | |
| AU749513B2 (en) | Process for converting 9-dihydro-13-acetylbaccatin III into taxol and derivatives thereof | |
| EP0935596B1 (de) | Verfahren zur hertellung von paclitaxel | |
| RU2188198C2 (ru) | Производные таксана | |
| SK156995A3 (en) | Method for preparation of oxazolidinecarboxylic acid useful for preparation therapeutically active taxoids | |
| CA2583366C (en) | Semi-synthesis of taxane intermediates from 9-dihydro-13-acetylbaccatin iii | |
| EA000436B1 (ru) | Способ получения паклитаксела | |
| US5608102A (en) | Process for the preparation of β-phenylisoserine and its analogues | |
| CA2319043A1 (en) | Synthesis of paclitaxel baccatin iii by protecting the 7-hydroxyl using a strong base and an electrophile | |
| JP2001247594A (ja) | フラボノイド化合物の製造法 | |
| JP4068663B2 (ja) | バッカチン誘導体の選択的保護のための方法及びタキサン合成へのその適用 | |
| EP1255745A2 (de) | Synthese von wasserlöslischem 9-dihydroplacitaxel derivate aus 9-dihydro-13-acetylbacchatin iii | |
| RU2109010C1 (ru) | ПРОИЗВОДНОЕ β -ФЕНИЛИЗОСЕРИНА, СПОСОБ ЕГО СТЕРЕОСЕЛЕКТИВНОГО ПОЛУЧЕНИЯ, ИСХОДНОЕ СОЕДИНЕНИЕ ДЛЯ ЕГО ПОЛУЧЕНИЯ, СПОСОБ ПОЛУЧЕНИЯ ТАКСАНА И ПРОМЕЖУТОЧНЫЕ ПРОДУКТЫ | |
| WO2002012216A1 (en) | An improved process for the preparation of docetaxel |