SK100894A3 - Indole compounds, method of their producing, intermediates and pharmaceutical preparations on their base - Google Patents
Indole compounds, method of their producing, intermediates and pharmaceutical preparations on their base Download PDFInfo
- Publication number
- SK100894A3 SK100894A3 SK1008-94A SK100894A SK100894A3 SK 100894 A3 SK100894 A3 SK 100894A3 SK 100894 A SK100894 A SK 100894A SK 100894 A3 SK100894 A3 SK 100894A3
- Authority
- SK
- Slovakia
- Prior art keywords
- formula
- compound
- alkyl
- group
- alkoxy
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/06—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing three or more hetero rings
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Engineering & Computer Science (AREA)
- General Health & Medical Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Endocrinology (AREA)
- Dermatology (AREA)
- Urology & Nephrology (AREA)
- Reproductive Health (AREA)
- Diabetes (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Indole Compounds (AREA)
- Steroid Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB929204365A GB9204365D0 (en) | 1992-02-28 | 1992-02-28 | Indoles |
| PCT/EP1993/000380 WO1993017014A1 (en) | 1992-02-28 | 1993-02-16 | Indole derivatives as steroid 5 alpha-reductase inhibitors |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| SK100894A3 true SK100894A3 (en) | 1995-04-12 |
Family
ID=10711259
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| SK1008-94A SK100894A3 (en) | 1992-02-28 | 1994-08-24 | Indole compounds, method of their producing, intermediates and pharmaceutical preparations on their base |
Country Status (24)
| Country | Link |
|---|---|
| US (1) | US5767139A (da) |
| EP (1) | EP0628040B1 (da) |
| JP (1) | JP2540016B2 (da) |
| KR (1) | KR950700287A (da) |
| CN (1) | CN1079465A (da) |
| AT (1) | ATE164376T1 (da) |
| AU (1) | AU3497793A (da) |
| BR (1) | BR9305991A (da) |
| CA (1) | CA2117610C (da) |
| CZ (1) | CZ207794A3 (da) |
| DE (1) | DE69317651T2 (da) |
| DK (1) | DK0628040T3 (da) |
| ES (1) | ES2115053T3 (da) |
| FI (2) | FI943931A (da) |
| GB (1) | GB9204365D0 (da) |
| HR (1) | HRP930227A2 (da) |
| HU (1) | HUT71126A (da) |
| IL (1) | IL104816A0 (da) |
| MX (1) | MX9301112A (da) |
| NO (1) | NO943187L (da) |
| RU (1) | RU94042391A (da) |
| SK (1) | SK100894A3 (da) |
| WO (1) | WO1993017014A1 (da) |
| ZA (1) | ZA931383B (da) |
Families Citing this family (13)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| IL109728A0 (en) * | 1993-05-28 | 1994-08-26 | Pfizer Res & Dev | Indoles |
| ES2099007B1 (es) * | 1993-07-16 | 1997-12-01 | Pfizer Res & Dev | Derivados de indol. |
| GB9317096D0 (en) * | 1993-08-17 | 1993-09-29 | Pfizer Ltd | Indoles |
| GB9403516D0 (en) * | 1994-02-24 | 1994-04-13 | Pfizer Ltd | Indoles |
| GB9409583D0 (en) * | 1994-05-13 | 1994-07-06 | Pfizer Ltd | Indoles |
| KR100430059B1 (ko) * | 1995-04-10 | 2004-09-24 | 후지사와 야꾸힝 고교 가부시키가이샤 | cGMP-PDE억제제로서의인돌유도체 |
| WO2000007590A1 (en) * | 1998-08-03 | 2000-02-17 | Eli Lilly And Company | INDOLE sPLA2 INHIBITORS |
| FR2796279B1 (fr) | 1999-07-16 | 2001-09-21 | Oreal | Utilisation de l'acide 4,6-dimethoxy-indole 2-carboxylique ou de ses derives pour le traitement de la seborrhee |
| FR2796274B1 (fr) * | 1999-07-16 | 2001-09-21 | Oreal | Utilisation de l'acide 4,6-dimethoxy-indole 2-carboxylique ou de ses derives pour stimuler ou induire la pousse des cheveux et/ou stopper leur chute |
| UA79504C2 (en) * | 2002-11-07 | 2007-06-25 | Organon Nv | Indols for treating diseases associated with androgen receptors |
| KR20050072812A (ko) * | 2002-11-07 | 2005-07-12 | 악조 노벨 엔.브이. | 안드로겐-수용체와 관련된 질병의 치료에 효과적인 인돌 |
| TW200602317A (en) | 2004-04-23 | 2006-01-16 | Akzo Nobel Nv | Novel androgens |
| GB201102913D0 (en) | 2011-02-18 | 2011-04-06 | Univ Birmingham | Novel therapeutic |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3557142A (en) * | 1968-02-20 | 1971-01-19 | Sterling Drug Inc | 4,5,6,7-tetrahydro-indole-lower-alkanoic acids and esters |
| PH23498A (en) * | 1984-08-06 | 1989-08-16 | Sterling Drug Inc | 3-carbonyl-1-aminoalkyl-1h-indoles,composition and use thereof |
| CA2036307C (en) * | 1990-03-08 | 2002-07-09 | Susan Jean Ward | 3-arylcarbonyl-1-aminoalkyl-1h-indole-containing antiglaucoma compositions and method |
| GB9011335D0 (en) * | 1990-05-21 | 1990-07-11 | Fujisawa Pharmaceutical Co | Indolebutyric acid derivatives and process for preparation thereof |
| IL109728A0 (en) * | 1993-05-28 | 1994-08-26 | Pfizer Res & Dev | Indoles |
-
1992
- 1992-02-28 GB GB929204365A patent/GB9204365D0/en active Pending
-
1993
- 1993-02-16 HU HU9402466A patent/HUT71126A/hu unknown
- 1993-02-16 AT AT93903984T patent/ATE164376T1/de not_active IP Right Cessation
- 1993-02-16 CA CA002117610A patent/CA2117610C/en not_active Expired - Fee Related
- 1993-02-16 DE DE69317651T patent/DE69317651T2/de not_active Expired - Fee Related
- 1993-02-16 WO PCT/EP1993/000380 patent/WO1993017014A1/en active Application Filing
- 1993-02-16 RU RU94042391/04A patent/RU94042391A/ru unknown
- 1993-02-16 CZ CZ942077A patent/CZ207794A3/cs unknown
- 1993-02-16 DK DK93903984.8T patent/DK0628040T3/da active
- 1993-02-16 JP JP5514517A patent/JP2540016B2/ja not_active Expired - Fee Related
- 1993-02-16 EP EP93903984A patent/EP0628040B1/en not_active Expired - Lifetime
- 1993-02-16 ES ES93903984T patent/ES2115053T3/es not_active Expired - Lifetime
- 1993-02-16 US US08/256,734 patent/US5767139A/en not_active Expired - Fee Related
- 1993-02-16 BR BR9305991A patent/BR9305991A/pt not_active Application Discontinuation
- 1993-02-16 AU AU34977/93A patent/AU3497793A/en not_active Abandoned
- 1993-02-22 IL IL104816A patent/IL104816A0/xx unknown
- 1993-02-24 HR HR9204365.2A patent/HRP930227A2/hr not_active Application Discontinuation
- 1993-02-26 ZA ZA931383A patent/ZA931383B/xx unknown
- 1993-02-26 MX MX9301112A patent/MX9301112A/es unknown
- 1993-02-27 CN CN93103673A patent/CN1079465A/zh active Pending
-
1994
- 1994-08-24 SK SK1008-94A patent/SK100894A3/sk unknown
- 1994-08-26 FI FI943931A patent/FI943931A/fi not_active IP Right Cessation
- 1994-08-27 KR KR1019940703018A patent/KR950700287A/ko not_active Application Discontinuation
- 1994-08-29 NO NO943187A patent/NO943187L/no unknown
-
2000
- 2000-08-09 FI FI20001771A patent/FI20001771A/fi not_active IP Right Cessation
Also Published As
| Publication number | Publication date |
|---|---|
| IL104816A0 (en) | 1993-06-10 |
| EP0628040B1 (en) | 1998-03-25 |
| JP2540016B2 (ja) | 1996-10-02 |
| EP0628040A1 (en) | 1994-12-14 |
| FI943931A0 (fi) | 1994-08-26 |
| MX9301112A (es) | 1994-07-29 |
| DK0628040T3 (da) | 1998-04-27 |
| CA2117610A1 (en) | 1993-09-02 |
| ZA931383B (en) | 1994-08-26 |
| ES2115053T3 (es) | 1998-06-16 |
| RU94042391A (ru) | 1996-08-10 |
| CA2117610C (en) | 2000-07-18 |
| JPH07500347A (ja) | 1995-01-12 |
| FI20001771A (fi) | 2000-08-09 |
| NO943187D0 (no) | 1994-08-29 |
| HUT71126A (en) | 1995-11-28 |
| CN1079465A (zh) | 1993-12-15 |
| KR950700287A (ko) | 1995-01-16 |
| US5767139A (en) | 1998-06-16 |
| NO943187L (no) | 1994-09-13 |
| AU3497793A (en) | 1993-09-13 |
| WO1993017014A1 (en) | 1993-09-02 |
| HRP930227A2 (en) | 1996-10-31 |
| ATE164376T1 (de) | 1998-04-15 |
| DE69317651T2 (de) | 1998-07-09 |
| FI943931A (fi) | 1994-08-26 |
| GB9204365D0 (en) | 1992-04-08 |
| BR9305991A (pt) | 1997-10-21 |
| DE69317651D1 (en) | 1998-04-30 |
| HU9402466D0 (en) | 1994-10-28 |
| CZ207794A3 (en) | 1995-01-18 |
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