SI21655A - Sinteza optično čistega (R)-5-(2-aminopropil)-2-metoksibenzensulfonamida - Google Patents

Sinteza optično čistega (R)-5-(2-aminopropil)-2-metoksibenzensulfonamida Download PDF

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Publication number
SI21655A
SI21655A SI200300320A SI200300320A SI21655A SI 21655 A SI21655 A SI 21655A SI 200300320 A SI200300320 A SI 200300320A SI 200300320 A SI200300320 A SI 200300320A SI 21655 A SI21655 A SI 21655A
Authority
SI
Slovenia
Prior art keywords
aminopropyl
synthesis
methoxybenzenesulfonamide
tamsulosin
group
Prior art date
Application number
SI200300320A
Other languages
English (en)
Slovenian (sl)
Inventor
Barbara Mohar
Original Assignee
LEK farmacevtska dru�ba d.d.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by LEK farmacevtska dru�ba d.d. filed Critical LEK farmacevtska dru�ba d.d.
Priority to SI200300320A priority Critical patent/SI21655A/sl
Priority to AU2004309314A priority patent/AU2004309314B2/en
Priority to EP04809254A priority patent/EP1704140B1/de
Priority to CA2549604A priority patent/CA2549604C/en
Priority to PCT/SI2004/000046 priority patent/WO2005063701A1/en
Priority to RU2006127298/04A priority patent/RU2419605C2/ru
Priority to SI200431679T priority patent/SI1704140T1/sl
Priority to AT04809254T priority patent/ATE502007T1/de
Priority to CN2004800394296A priority patent/CN1902165B/zh
Priority to US10/584,369 priority patent/US7538246B2/en
Priority to JP2006546936A priority patent/JP4695095B2/ja
Priority to BRPI0418219-7A priority patent/BRPI0418219A/pt
Priority to DE602004031879T priority patent/DE602004031879D1/de
Publication of SI21655A publication Critical patent/SI21655A/sl
Priority to ZA200604812A priority patent/ZA200604812B/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C303/00—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides
    • C07C303/36—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides of amides of sulfonic acids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/08—Drugs for disorders of the urinary system of the prostate
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C303/00—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides
    • C07C303/02—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides of sulfonic acids or halides thereof
    • C07C303/04—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides of sulfonic acids or halides thereof by substitution of hydrogen atoms by sulfo or halosulfonyl groups
    • C07C303/08—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides of sulfonic acids or halides thereof by substitution of hydrogen atoms by sulfo or halosulfonyl groups by reaction with halogenosulfonic acids
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C303/00—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides
    • C07C303/36—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides of amides of sulfonic acids
    • C07C303/38—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides of amides of sulfonic acids by reaction of ammonia or amines with sulfonic acids, or with esters, anhydrides, or halides thereof
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C303/00—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides
    • C07C303/36—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides of amides of sulfonic acids
    • C07C303/40—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides of amides of sulfonic acids by reactions not involving the formation of sulfonamide groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C311/00—Amides of sulfonic acids, i.e. compounds having singly-bound oxygen atoms of sulfo groups replaced by nitrogen atoms, not being part of nitro or nitroso groups
    • C07C311/30—Sulfonamides, the carbon skeleton of the acid part being further substituted by singly-bound nitrogen atoms, not being part of nitro or nitroso groups
    • C07C311/37—Sulfonamides, the carbon skeleton of the acid part being further substituted by singly-bound nitrogen atoms, not being part of nitro or nitroso groups having the sulfur atom of at least one of the sulfonamide groups bound to a carbon atom of a six-membered aromatic ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C311/00—Amides of sulfonic acids, i.e. compounds having singly-bound oxygen atoms of sulfo groups replaced by nitrogen atoms, not being part of nitro or nitroso groups
    • C07C311/30—Sulfonamides, the carbon skeleton of the acid part being further substituted by singly-bound nitrogen atoms, not being part of nitro or nitroso groups
    • C07C311/45—Sulfonamides, the carbon skeleton of the acid part being further substituted by singly-bound nitrogen atoms, not being part of nitro or nitroso groups at least one of the singly-bound nitrogen atoms being part of any of the groups, X being a hetero atom, Y being any atom, e.g. N-acylaminosulfonamides
    • C07C311/46—Y being a hydrogen or a carbon atom

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
SI200300320A 2003-12-29 2003-12-29 Sinteza optično čistega (R)-5-(2-aminopropil)-2-metoksibenzensulfonamida SI21655A (sl)

Priority Applications (14)

Application Number Priority Date Filing Date Title
SI200300320A SI21655A (sl) 2003-12-29 2003-12-29 Sinteza optično čistega (R)-5-(2-aminopropil)-2-metoksibenzensulfonamida
AT04809254T ATE502007T1 (de) 2003-12-29 2004-12-27 Synthese von optisch reinem (r)-5-(2-aminopropyl)-2-methoxybenzolsulphonami
CN2004800394296A CN1902165B (zh) 2003-12-29 2004-12-27 光学纯(r)-5-(2-氨基丙基)-2-甲氧基苯磺酰胺的合成
CA2549604A CA2549604C (en) 2003-12-29 2004-12-27 Synthesis of optically pure (r)-5-(2-aminopropyl)-2-methoxybenzenesulphonamide
PCT/SI2004/000046 WO2005063701A1 (en) 2003-12-29 2004-12-27 Synthesis of optically pure (r)-5-(2-aminopropyl)-2-methoxybenzenesulphonamide
RU2006127298/04A RU2419605C2 (ru) 2003-12-29 2004-12-27 Синтез оптически чистого (r)-5-(2-аминопропил)-2-метоксибензолсульфонамида
SI200431679T SI1704140T1 (sl) 2003-12-29 2004-12-27 Postopek za pripravo (R)-5-(2-aminopril)-2-metoksibenzensulfonamida
AU2004309314A AU2004309314B2 (en) 2003-12-29 2004-12-27 Synthesis of optically pure (R)-5-(2-aminopropyl)-2-methoxybenzenesulphonamide
EP04809254A EP1704140B1 (de) 2003-12-29 2004-12-27 Synthese von optisch reinem (r)-5-(2-aminopropyl)-2-methoxybenzolsulphonamid
US10/584,369 US7538246B2 (en) 2003-12-29 2004-12-27 Synthesis of optically pure(r)-5-(2-amynopropyl)-2-methoxybenzenesulphonamide
JP2006546936A JP4695095B2 (ja) 2003-12-29 2004-12-27 光学的に純粋な（ｒ）−５−（２−アミノプロピル）−２−メトキシベンゼンスルホンアミドの合成
BRPI0418219-7A BRPI0418219A (pt) 2003-12-29 2004-12-27 sìntese de (r)-5-(2-aminopropil)-2-metoxibenzenossulfonamida opticamente pura
DE602004031879T DE602004031879D1 (en) 2003-12-29 2004-12-27 Synthese von optisch reinem (r)-5-(2-aminopropyl)-2-methoxybenzolsulphonamid
ZA200604812A ZA200604812B (en) 2003-12-29 2006-06-12 Synthesis of optically pure (R)-5-(2-aminopropyl)-2-methoxybenzenesulphonamide

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
SI200300320A SI21655A (sl) 2003-12-29 2003-12-29 Sinteza optično čistega (R)-5-(2-aminopropil)-2-metoksibenzensulfonamida

Publications (1)

Publication Number Publication Date
SI21655A true SI21655A (sl) 2005-06-30

Family

ID=34738130

Family Applications (2)

Application Number Title Priority Date Filing Date
SI200300320A SI21655A (sl) 2003-12-29 2003-12-29 Sinteza optično čistega (R)-5-(2-aminopropil)-2-metoksibenzensulfonamida
SI200431679T SI1704140T1 (sl) 2003-12-29 2004-12-27 Postopek za pripravo (R)-5-(2-aminopril)-2-metoksibenzensulfonamida

Family Applications After (1)

Application Number Title Priority Date Filing Date
SI200431679T SI1704140T1 (sl) 2003-12-29 2004-12-27 Postopek za pripravo (R)-5-(2-aminopril)-2-metoksibenzensulfonamida

Country Status (13)

Country Link
US (1) US7538246B2 (de)
EP (1) EP1704140B1 (de)
JP (1) JP4695095B2 (de)
CN (1) CN1902165B (de)
AT (1) ATE502007T1 (de)
AU (1) AU2004309314B2 (de)
BR (1) BRPI0418219A (de)
CA (1) CA2549604C (de)
DE (1) DE602004031879D1 (de)
RU (1) RU2419605C2 (de)
SI (2) SI21655A (de)
WO (1) WO2005063701A1 (de)
ZA (1) ZA200604812B (de)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN101284807B (zh) * 2008-06-11 2010-12-08 药源药物化学（上海）有限公司 盐酸坦索罗辛的制备方法
CN102898336B (zh) * 2012-10-16 2013-11-27 北京悦康科创医药科技有限公司 一种盐酸坦索罗辛的制备方法
JPWO2016043189A1 (ja) * 2014-09-16 2017-06-29 塩野義製薬株式会社 トリフェニルブテン誘導体の製造方法
EA039048B1 (ru) 2016-03-15 2021-11-26 Сионоги Энд Ко., Лтд. Способ получения производных феноксиэтанола
CN110156643A (zh) * 2019-06-24 2019-08-23 新乡市锦源化工有限公司 一种对乙酰氨基苯磺酰氯高效催化制备方法
CN113582947B (zh) * 2021-09-07 2023-06-20 南开大学 一种脱除胺的磺酰基保护的方法

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3860647A (en) * 1973-08-20 1975-01-14 Smithkline Corp {60 -Aminomethyl-4-hydroxy-3-sulfamyl-benzyl alcohols and 4-hydroxy-3-sulfamyl phenethylamines
JPS56110665A (en) * 1980-02-08 1981-09-01 Yamanouchi Pharmaceut Co Ltd Sulfamoyl-substituted phenetylamine derivative and its preparation
JPS62114952A (ja) * 1985-11-13 1987-05-26 Yamanouchi Pharmaceut Co Ltd 置換フエネチルアミン誘導体の製造法
JP2696363B2 (ja) * 1988-02-19 1998-01-14 北陸製薬株式会社 フェノキシエチルアミン誘導体
CZ20013848A3 (cs) 2001-10-25 2003-05-14 Léčiva, A.S. Způsob výroby (R)-(-)-5-[2-[2-(2-ethoxyfenoxy)ethylamino]propyl]-2-methoxybenzensulfonamidu

Also Published As

Publication number Publication date
BRPI0418219A (pt) 2007-04-27
RU2419605C2 (ru) 2011-05-27
RU2006127298A (ru) 2008-02-10
AU2004309314A1 (en) 2005-07-14
WO2005063701A1 (en) 2005-07-14
JP4695095B2 (ja) 2011-06-08
US7538246B2 (en) 2009-05-26
ZA200604812B (en) 2007-09-26
CA2549604A1 (en) 2005-07-14
EP1704140A1 (de) 2006-09-27
CN1902165B (zh) 2010-06-16
DE602004031879D1 (en) 2011-04-28
JP2007517796A (ja) 2007-07-05
EP1704140B1 (de) 2011-03-16
CN1902165A (zh) 2007-01-24
AU2004309314B2 (en) 2011-09-01
SI1704140T1 (sl) 2011-10-28
ATE502007T1 (de) 2011-04-15
US20070155989A1 (en) 2007-07-05
CA2549604C (en) 2012-09-18

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Effective date: 20040517

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Effective date: 20130808