SI1910403T1 - Postopek za pripravo 3-okso-pregn-4-en-21,17-karbolaktonov z oksidacijo 17-(3-hidroksipropil)-3,17-dihidroksiandrostanov brez uporabe kovine - Google Patents

Postopek za pripravo 3-okso-pregn-4-en-21,17-karbolaktonov z oksidacijo 17-(3-hidroksipropil)-3,17-dihidroksiandrostanov brez uporabe kovine

Info

Publication number
SI1910403T1
SI1910403T1 SI200632075A SI200632075A SI1910403T1 SI 1910403 T1 SI1910403 T1 SI 1910403T1 SI 200632075 A SI200632075 A SI 200632075A SI 200632075 A SI200632075 A SI 200632075A SI 1910403 T1 SI1910403 T1 SI 1910403T1
Authority
SI
Slovenia
Prior art keywords
dihydroxyandrostanes
carbolactones
pregn
ene
oxo
Prior art date
Application number
SI200632075A
Other languages
English (en)
Inventor
Carsten Seilz
Hartmut Seba
Original Assignee
Bayer Pharma AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=37434272&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=SI1910403(T1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from EP05090214.7A external-priority patent/EP1746101B2/de
Priority claimed from US11/185,984 external-priority patent/US7319154B2/en
Application filed by Bayer Pharma AG filed Critical Bayer Pharma AG
Publication of SI1910403T1 publication Critical patent/SI1910403T1/sl

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J53/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton has been modified by condensation with a carbocyclic rings or by formation of an additional ring by means of a direct link between two ring carbon atoms, including carboxyclic rings fused to the cyclopenta(a)hydrophenanthrene skeleton are included in this class
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J53/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton has been modified by condensation with a carbocyclic rings or by formation of an additional ring by means of a direct link between two ring carbon atoms, including carboxyclic rings fused to the cyclopenta(a)hydrophenanthrene skeleton are included in this class
    • C07J53/002—Carbocyclic rings fused
    • C07J53/004—3 membered carbocyclic rings
    • C07J53/008—3 membered carbocyclic rings in position 15/16

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
SI200632075A 2005-07-21 2006-07-20 Postopek za pripravo 3-okso-pregn-4-en-21,17-karbolaktonov z oksidacijo 17-(3-hidroksipropil)-3,17-dihidroksiandrostanov brez uporabe kovine SI1910403T1 (sl)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
EP05090214.7A EP1746101B2 (de) 2005-07-21 2005-07-21 Verfahren zur Herstellung von 3-Oxo-pregn-4-en-21,17-carbolactonen durch die metallfreie Oxidation von 17-(3-hydroxypropyl)-3,17-dihydroxyandrostanen
US11/185,984 US7319154B2 (en) 2005-07-21 2005-07-21 Process for the production of 3-oxo-pregn-4-ene-21, 17-carbolactones by the metal free oxidation of 17-(3-hydroxypropyl)-3, 17-dihydroxyandrostanes
EP06762786.9A EP1910403B1 (en) 2005-07-21 2006-07-20 Process for the production of 3-oxo-pregn-4-ene-21,17-carbolactones by the metal-free oxidation of 17-(3-hydroxypropyl)-3,17-dihydroxyandrostanes
PCT/EP2006/007287 WO2007009821A1 (en) 2005-07-21 2006-07-20 Process for the production of 3-oxo-pregn-4-ene-21,17-carbolactones by the metal-free oxidation of 17-(3-hydroxypropyl)-3,17-dihydroxyandrostanes

Publications (1)

Publication Number Publication Date
SI1910403T1 true SI1910403T1 (sl) 2016-08-31

Family

ID=37434272

Family Applications (2)

Application Number Title Priority Date Filing Date
SI200632075A SI1910403T1 (sl) 2005-07-21 2006-07-20 Postopek za pripravo 3-okso-pregn-4-en-21,17-karbolaktonov z oksidacijo 17-(3-hidroksipropil)-3,17-dihidroksiandrostanov brez uporabe kovine
SI200632250T SI2527356T1 (sl) 2005-07-21 2006-07-20 Postopek za pripravo 3-okso-pregn-4-en-21,17-karbolaktonov z oksidacijo 17-(3-hidroksipropil)-3,17-dihidroksiandrostanov brez uporabe kovine

Family Applications After (1)

Application Number Title Priority Date Filing Date
SI200632250T SI2527356T1 (sl) 2005-07-21 2006-07-20 Postopek za pripravo 3-okso-pregn-4-en-21,17-karbolaktonov z oksidacijo 17-(3-hidroksipropil)-3,17-dihidroksiandrostanov brez uporabe kovine

Country Status (23)

Country Link
EP (2) EP1910403B1 (sl)
KR (1) KR101410583B1 (sl)
AU (1) AU2006271885B8 (sl)
BR (1) BRPI0613679A2 (sl)
CA (1) CA2614804C (sl)
CR (1) CR9669A (sl)
DK (2) DK1910403T3 (sl)
EA (1) EA016411B1 (sl)
EC (1) ECSP088124A (sl)
ES (2) ES2663399T3 (sl)
HK (1) HK1120520A1 (sl)
HR (2) HRP20160853T1 (sl)
HU (2) HUE038504T2 (sl)
IL (1) IL188619A (sl)
LT (1) LT2527356T (sl)
MX (1) MX2008000936A (sl)
NO (1) NO344680B1 (sl)
NZ (1) NZ565247A (sl)
PL (2) PL1910403T3 (sl)
PT (2) PT1910403T (sl)
RS (2) RS54927B1 (sl)
SI (2) SI1910403T1 (sl)
WO (1) WO2007009821A1 (sl)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MX2008016571A (es) 2007-05-01 2009-03-09 Sicor Inc Proceso para preparar drospirenona y su intermediarios.
DE102007030596B3 (de) * 2007-06-28 2009-03-12 Bayer Schering Pharma Aktiengesellschaft Verfahren zur Herstellung von 17-(3-Hydroxypropyl)-17-hydroxysteroiden
ES2432063T3 (es) * 2009-06-16 2013-11-29 Crystal Pharma, S.A.U. Procedimiento para la obtención de 17-espirolactonas en esteroides
CN102040650B (zh) * 2010-10-26 2014-03-26 西安科技大学 串联反应构建甾体-6β,7β-亚甲基结构的方法
ITMI20111383A1 (it) 2011-07-25 2013-01-26 Ind Chimica Srl Processo per la preparazione di drospirenone

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4069219A (en) 1976-12-27 1978-01-17 G. D. Searle & Co. 7ξ-(Alkoxycarbonyl)-6ξ-alkyl/halo-17-hydroxy-3-oxo-17α-pregn-4-ene-21-carboxylic acid γ-lactones and corresponding 21-carboxylic acids, their salts, and esters
DE3026783C2 (de) 1980-07-11 1982-07-29 Schering Ag, 1000 Berlin Und 4619 Bergkamen Verfahren zur Herstellung von 5β-Hydroxy-δ↑6↑-steroiden
DE3042136A1 (de) 1980-11-03 1982-06-09 Schering Ag, 1000 Berlin Und 4619 Bergkamen Verfahren zur herstellung von 3 (beta), 7 (beta) -dihydroxy- (delta) (pfeil hoch)5(pfeil hoch) -steroiden
ATE15206T1 (de) 1981-09-21 1985-09-15 Schering Ag 3-beta,7-beta,15-alpha-trihydroxy-5-androsten-1 - one, ihre 3,15-trimethylessigsaeure-ester und ihre herstellung.
DE19633685C1 (de) 1996-08-12 1997-10-09 Schering Ag Verfahren zur Herstellung von Drospirenon (6beta,7beta;15 beta,16beta-Dimethyl-en-3-oxo-17alpha-pregn-4-en-21,17-carbolacton, DRSP) sowie 7alpha-(3-Hydroxy-1-propyl)-6beta,7beta;15beta, 16beta-dimethylen-5beta-androstan-3beta,5,17beta-triol (ZK 92836) und 6beta,7beta;15beta,16beta-dimethylen-5beta-hydroxy-3-oxo-17alpha-androstan-21,17-carbolacton (90965) als Zwischenprodukte des Verfahrens
EP1534732B1 (en) * 2002-08-16 2006-09-13 Pharmacia & Upjohn Company LLC 5 androsten-3-ol steroid intermediates and processes for their preparation
ITMI20040367A1 (it) * 2004-03-01 2004-06-01 Ind Chimica Srl Processo per la preparazione di drospirenone
ITMI20042338A1 (it) 2004-12-06 2005-03-06 Ind Chimica Srl Processo per la preparazione di drospirenone

Also Published As

Publication number Publication date
AU2006271885A1 (en) 2007-01-25
PL2527356T3 (pl) 2018-06-29
SI2527356T1 (sl) 2018-04-30
CA2614804C (en) 2014-09-23
HRP20180454T1 (hr) 2018-05-04
EP2527356A2 (en) 2012-11-28
RS56982B1 (sr) 2018-05-31
EP1910403B1 (en) 2016-04-27
ECSP088124A (es) 2008-02-20
HRP20160853T1 (hr) 2016-09-23
MX2008000936A (es) 2008-03-27
CR9669A (es) 2008-02-20
PT1910403T (pt) 2016-07-14
EP2527356A3 (en) 2014-04-09
ES2581735T3 (es) 2016-09-07
HUE038504T2 (hu) 2018-10-29
AU2006271885B8 (en) 2012-03-08
AU2006271885A8 (en) 2008-02-21
NZ565247A (en) 2011-02-25
CA2614804A1 (en) 2007-01-25
KR101410583B1 (ko) 2014-06-23
BRPI0613679A2 (pt) 2011-01-25
HK1120520A1 (en) 2009-04-03
EA200800326A1 (ru) 2008-08-29
WO2007009821A1 (en) 2007-01-25
RS54927B1 (sr) 2016-10-31
PT2527356T (pt) 2018-03-26
AU2006271885B2 (en) 2012-02-16
LT2527356T (lt) 2018-04-10
KR20080033428A (ko) 2008-04-16
NO344680B1 (no) 2020-03-02
HUE027858T2 (en) 2016-11-28
IL188619A (en) 2016-06-30
EA016411B1 (ru) 2012-04-30
DK1910403T3 (en) 2016-08-01
PL1910403T3 (pl) 2016-10-31
ES2663399T3 (es) 2018-04-12
NO20080894L (no) 2008-04-21
IL188619A0 (en) 2008-04-13
EP2527356B1 (en) 2018-01-03
DK2527356T3 (en) 2018-04-09
EP1910403A1 (en) 2008-04-16

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