SI0770615T1 - Process for the preparation of dihaloazolopyrimidines - Google Patents

Process for the preparation of dihaloazolopyrimidines

Info

Publication number
SI0770615T1
SI0770615T1 SI9630630T SI9630630T SI0770615T1 SI 0770615 T1 SI0770615 T1 SI 0770615T1 SI 9630630 T SI9630630 T SI 9630630T SI 9630630 T SI9630630 T SI 9630630T SI 0770615 T1 SI0770615 T1 SI 0770615T1
Authority
SI
Slovenia
Prior art keywords
dihaloazolopyrimidines
preparation
Prior art date
Application number
SI9630630T
Other languages
English (en)
Slovenian (sl)
Inventor
G�nther Krummel
Karl-Otto Stumm
Klaus-J�Rgen Pees
Peter Heinz Rudi Liers
Original Assignee
Basf Aktiengesellschaft
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Basf Aktiengesellschaft filed Critical Basf Aktiengesellschaft
Publication of SI0770615T1 publication Critical patent/SI0770615T1/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
SI9630630T 1995-10-27 1996-10-16 Process for the preparation of dihaloazolopyrimidines SI0770615T1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US802295P 1995-10-27 1995-10-27
EP96307528A EP0770615B1 (en) 1995-10-27 1996-10-16 Process for the preparation of dihaloazolopyrimidines

Publications (1)

Publication Number Publication Date
SI0770615T1 true SI0770615T1 (en) 2003-12-31

Family

ID=21729405

Family Applications (1)

Application Number Title Priority Date Filing Date
SI9630630T SI0770615T1 (en) 1995-10-27 1996-10-16 Process for the preparation of dihaloazolopyrimidines

Country Status (22)

Country Link
US (1) US5808066A (ko)
EP (1) EP0770615B1 (ko)
JP (1) JP4018182B2 (ko)
KR (1) KR100443182B1 (ko)
AR (1) AR004122A1 (ko)
AT (1) ATE243211T1 (ko)
BR (1) BR9605258A (ko)
CA (1) CA2188905C (ko)
DE (1) DE69628712T2 (ko)
DK (1) DK0770615T3 (ko)
ES (1) ES2202419T3 (ko)
HU (1) HU217773B (ko)
IL (1) IL119496A (ko)
MX (1) MX9604882A (ko)
PT (1) PT770615E (ko)
RU (1) RU2147584C1 (ko)
SG (1) SG55239A1 (ko)
SI (1) SI0770615T1 (ko)
SK (1) SK284071B6 (ko)
TR (1) TR199600792A2 (ko)
UA (1) UA48132C2 (ko)
ZA (1) ZA968957B (ko)

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US6117876A (en) 1997-04-14 2000-09-12 American Cyanamid Company Fungicidal trifluorophenyl-triazolopyrimidines
JP3423290B2 (ja) * 1998-02-11 2003-07-07 アメリカン・サイアナミド・カンパニー 殺菌剤７−アルキル−トリアゾロピリミジン
US6117865A (en) * 1998-09-10 2000-09-12 American Cyanamid Company Fungicidal trifluorophenyl-triazolopyrimidines
US6156925A (en) * 1998-09-25 2000-12-05 American Cyanamid Company Process for the preparation of halogenated phenylmaloates
US6380202B1 (en) * 1998-09-25 2002-04-30 Basf Aktiengesellschaft Fungicidal fluoro-substituted 7-heterocyclyl-triazolopyrimidines
US6242451B1 (en) * 1998-09-25 2001-06-05 Klaus-Juergen Pees Fungicidal trihalophenyl-triazolopyrimidines
US6559151B2 (en) 2000-05-08 2003-05-06 Basf Aktiengesellschaft 6-(2-trifluoromethyl-phenyl)-triazolopyrimidines
US6756379B2 (en) * 2001-07-26 2004-06-29 Taro Pharmaceutical Industries Ltd. Non-sedating barbiturate compounds as neuroprotective agents
US7683071B2 (en) * 2000-07-26 2010-03-23 Taro Pharmaceuticals Industries Ltd. Composition and method for improved bioavailability and enhanced brain delivery of 5,5-diphenyl barbituric acid
US6939873B2 (en) * 2000-07-26 2005-09-06 Taro Pharmaceuticals Industries Limited Non-sedating barbituric acid derivatives
DE10063115A1 (de) * 2000-12-18 2002-06-27 Bayer Ag Triazolopyrimidine
JP2002249492A (ja) * 2000-12-22 2002-09-06 Nippon Bayer Agrochem Co Ltd トリアゾロピリミジン類
DE10121101A1 (de) * 2001-04-27 2002-10-31 Bayer Ag Triazolopyrimidine
PL367776A1 (en) 2001-07-05 2005-03-07 Basf Aktiengesellschaft Fungicidal triazolopyrimidines, method for the production thereof and use thereof in controlling noxious fungi and agents containing said compounds
US7038047B2 (en) 2001-07-18 2006-05-02 Basf Aktiengesellschaft Substituted 6-(2-methoxyphenyl) triazolopyrimides as fungicides
BR0211427A (pt) 2001-07-26 2004-07-13 Basf Ag Compostos, processo para preparar os mesmos, composição adequada para combater fungos danosos, uso de compostos, e, processo para combater fungos danosos
ATE362933T1 (de) 2001-09-04 2007-06-15 Sumitomo Chemical Co Imidazo(1,2-a)pyrimidine und diese enthaltende fungizidzusammensetzungen
EP1490372B1 (de) 2002-03-21 2008-01-16 Basf Aktiengesellschaft Fungizide triazolopyrimidine, verfahren zu ihrer herstellung und ihre verwendung zur bekämpfung von schadpilzen sowie sie enthaltende mittel
PT1569627E (pt) 2002-12-11 2009-01-20 Taro Pharma Ind Método de tratamento de doenças do movimento utilizando derivados do ácido barbitúrico
US7419982B2 (en) * 2003-09-24 2008-09-02 Wyeth Holdings Corporation Crystalline forms of 5-chloro-6-{2,6-difluoro-4-[3-(methylamino)propoxy]phenyl}-N-[(1S)-2,2,2-trifluoro-1-methylethyl][1,2,4]triazolo[1,5-a]pyrimidin-7-amine salts
ATE398452T1 (de) * 2003-09-24 2008-07-15 Wyeth Corp 6-aryl-7-halo-imidazoä1,2-aüpyrimidine als mittel gegen krebs
CN100519559C (zh) * 2003-09-24 2009-07-29 惠氏控股公司 作为抗癌剂的6-[(经取代的)苯基]三唑并嘧啶
MY179926A (en) * 2003-12-08 2020-11-19 Wyeth Corp Process for the preparation of tubulin inhibitors
TW200533670A (en) * 2003-12-19 2005-10-16 Basf Ag 6-(aminocarbonylphenyl)triazolopyrimidines, their preparation and their use for controlling harmful fungi, and compositions comprising these compounds
DE102004007076A1 (de) * 2004-02-13 2005-08-25 Bayer Cropscience Ag Imidazolopyrimidine
KR20060130720A (ko) * 2004-03-10 2006-12-19 바스프 악티엔게젤샤프트 5,6-디알킬-7-아미노-트리아졸로피리미딘, 그의 제조 방법,그의 병원성 진균류 방제를 위한 용도 및 상기 화합물을포함하는 제제
JP5005528B2 (ja) * 2004-03-10 2012-08-22 ビーエーエスエフ ソシエタス・ヨーロピア ５，６−ジアルキル−７−アミノトリアゾロピリミジン、その調製、および有害真菌を防除するためのその使用、ならびにそれらの化合物を含む組成物
PE20060020A1 (es) * 2004-03-30 2006-03-10 Basf Ag 5-6-cicloalquil-7-amino-triazolopirimidinas para combatir hongos fitopatogenos y procedimientos para su obtencion
CA2572797A1 (en) * 2004-07-02 2006-01-12 Daniella Gutman A process for preparing 1-methoxymethyl-5,5-diphenylbarbituric acid
WO2006092413A1 (de) * 2005-03-01 2006-09-08 Basf Aktiengesellschaft 5,6-dialkyl-7-amino-azolopyrimidine, verfahren zu ihrer herstellung und ihre verwendung zur bekämpfung von schadpilzen sowie sie enthaltende mittel
TW200714602A (en) * 2005-03-01 2007-04-16 Basf Ag 5,6-dialkyl-7-aminoazolopyrimidines, their preparation and their use for controlling harmful fungi, and compositions comprising these compounds
CN101119999A (zh) * 2005-03-01 2008-02-06 巴斯福股份公司 5,6-二烷基-7-氨基唑并嘧啶、其制备方法及其在防治有害真菌中的用途以及包含这些化合物的组合物
EP1856122A2 (de) * 2005-03-02 2007-11-21 Basf Aktiengesellschaft 2-substituierte 7-amino-azolopyrimidine, verfahren zu ihrer herstellung und ihre verwendung zur bekämpfung von schadpilzen sowie sie enthaltende mittel
US20080176744A1 (en) * 2005-03-10 2008-07-24 Basf Aktiengesellschaft Use of 4-Aminopyrimidines for Controlling Harmful Fungi, Novel 4-Aminopyrimidines, Processes for Their Preparation and Compositions Comprising Them
US20080146839A1 (en) * 2005-03-18 2008-06-19 Basf Aktiengesellschaft Method for Producing 5-Halo-2,4,6-Trifluoroisophthalic Acid
US20080200675A1 (en) * 2005-06-27 2008-08-21 Basf Aktiengesellschaft Method for Production of Substituted Phenylmalonate Esters, Novel Phenylmalonate Esters and Use Thereof
US20090131708A1 (en) * 2005-06-27 2009-05-21 Basf Aktiengesellschaft Method For Production of Substituted Phenylmalonate Esters, Intermediate Compounds and The Use Thereof for production of 5, 7-dihydroxy-6-(2,4,5-trifluorophenyl)-(1,2,4)triazolo(1,5-A)pyrimidines
EP2081576A4 (en) * 2006-11-14 2010-06-30 Taro Pharmaceuticals North Ame METHOD FOR IMPROVING BIOAVAILABILITY FOR NON-EDMING BARBITURATES
JP2010515706A (ja) * 2007-01-11 2010-05-13 ビーエーエスエフ ソシエタス・ヨーロピア アリール置換縮合ピリミジンの製造方法
US8343977B2 (en) * 2009-12-30 2013-01-01 Arqule, Inc. Substituted triazolo-pyrimidine compounds

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US3907799A (en) * 1971-08-16 1975-09-23 Icn Pharmaceuticals Xanthine oxidase inhibitors
JPS5962593A (ja) * 1982-09-30 1984-04-10 Ss Pharmaceut Co Ltd ３―置換―５，７―ジクロルトリアゾロピリミジン誘導体
DE3522463A1 (de) * 1985-06-22 1987-01-02 Bayer Ag Herbizide mittel
US4910306A (en) * 1987-11-09 1990-03-20 The Dow Chemical Company Preparation of substituted 1,2,4-triazolo[1,5-a]pyrimidine-2-sulfonanilides
US4892945A (en) * 1987-12-21 1990-01-09 Ciba-Geigy Corporation Isoindoline pigments containing at least one triazolopyrimidone radical
US5006656A (en) * 1990-02-26 1991-04-09 Dowelanco Preparation of 5,7-dihydroxy-1,2,4-triazolo[1,5-a]pyrimidine-2-sulfonanilides
US5177206A (en) * 1991-10-08 1993-01-05 Dowelanco Process for the preparation of substituted N-(aryl)-1,2,4-triazolopyrimidine-2-sulfonamides
TW224044B (ko) * 1991-12-30 1994-05-21 Shell Internat Res Schappej B V
IL108731A (en) * 1993-03-04 1997-03-18 Shell Int Research 6, N-DISUBSTITUTED-£1, 2, 4| TRIAZOLO-£1, 5-a| PYRIMIDINE- 7-AMINE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS FUNGICIDES
AU681913B2 (en) * 1993-10-18 1997-09-11 Dow Agrosciences Llc Process for preparing N-(2,6-dichloro-3-methylphenyl)-5-7-dihalo(1,2,4)triazolo(1, 5A)pyrimidine-2-sulfonamide by cyclization and halo-dehydroxylation

Also Published As

Publication number Publication date
KR970021081A (ko) 1997-05-28
IL119496A0 (en) 1997-01-10
MX9604882A (es) 1997-04-30
DE69628712D1 (de) 2003-07-24
PT770615E (pt) 2003-10-31
US5808066A (en) 1998-09-15
RU2147584C1 (ru) 2000-04-20
JP4018182B2 (ja) 2007-12-05
DK0770615T3 (da) 2003-07-14
ES2202419T3 (es) 2004-04-01
EP0770615B1 (en) 2003-06-18
UA48132C2 (uk) 2002-08-15
AR004122A1 (es) 1998-09-30
DE69628712T2 (de) 2004-04-29
ZA968957B (en) 1998-04-24
SK137796A3 (en) 1997-05-07
HU217773B (hu) 2000-04-28
SK284071B6 (sk) 2004-09-08
JPH09124651A (ja) 1997-05-13
BR9605258A (pt) 1998-07-21
IL119496A (en) 2001-07-24
CA2188905C (en) 2005-12-06
ATE243211T1 (de) 2003-07-15
SG55239A1 (en) 1998-12-21
TR199600792A2 (tr) 1997-05-21
HUP9602957A2 (en) 1997-06-30
HU9602957D0 (en) 1996-12-30
KR100443182B1 (ko) 2005-04-19
HUP9602957A3 (en) 1998-01-28
CA2188905A1 (en) 1997-04-28
EP0770615A1 (en) 1997-05-02

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