SE7704739L - Antibacterial agents - Google Patents
Antibacterial agentsInfo
- Publication number
- SE7704739L SE7704739L SE7704739A SE7704739A SE7704739L SE 7704739 L SE7704739 L SE 7704739L SE 7704739 A SE7704739 A SE 7704739A SE 7704739 A SE7704739 A SE 7704739A SE 7704739 L SE7704739 L SE 7704739L
- Authority
- SE
- Sweden
- Prior art keywords
- antibacterial agents
- alpha
- cephem
- acetamido
- hydroxyphenyl
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/54—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
- A61K31/542—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame ortho- or peri-condensed with heterocyclic ring systems
- A61K31/545—Compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins, cefaclor, or cephalexine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
Landscapes
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Epidemiology (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Cephalosporin Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GB17028/76A GB1532682A (en) | 1976-04-27 | 1976-04-27 | Process for the preparation of cephadroxil |
Publications (2)
Publication Number | Publication Date |
---|---|
SE7704739L true SE7704739L (sv) | 1977-12-01 |
SE437521B SE437521B (sv) | 1985-03-04 |
Family
ID=10087928
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
SE7704739A SE437521B (sv) | 1976-04-27 | 1977-04-25 | Ett forbettrat forfarande for framstellning av 7-(d-alfa-amino-alfa-(p-hydroxifenyl)-acetamido)-3-metyl-3-cefem-4-karboxylsyra |
Country Status (26)
Country | Link |
---|---|
US (3) | US4234721A (sv) |
JP (2) | JPS6022717B2 (sv) |
AT (1) | AT350183B (sv) |
AU (1) | AU510338B2 (sv) |
BE (1) | BE853974A (sv) |
CA (1) | CA1115268A (sv) |
CH (1) | CH632270A5 (sv) |
CY (1) | CY1066A (sv) |
DE (1) | DE2718741C2 (sv) |
DK (1) | DK157026C (sv) |
ES (1) | ES458241A1 (sv) |
FI (1) | FI67704C (sv) |
FR (2) | FR2349589A1 (sv) |
GB (1) | GB1532682A (sv) |
GR (1) | GR72788B (sv) |
HK (1) | HK39780A (sv) |
IE (1) | IE44872B1 (sv) |
IT (1) | IT8049917A0 (sv) |
KE (1) | KE3064A (sv) |
LU (1) | LU77202A1 (sv) |
MY (1) | MY8100135A (sv) |
NL (1) | NL7704618A (sv) |
PH (2) | PH16581A (sv) |
SE (1) | SE437521B (sv) |
YU (2) | YU39801B (sv) |
ZA (1) | ZA772485B (sv) |
Families Citing this family (48)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
KR820001564B1 (ko) * | 1981-05-09 | 1982-09-02 | 동신제약 주식회사 | 새로운 실릴화제를 이용한 세팔로스포린 유도체의 제조방법 |
FR2555989B1 (fr) * | 1983-12-06 | 1987-02-20 | Bristol Myers Sa | Monohydrate de chlorocephadroxyle |
JPS60169486A (ja) * | 1984-02-10 | 1985-09-02 | Yamanouchi Pharmaceut Co Ltd | 7−アミノ−3−置換メチル−3−セフエム−4−カルボン酸およびその低級アルキルシリル誘導体の製造法 |
GB8714180D0 (en) * | 1987-06-17 | 1987-07-22 | Rifar Srl | Anhydrous crystalline cefadroxil |
US4962195A (en) * | 1987-04-24 | 1990-10-09 | Rifar S.R.L. | Solvate of cefadroxyl |
US4904776A (en) * | 1987-04-24 | 1990-02-27 | Rifar S.R.L. | Method for producing crystalline cefadroxil hemihydrate |
US5023331A (en) * | 1987-04-24 | 1991-06-11 | Rifar S.R.L. | Cefadroxil solvates |
US4898938A (en) * | 1987-08-03 | 1990-02-06 | Rifar S.R.L. | Method for preparing crystalline cefadroxil monohydrate |
IT1233863B (it) * | 1988-02-24 | 1992-04-21 | Opos Biochimica Srl | Procedimento per la preparazione dell'acido 7-(d(-)-alfa-amino-alfa- (p-idrossifenil)acetamido)-3-metil-3-cefem-4-carbossilico monoidrato |
US5034522A (en) * | 1988-08-02 | 1991-07-23 | Biocraft Laboratories, Inc. | Method for the production of 3-methyl cephem derivatives |
ES2063974T3 (es) * | 1989-07-10 | 1995-01-16 | Chemferm Vof | Una nueva forma estable de cefradina, un proceso para su produccion y compuestos intermedios usados en tal proceso. |
US5142043A (en) * | 1990-05-10 | 1992-08-25 | Biocraft Laboratories, Inc. | Process for preparing cephalexin monohydrate |
AT396106B (de) * | 1991-03-08 | 1993-06-25 | Biochemie Gmbh | Neues verfahren zur herstellung von 3-vinylcephalosporinverbindungen |
US6248881B1 (en) | 1991-03-08 | 2001-06-19 | Biochemie Gmbh | Intermediates and process for the production of 3-vinyl cephalosporins |
ATE201025T1 (de) | 1991-03-08 | 2001-05-15 | Biochemie Gmbh | Verfahren zur herstellung von cephalosporinen und zwischenprodukte in diesem verfahren |
CA2155322C (en) * | 1993-03-12 | 2000-02-29 | Michael J. Dunn | Crystalline ceftiofur free acid |
US5604222A (en) * | 1993-12-27 | 1997-02-18 | Lupin Laboratories, Ltd. | Method for the preparation of 2-chloro sulfinyl azetidinones |
WO1995028398A1 (en) | 1994-04-15 | 1995-10-26 | The Upjohn Company | Novel crystal forms of 1-[5-methanesulfonamidoindolyl-2-carbonyl]-4-[3-(1-methylethylamino)-2-pyridinyl]piperazine |
US5578721A (en) * | 1994-07-11 | 1996-11-26 | Lupin Laboratories Limited | Process for preparation of 3-exomethylene cepham sulfoxide esters |
US5574154A (en) * | 1994-09-29 | 1996-11-12 | Alnejma Bulk Pharmaceutical Co. A.B.P.C. | Process for the preparation of cephalosporanic compounds |
GB9423459D0 (en) * | 1994-11-21 | 1995-01-11 | Biochemie Gmbh | Silylation process |
IT1289955B1 (it) * | 1997-02-21 | 1998-10-19 | Solchem Italiana Spa | Acyclovir sale sodico biidrato e sua preparazione |
US6080427A (en) * | 1997-04-17 | 2000-06-27 | Bristol-Myers Squibb Company | Cefadroxil monohydrate tablet formulation |
IN190389B (sv) | 1999-07-14 | 2003-07-26 | Ranbaxy Lab Ltd | |
AU5418300A (en) * | 1999-07-14 | 2001-01-30 | Ranbaxy Laboratories Limited | Process for preparing crystalline cefadroxil hemihydrate from cefadroxil dimethylformamide solvate |
US6569887B2 (en) * | 2001-08-24 | 2003-05-27 | Dov Pharmaceuticals Inc. | (−)-1-(3,4-Dichlorophenyl)-3-azabicyclo[3.1.0]hexane, compositions thereof, and uses as a dopamine-reuptake |
WO2004043920A1 (en) * | 2002-11-08 | 2004-05-27 | Dov Pharmaceuticals, Inc. | Polymorphs of bicifadine hydrochloride |
US20060173064A1 (en) * | 2001-08-24 | 2006-08-03 | Lippa Arnold S | (-)-1-(3,4-Dichlorophenyl)-3-azabi cyclo[3.1.0]hexane, compositions thereof, and uses for treating alcohol-related disorders |
US7235655B2 (en) * | 2002-03-22 | 2007-06-26 | Pharmacia & Upjohn Company | Processes to prepare eplerenone |
US20080081834A1 (en) | 2002-07-31 | 2008-04-03 | Lippa Arnold S | Methods and compositions employing bicifadine for treating disability or functional impairment associated with acute pain, chronic pain, or neuropathic disorders |
US20040077849A1 (en) * | 2002-10-16 | 2004-04-22 | Orchid Chemicals & Pharmaceuticals Limited | Process for the preparation of cefadroxil |
US7842791B2 (en) * | 2002-12-19 | 2010-11-30 | Nancy Jean Britten | Dispersible pharmaceutical compositions |
US7230097B2 (en) | 2003-03-10 | 2007-06-12 | Lupin Ltd. | Process for preparation of 7-[α-Amino (4-hydroxyphenyl) acetamido]-3-substituted-3-cephem-4-carboxylic acid |
US20070072945A1 (en) * | 2004-03-31 | 2007-03-29 | Pohoreski Anton | Sulphur-containing oils for controlling plant pathogens and stimulating nutrient uptake |
US20070043100A1 (en) * | 2005-08-16 | 2007-02-22 | Hagen Eric J | Novel polymorphs of azabicyclohexane |
US20060100263A1 (en) * | 2004-11-05 | 2006-05-11 | Anthony Basile | Antipyretic compositions and methods |
PL2719384T3 (pl) | 2005-07-27 | 2019-02-28 | Otsuka America Pharmaceutical, Inc. | Nowe 1-naftylo-3-azabicyklo[3.1.0]heksany: wytwarzanie i zastosowanie do leczenia zaburzeń neuropsychiatrycznych |
US20080045725A1 (en) | 2006-04-28 | 2008-02-21 | Murry Jerry A | Process For The Synthesis of (+) And (-)-1-(3,4-Dichlorophenyl)-3-Azabicyclo[3.1.0]Hexane |
CN101448842A (zh) * | 2006-05-19 | 2009-06-03 | 帝斯曼知识产权资产管理有限公司 | 一种用于结晶头孢羟氨苄的方法 |
US8138377B2 (en) * | 2006-11-07 | 2012-03-20 | Dov Pharmaceutical, Inc. | Arylbicyclo[3.1.0]hexylamines and methods and compositions for their preparation and use |
US20080269348A1 (en) * | 2006-11-07 | 2008-10-30 | Phil Skolnick | Novel Arylbicyclo[3.1.0]Hexylamines And Methods And Compositions For Their Preparation And Use |
ES2454966T3 (es) | 2007-02-01 | 2014-04-14 | Resverlogix Corp. | Compuestos para la prevención y el tratamiento de enfermedades cardiovasculares |
US9133159B2 (en) | 2007-06-06 | 2015-09-15 | Neurovance, Inc. | 1-heteroaryl-3-azabicyclo[3.1.0]hexanes, methods for their preparation and their use as medicaments |
WO2008153937A2 (en) * | 2007-06-06 | 2008-12-18 | Dov Pharmaceutical, Inc. | Novel 1- heteroaryl-3-azabicyclo[3.1.0]hexanes, methods for their preparation and their use as medicaments |
NZ595747A (en) | 2009-03-18 | 2015-06-26 | Resverlogix Corp | Novel quinazolinones and related compounds for use as anti-inflammatory agents |
CN102408438B (zh) * | 2010-09-26 | 2015-01-07 | 石药集团中奇制药技术(石家庄)有限公司 | 一种头孢丙烯一水合物的制备方法 |
CN102134250B (zh) * | 2011-01-19 | 2013-03-13 | 天津大学 | 一种头孢羟氨苄单水合物的结晶方法及结晶 |
US20140206740A1 (en) | 2011-07-30 | 2014-07-24 | Neurovance, Inc. | Use Of (1R,5S)-(+)-(Napthalen-2-yl)-3-Azabicyclo[3.1.0]Hexane In The Treatment Of Conditions Affected By Monoamine Neurotransmitters |
Family Cites Families (18)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US29164A (en) * | 1860-07-17 | Improvement in fish-oils | ||
USRE29164E (en) | 1967-09-05 | 1977-03-29 | Bristol-Myers Company | 7-Amino-cephalosporanic and decephalosporanic acid derivatives |
CY773A (en) | 1967-09-05 | 1975-03-01 | Bristol Myers Co | Antibacterial agents and a process for the preparation thereof |
US3655656A (en) * | 1970-06-04 | 1972-04-11 | Lilly Co Eli | Crystalline cephalexin monohydrate |
US3694437A (en) * | 1970-08-19 | 1972-09-26 | Lilly Co Eli | Process for preparing cephalosporin compounds |
US3781282A (en) * | 1971-01-20 | 1973-12-25 | W Garbrecht | Cephalosporin process and product |
JPS5318515B2 (sv) | 1971-12-17 | 1978-06-15 | ||
DE2163514A1 (de) * | 1971-12-21 | 1973-07-05 | Toyama Chemical Co Ltd | Verfahren zur herstellung von cephalosporinen |
FR2166316A1 (en) * | 1972-01-07 | 1973-08-17 | Toyama Chemical Co Ltd | 7-acylcephalosporins - prepd via a silylated inter |
US3985741A (en) * | 1972-09-15 | 1976-10-12 | Bristol-Myers Company | Production of p-hydroxycephalexin |
BE806868A (fr) | 1972-11-02 | 1974-02-15 | Lorenzini Sas Inst Biochim | Procede de preparation de l'acide 7-(d-alpha-aminophenylacetamido) -3-desacetoxycephalosporanique |
GB1472746A (en) * | 1973-07-05 | 1977-05-04 | Glaxo Lab Ltd | Cephalosporin compounds |
GB1476981A (en) | 1974-06-05 | 1977-06-16 | Bristol Myers Co | Substituted penicillanic acids |
US4091215A (en) * | 1974-06-05 | 1978-05-23 | Bristol-Myers Company | 7-D-α-Amino-.alpha.-(p-acetoxyphenyl)acetamido-3-methyl-3-cephem-4-carboxylic acid |
AU2550077A (en) * | 1976-06-14 | 1978-11-30 | Merck Patent Gmbh | Penicillins and cephalosporins |
US4160863A (en) * | 1977-04-07 | 1979-07-10 | Bristol-Myers Company | Process for the preparation of the crystalline monohydrate of 7-[D-α-aα-(p-hydroxyphenyl)acetamido]-3-methyl-3-cephem-4-carboxylic acid |
NL162387C (nl) * | 1977-09-06 | 1980-05-16 | Gist Brocades Nv | Werkwijze voor het bereiden van 6-(d-alpha-amino-p- -hydroxyfenylacetamido)penicillanzuur. |
IT1126544B (it) * | 1979-12-07 | 1986-05-21 | Dobfar Spa | Procedimento per la preparazione di derivati dell'acido 7-amino-desacetossi cefalosporanico |
-
1976
- 1976-04-27 GB GB17028/76A patent/GB1532682A/en not_active Expired
-
1977
- 1977-03-07 CY CY1066A patent/CY1066A/xx unknown
- 1977-04-25 ZA ZA00772485A patent/ZA772485B/xx unknown
- 1977-04-25 SE SE7704739A patent/SE437521B/sv not_active IP Right Cessation
- 1977-04-26 IE IE835/77A patent/IE44872B1/en not_active IP Right Cessation
- 1977-04-26 FR FR7712622A patent/FR2349589A1/fr active Granted
- 1977-04-26 CA CA276,959A patent/CA1115268A/en not_active Expired
- 1977-04-26 YU YU1086/77A patent/YU39801B/xx unknown
- 1977-04-26 BE BE177035A patent/BE853974A/xx not_active IP Right Cessation
- 1977-04-26 LU LU77202A patent/LU77202A1/xx unknown
- 1977-04-26 GR GR53296A patent/GR72788B/el unknown
- 1977-04-26 DK DK183277A patent/DK157026C/da not_active IP Right Cessation
- 1977-04-26 PH PH19706A patent/PH16581A/en unknown
- 1977-04-27 JP JP52048003A patent/JPS6022717B2/ja not_active Expired
- 1977-04-27 AU AU24607/77A patent/AU510338B2/en not_active Expired
- 1977-04-27 ES ES77458241A patent/ES458241A1/es not_active Expired
- 1977-04-27 DE DE2718741A patent/DE2718741C2/de not_active Expired
- 1977-04-27 FI FI771339A patent/FI67704C/fi not_active IP Right Cessation
- 1977-04-27 AT AT296277A patent/AT350183B/de not_active IP Right Cessation
- 1977-04-27 CH CH523277A patent/CH632270A5/de not_active IP Right Cessation
- 1977-04-27 NL NL7704618A patent/NL7704618A/xx active Search and Examination
- 1977-12-22 FR FR7738820A patent/FR2365570A1/fr active Granted
-
1979
- 1979-05-21 US US06/071,951 patent/US4234721A/en not_active Expired - Lifetime
- 1979-07-27 PH PH22820A patent/PH17254A/en unknown
-
1980
- 1980-07-09 KE KE3064A patent/KE3064A/xx unknown
- 1980-07-31 HK HK397/80A patent/HK39780A/xx unknown
- 1980-10-16 IT IT8049917A patent/IT8049917A0/it unknown
-
1981
- 1981-12-31 MY MY1981135A patent/MY8100135A/xx unknown
-
1982
- 1982-03-16 US US06/358,567 patent/US4504657A/en not_active Expired - Lifetime
- 1982-06-24 YU YU1379/82A patent/YU43081B/xx unknown
- 1982-11-30 US US06/455,398 patent/USRE31730E/en not_active Expired - Lifetime
-
1985
- 1985-01-29 JP JP60013652A patent/JPS60185718A/ja active Granted
Also Published As
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SE8601963L (sv) | O-sulfaterade beta-laktamhydroxamsyror | |
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SE438151B (sv) | Ketenimin till anvendning for framstellning av antibakteriellt aktiva penicillinderivat |
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