SE437158B - Substituerade pyrido/1,2-a/pyrimidiner, forfarande for framstellning derav och farmaceutisk komposition - Google Patents

Substituerade pyrido/1,2-a/pyrimidiner, forfarande for framstellning derav och farmaceutisk komposition

Info

Publication number
SE437158B
SE437158B SE8003433A SE8003433A SE437158B SE 437158 B SE437158 B SE 437158B SE 8003433 A SE8003433 A SE 8003433A SE 8003433 A SE8003433 A SE 8003433A SE 437158 B SE437158 B SE 437158B
Authority
SE
Sweden
Prior art keywords
trans
oxo
ethenyl
carboxylic acid
pyrimidine
Prior art date
Application number
SE8003433A
Other languages
English (en)
Swedish (sv)
Other versions
SE8003433L (sv
Inventor
G Doria
C Romeo
P Sberze
M Tibolla
M L Corno
Original Assignee
Erba Farmitalia
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Erba Farmitalia filed Critical Erba Farmitalia
Publication of SE8003433L publication Critical patent/SE8003433L/xx
Publication of SE437158B publication Critical patent/SE437158B/sv

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/08—Antiepileptics; Anticonvulsants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Immunology (AREA)
  • Pulmonology (AREA)
  • Pain & Pain Management (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
SE8003433A 1979-05-08 1980-05-07 Substituerade pyrido/1,2-a/pyrimidiner, forfarande for framstellning derav och farmaceutisk komposition SE437158B (sv)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB7915810 1979-05-08

Publications (2)

Publication Number Publication Date
SE8003433L SE8003433L (sv) 1980-11-09
SE437158B true SE437158B (sv) 1985-02-11

Family

ID=10504995

Family Applications (1)

Application Number Title Priority Date Filing Date
SE8003433A SE437158B (sv) 1979-05-08 1980-05-07 Substituerade pyrido/1,2-a/pyrimidiner, forfarande for framstellning derav och farmaceutisk komposition

Country Status (28)

Country Link
US (2) US4310526A (it)
JP (1) JPS562983A (it)
AT (1) AT375370B (it)
AU (1) AU527931B2 (it)
BE (1) BE883150A (it)
CA (1) CA1134359A (it)
CH (1) CH647777A5 (it)
CS (2) CS528780A2 (it)
DE (1) DE3015738A1 (it)
DK (1) DK200280A (it)
ES (1) ES8104287A1 (it)
FI (1) FI68824C (it)
FR (1) FR2456093A1 (it)
GB (1) GB2050353B (it)
GR (1) GR68075B (it)
HU (1) HU181778B (it)
IE (1) IE49787B1 (it)
IL (1) IL59802A (it)
IT (1) IT1209326B (it)
LU (1) LU82419A1 (it)
NL (1) NL8002656A (it)
NO (1) NO153137C (it)
NZ (1) NZ193579A (it)
PH (1) PH16695A (it)
PT (1) PT71197A (it)
SE (1) SE437158B (it)
SU (2) SU1217259A3 (it)
ZA (1) ZA802390B (it)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AT377586B (de) 1981-06-30 1985-04-10 Erba Farmitalia Verfahren zur herstellung von substituierten pyrrolo-(2,1-b)-chinazolinen und pyrido(2,1-b)chinazolinen
US4537962A (en) * 1982-02-04 1985-08-27 Farmitalia Carlo Erba, S.P.A. Substituted 1,3,4-thiadiazolo[3,2-A]pyrimidines and compositions containing them
CA1211111A (en) * 1982-02-15 1986-09-09 Isao Yanagisawa Process for preparing novel pyrimidone compounds
ES8406476A1 (es) * 1982-04-29 1984-07-01 Erba Farmitalia Procedimiento para preparar derivados cicloalifaticos condensados de pirido(1,2-a)pirimidinas sustituidas.
IL69274A (en) * 1982-08-05 1986-08-31 Erba Farmitalia (substituted amino)derivatives of 3-benzylidene-pyrrolo(2,1-b)quinazolin-9-ones and 6-benzylidene-pyrido(2,1-b)quinazolin-11-ones,their preparation and pharmaceutical compositions containing them
GB8300728D0 (en) * 1983-01-12 1983-02-16 Erba Farmitalia Substituted carboxy-thiazolo / 3 2 - a / pyrimidine derivatives
US4457932A (en) * 1983-07-22 1984-07-03 Bristol-Myers Company Anti-ulcer agents
GB8501015D0 (en) * 1985-01-16 1985-02-20 Riker Laboratories Inc Drug
JP2668259B2 (ja) * 1988-02-18 1997-10-27 塩野義製薬株式会社 複素環化合物および抗潰瘍剤
MX2010005769A (es) * 2008-01-11 2010-11-12 Glenmark Pharmaceuticals Sa Derivados de pirimidina fusionados como moduladores del trpv3.

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4209622A (en) * 1973-03-30 1980-06-24 Chinoin Gygyszer es Vegyeszeti Termekek Gyara Rt. 3-(Ethoxycarbonyl-methyl)-6-methyl-4-oxo-6,7,8,9-tetrahydro-4H-pyrido[1,2-a]pyrimidine
US3935197A (en) * 1975-05-16 1976-01-27 E. R. Squibb & Sons, Inc. 2-Styryl-4H-pyrido(1,2-a)pyrimidin-4-ones
HU178910B (en) 1977-08-19 1982-07-28 Chinoin Gyogyszer Es Vegyeszet Process for preparing 2,3-disubstituted-4-oxo-4h-pyrido/1,2-a/-pyrimidines
HU180701B (en) 1977-12-29 1983-04-29 Chinoin Gyogyszer Es Vegyeszet Process for preparing pyrido-/1,2-a/pyrimidines containing a carboxylic or ester group on the pirimidimering
HU184058B (en) 1977-12-29 1984-06-28 Chinoin Gyogyszer Es Vegyeszet Process for preparing new compounds with nitrogen bridge head

Also Published As

Publication number Publication date
IT1209326B (it) 1989-07-16
GB2050353B (en) 1983-04-27
CA1134359A (en) 1982-10-26
CS321380A2 (en) 1984-12-14
FR2456093B1 (it) 1984-02-03
NL8002656A (nl) 1980-11-11
ZA802390B (en) 1981-04-29
ES491238A0 (es) 1981-04-01
IE800945L (en) 1980-11-08
SU1158045A3 (ru) 1985-05-23
CS244107B2 (en) 1986-07-17
IE49787B1 (en) 1985-12-11
GR68075B (it) 1981-10-30
NO153137B (no) 1985-10-14
IL59802A0 (en) 1980-06-30
SU1217259A3 (ru) 1986-03-07
DE3015738A1 (de) 1980-11-13
LU82419A1 (fr) 1980-07-31
DK200280A (da) 1980-11-09
GB2050353A (en) 1981-01-07
US4310526A (en) 1982-01-12
AU5731980A (en) 1980-11-13
PT71197A (en) 1980-06-01
SE8003433L (sv) 1980-11-09
JPS562983A (en) 1981-01-13
US4341780A (en) 1982-07-27
HU181778B (en) 1983-11-28
FI68824C (fi) 1985-11-11
PH16695A (en) 1984-01-06
AU527931B2 (en) 1983-03-31
FR2456093A1 (fr) 1980-12-05
IT8021821A0 (it) 1980-05-06
IL59802A (en) 1983-07-31
NZ193579A (en) 1982-09-07
NO153137C (no) 1986-01-22
FI68824B (fi) 1985-07-31
CS528780A2 (en) 1985-09-17
CH647777A5 (de) 1985-02-15
FI801464A (fi) 1980-11-09
ES8104287A1 (es) 1981-04-01
AT375370B (de) 1984-07-25
BE883150A (fr) 1980-11-07
ATA245680A (de) 1983-12-15
NO801342L (no) 1980-11-10

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