NO153137C - Analogifremgangsmaate for fremstilling av terapeutisk aktive substituerte pyrido(1,2-a)pyrimidiner. - Google Patents

Analogifremgangsmaate for fremstilling av terapeutisk aktive substituerte pyrido(1,2-a)pyrimidiner.

Info

Publication number
NO153137C
NO153137C NO801342A NO801342A NO153137C NO 153137 C NO153137 C NO 153137C NO 801342 A NO801342 A NO 801342A NO 801342 A NO801342 A NO 801342A NO 153137 C NO153137 C NO 153137C
Authority
NO
Norway
Prior art keywords
pyrimidines
preparation
therapeutic active
substituted pyrido
active substituted
Prior art date
Application number
NO801342A
Other languages
English (en)
Norwegian (no)
Other versions
NO153137B (no
NO801342L (no
Inventor
Gianfederico Doria
Ciriaco Romeo
Piero Sberze
Marcellino Tibolla
Maria Luisa Corno
Original Assignee
Erba Farmitalia
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Erba Farmitalia filed Critical Erba Farmitalia
Publication of NO801342L publication Critical patent/NO801342L/no
Publication of NO153137B publication Critical patent/NO153137B/no
Publication of NO153137C publication Critical patent/NO153137C/no

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/08Antiepileptics; Anticonvulsants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/08Antiallergic agents

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Immunology (AREA)
  • Pulmonology (AREA)
  • Pain & Pain Management (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
NO801342A 1979-05-08 1980-05-07 Analogifremgangsmaate for fremstilling av terapeutisk aktive substituerte pyrido(1,2-a)pyrimidiner. NO153137C (no)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB7915810 1979-05-08

Publications (3)

Publication Number Publication Date
NO801342L NO801342L (no) 1980-11-10
NO153137B NO153137B (no) 1985-10-14
NO153137C true NO153137C (no) 1986-01-22

Family

ID=10504995

Family Applications (1)

Application Number Title Priority Date Filing Date
NO801342A NO153137C (no) 1979-05-08 1980-05-07 Analogifremgangsmaate for fremstilling av terapeutisk aktive substituerte pyrido(1,2-a)pyrimidiner.

Country Status (28)

Country Link
US (2) US4310526A (it)
JP (1) JPS562983A (it)
AT (1) AT375370B (it)
AU (1) AU527931B2 (it)
BE (1) BE883150A (it)
CA (1) CA1134359A (it)
CH (1) CH647777A5 (it)
CS (2) CS528780A2 (it)
DE (1) DE3015738A1 (it)
DK (1) DK200280A (it)
ES (1) ES8104287A1 (it)
FI (1) FI68824C (it)
FR (1) FR2456093A1 (it)
GB (1) GB2050353B (it)
GR (1) GR68075B (it)
HU (1) HU181778B (it)
IE (1) IE49787B1 (it)
IL (1) IL59802A (it)
IT (1) IT1209326B (it)
LU (1) LU82419A1 (it)
NL (1) NL8002656A (it)
NO (1) NO153137C (it)
NZ (1) NZ193579A (it)
PH (1) PH16695A (it)
PT (1) PT71197A (it)
SE (1) SE437158B (it)
SU (2) SU1217259A3 (it)
ZA (1) ZA802390B (it)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AT377586B (de) 1981-06-30 1985-04-10 Erba Farmitalia Verfahren zur herstellung von substituierten pyrrolo-(2,1-b)-chinazolinen und pyrido(2,1-b)chinazolinen
US4537962A (en) * 1982-02-04 1985-08-27 Farmitalia Carlo Erba, S.P.A. Substituted 1,3,4-thiadiazolo[3,2-A]pyrimidines and compositions containing them
CA1211111A (en) * 1982-02-15 1986-09-09 Isao Yanagisawa Process for preparing novel pyrimidone compounds
ES8406476A1 (es) * 1982-04-29 1984-07-01 Erba Farmitalia Procedimiento para preparar derivados cicloalifaticos condensados de pirido(1,2-a)pirimidinas sustituidas.
IL69274A (en) * 1982-08-05 1986-08-31 Erba Farmitalia (substituted amino)derivatives of 3-benzylidene-pyrrolo(2,1-b)quinazolin-9-ones and 6-benzylidene-pyrido(2,1-b)quinazolin-11-ones,their preparation and pharmaceutical compositions containing them
GB8300728D0 (en) * 1983-01-12 1983-02-16 Erba Farmitalia Substituted carboxy-thiazolo / 3 2 - a / pyrimidine derivatives
US4457932A (en) * 1983-07-22 1984-07-03 Bristol-Myers Company Anti-ulcer agents
GB8501015D0 (en) * 1985-01-16 1985-02-20 Riker Laboratories Inc Drug
JP2668259B2 (ja) * 1988-02-18 1997-10-27 塩野義製薬株式会社 複素環化合物および抗潰瘍剤
MX2010005769A (es) * 2008-01-11 2010-11-12 Glenmark Pharmaceuticals Sa Derivados de pirimidina fusionados como moduladores del trpv3.

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4209622A (en) * 1973-03-30 1980-06-24 Chinoin Gygyszer es Vegyeszeti Termekek Gyara Rt. 3-(Ethoxycarbonyl-methyl)-6-methyl-4-oxo-6,7,8,9-tetrahydro-4H-pyrido[1,2-a]pyrimidine
US3935197A (en) * 1975-05-16 1976-01-27 E. R. Squibb & Sons, Inc. 2-Styryl-4H-pyrido(1,2-a)pyrimidin-4-ones
HU178910B (en) 1977-08-19 1982-07-28 Chinoin Gyogyszer Es Vegyeszet Process for preparing 2,3-disubstituted-4-oxo-4h-pyrido/1,2-a/-pyrimidines
HU180701B (en) 1977-12-29 1983-04-29 Chinoin Gyogyszer Es Vegyeszet Process for preparing pyrido-/1,2-a/pyrimidines containing a carboxylic or ester group on the pirimidimering
HU184058B (en) 1977-12-29 1984-06-28 Chinoin Gyogyszer Es Vegyeszet Process for preparing new compounds with nitrogen bridge head

Also Published As

Publication number Publication date
IT1209326B (it) 1989-07-16
GB2050353B (en) 1983-04-27
CA1134359A (en) 1982-10-26
CS321380A2 (en) 1984-12-14
FR2456093B1 (it) 1984-02-03
NL8002656A (nl) 1980-11-11
ZA802390B (en) 1981-04-29
ES491238A0 (es) 1981-04-01
IE800945L (en) 1980-11-08
SU1158045A3 (ru) 1985-05-23
CS244107B2 (en) 1986-07-17
IE49787B1 (en) 1985-12-11
GR68075B (it) 1981-10-30
NO153137B (no) 1985-10-14
IL59802A0 (en) 1980-06-30
SU1217259A3 (ru) 1986-03-07
DE3015738A1 (de) 1980-11-13
LU82419A1 (fr) 1980-07-31
DK200280A (da) 1980-11-09
GB2050353A (en) 1981-01-07
US4310526A (en) 1982-01-12
AU5731980A (en) 1980-11-13
PT71197A (en) 1980-06-01
SE8003433L (sv) 1980-11-09
JPS562983A (en) 1981-01-13
US4341780A (en) 1982-07-27
HU181778B (en) 1983-11-28
FI68824C (fi) 1985-11-11
PH16695A (en) 1984-01-06
SE437158B (sv) 1985-02-11
AU527931B2 (en) 1983-03-31
FR2456093A1 (fr) 1980-12-05
IT8021821A0 (it) 1980-05-06
IL59802A (en) 1983-07-31
NZ193579A (en) 1982-09-07
FI68824B (fi) 1985-07-31
CS528780A2 (en) 1985-09-17
CH647777A5 (de) 1985-02-15
FI801464A (fi) 1980-11-09
ES8104287A1 (es) 1981-04-01
AT375370B (de) 1984-07-25
BE883150A (fr) 1980-11-07
ATA245680A (de) 1983-12-15
NO801342L (no) 1980-11-10

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