SE405857B - Forfarande for substituerande av en grupp i 6-resp 7-stellning hos en penicillansyraforening eller cefalosporansyraforening - Google Patents

Forfarande for substituerande av en grupp i 6-resp 7-stellning hos en penicillansyraforening eller cefalosporansyraforening

Info

Publication number
SE405857B
SE405857B SE7214708A SE1470872A SE405857B SE 405857 B SE405857 B SE 405857B SE 7214708 A SE7214708 A SE 7214708A SE 1470872 A SE1470872 A SE 1470872A SE 405857 B SE405857 B SE 405857B
Authority
SE
Sweden
Prior art keywords
acid
benzyl
added
group
benzhydryl
Prior art date
Application number
SE7214708A
Other languages
English (en)
Swedish (sv)
Inventor
R A Firestone
L D Cama
B G Christensen
Original Assignee
Merck & Co Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck & Co Inc filed Critical Merck & Co Inc
Publication of SE405857B publication Critical patent/SE405857B/sv

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Cephalosporin Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
SE7214708A 1971-11-29 1972-11-13 Forfarande for substituerande av en grupp i 6-resp 7-stellning hos en penicillansyraforening eller cefalosporansyraforening SE405857B (sv)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US20305671A 1971-11-29 1971-11-29

Publications (1)

Publication Number Publication Date
SE405857B true SE405857B (sv) 1979-01-08

Family

ID=22752300

Family Applications (1)

Application Number Title Priority Date Filing Date
SE7214708A SE405857B (sv) 1971-11-29 1972-11-13 Forfarande for substituerande av en grupp i 6-resp 7-stellning hos en penicillansyraforening eller cefalosporansyraforening

Country Status (21)

Country Link
US (1) US4041029A (fi)
JP (2) JPS5850230B2 (fi)
AT (1) AT322098B (fi)
AU (1) AU470085B2 (fi)
CA (1) CA1023344A (fi)
CH (1) CH594680A5 (fi)
CS (1) CS177830B2 (fi)
DD (1) DD100955A5 (fi)
DE (1) DE2258221C2 (fi)
DK (1) DK145059C (fi)
ES (1) ES408972A1 (fi)
FI (1) FI56841C (fi)
FR (1) FR2186968A5 (fi)
GB (1) GB1401059A (fi)
HU (1) HU165582B (fi)
IE (1) IE36881B1 (fi)
NL (1) NL187633C (fi)
PL (1) PL85390B1 (fi)
SE (1) SE405857B (fi)
SU (1) SU467521A3 (fi)
YU (2) YU36181B (fi)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4447602A (en) * 1971-11-29 1984-05-08 Merck & Co., Inc. Process to prepare 7-substituted cephalosporins or 6-substituted penicillins
BE794554A (fr) * 1972-01-31 1973-07-26 Lilly Co Eli Nouveaux derives de penicilline et de cephalusporine
JPS5113788A (en) * 1974-07-24 1976-02-03 Sankyo Co Beetaaa rakutamukoseibutsushitsuno arukokishudotaino seiho
JPS5530714B2 (fi) * 1974-08-22 1980-08-13
JPS5159890A (en) * 1974-11-15 1976-05-25 Sankyo Co 77 arukokishisefuarosuhorinjudotaino seizoho
JPS5760345B2 (fi) * 1974-12-19 1982-12-18 Takeda Chemical Industries Ltd
DK154939C (da) * 1974-12-19 1989-06-12 Takeda Chemical Industries Ltd Analogifremgangsmaade til fremstilling af thiazolylacetamido-cephemforbindelser eller farmaceutisk acceptable salte eller estere deraf
GB1538051A (en) * 1975-01-17 1979-01-10 Beecham Group Ltd 6-methoxy-6-(alpha-carboxyacetamido)-penicillins
US4162251A (en) * 1976-04-05 1979-07-24 Sankyo Company Limited Process for the preparation of β-lactam compounds
JPS5321191A (en) * 1976-08-10 1978-02-27 Shionogi & Co Ltd 7-arylmalonamidocephem derivatives
JPS5630986A (en) * 1979-08-23 1981-03-28 Meiji Seika Kaisha Ltd Preparation of 7-methoxycephalosporin derivative and drug composition
NZ195030A (en) * 1979-10-09 1983-06-17 Beecham Group Ltd Preparation of 6 -methoxy-penam derivatives
DE3373475D1 (en) * 1982-12-14 1987-10-15 Beecham Group Plc Process for the preparation of beta-lactam compounds
US5455239A (en) * 1993-08-05 1995-10-03 Merck & Co. Inc. 3-aryl of heteroaryl-7-heteroaralkylamido cephalosporin compounds, compositions and methods of use
US5498777A (en) * 1994-07-20 1996-03-12 Merck & Co., Inc. 3-thioheteroaryl cephalosporin compounds, compositions and methods of use
US5565445A (en) * 1995-02-22 1996-10-15 Merck & Co., Inc. 3-thioheteroaryl 1-carba-1-dethiacephalosporin compounds, compositions and methods of use
CN102633819A (zh) * 2012-04-24 2012-08-15 齐鲁安替（临邑）制药有限公司 一种头孢西丁的制备方法
CN104230956B (zh) * 2012-04-24 2016-07-06 齐鲁安替（临邑）制药有限公司 一种头孢西丁的制备方法

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3778432A (en) * 1971-12-13 1973-12-11 Merck & Co Inc Isocyanates and carbamates of penicillins and 3-cephem-4-carboxylic acids
BE794554A (fr) * 1972-01-31 1973-07-26 Lilly Co Eli Nouveaux derives de penicilline et de cephalusporine

Also Published As

Publication number Publication date
DK145059C (da) 1983-01-24
DE2258221C2 (de) 1981-10-08
FI56841C (fi) 1980-04-10
IE36881L (en) 1973-05-29
SU467521A3 (ru) 1975-04-15
HU165582B (fi) 1974-09-28
AU4910472A (en) 1974-05-23
CA1023344A (en) 1977-12-27
FR2186968A5 (fi) 1974-01-11
DD100955A5 (fi) 1973-10-12
YU36181B (en) 1982-02-25
AU470085B2 (en) 1976-03-04
YU289972A (en) 1981-06-30
DE2258221A1 (de) 1973-06-14
GB1401059A (en) 1975-07-16
CS177830B2 (fi) 1977-08-31
ES408972A1 (es) 1975-10-01
US4041029A (en) 1977-08-09
NL187633B (nl) 1991-07-01
FI56841B (fi) 1979-12-31
CH594680A5 (fi) 1978-01-13
NL187633C (nl) 1991-12-02
JPS5850230B2 (ja) 1983-11-09
JPS5762290A (en) 1982-04-15
NL7215466A (fi) 1973-06-01
DK145059B (da) 1982-08-16
IE36881B1 (en) 1977-03-16
JPS4862791A (fi) 1973-09-01
AT322098B (de) 1975-05-12
JPS5852998B2 (ja) 1983-11-26
PL85390B1 (fi) 1976-04-30

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