RU94020717A - Применение тетрагидробенз[cd]индол-6-карбоксамидов для предотвращения рвоты и лечения половой дисфункции, фармацевтические препараты на их основе - Google Patents
Применение тетрагидробенз[cd]индол-6-карбоксамидов для предотвращения рвоты и лечения половой дисфункции, фармацевтические препараты на их основеInfo
- Publication number
- RU94020717A RU94020717A RU94020717/14A RU94020717A RU94020717A RU 94020717 A RU94020717 A RU 94020717A RU 94020717/14 A RU94020717/14 A RU 94020717/14A RU 94020717 A RU94020717 A RU 94020717A RU 94020717 A RU94020717 A RU 94020717A
- Authority
- RU
- Russia
- Prior art keywords
- tetrahydrobenz
- carboxamides
- indole
- pharmaceutical preparations
- sexual dysfunction
- Prior art date
Links
- 238000011282 treatment Methods 0.000 title claims abstract 5
- 201000001880 Sexual dysfunction Diseases 0.000 title claims abstract 3
- 206010047700 Vomiting Diseases 0.000 title claims abstract 3
- 239000000825 pharmaceutical preparation Substances 0.000 title claims abstract 3
- 231100000872 sexual dysfunction Toxicity 0.000 title claims abstract 3
- 230000008673 vomiting Effects 0.000 title claims abstract 3
- 230000002265 prevention Effects 0.000 title abstract 2
- 238000000034 method Methods 0.000 claims 2
- ZYVORBSWPVDTCX-UHFFFAOYSA-N 1,2,2a,3-tetrahydrobenzo[cd]indole Chemical class C1=CCC2CNC3=CC=CC1=C32 ZYVORBSWPVDTCX-UHFFFAOYSA-N 0.000 claims 1
- 241000124008 Mammalia Species 0.000 claims 1
- 230000000694 effects Effects 0.000 abstract 1
- 239000000126 substance Substances 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
- A61K31/403—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
- A61K31/404—Indoles, e.g. pindolol
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/08—Drugs for genital or sexual disorders; Contraceptives for gonadal disorders or for enhancing fertility, e.g. inducers of ovulation or of spermatogenesis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/10—Drugs for genital or sexual disorders; Contraceptives for impotence
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
Landscapes
- Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Epidemiology (AREA)
- Reproductive Health (AREA)
- Endocrinology (AREA)
- Gynecology & Obstetrics (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Hospice & Palliative Care (AREA)
- Otolaryngology (AREA)
- Pregnancy & Childbirth (AREA)
- Urology & Nephrology (AREA)
- Neurosurgery (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Indole Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Abstract
Предлагаемое изобретение предусматривает способы предотвращения рвоты и лечения половой дисфункции у млекопитающих с использованием некоторых тетрагидробенз [cd] индолов. Изобретение также предлагает фармацевтические препараты, пригодные для использования в таких способах лечения.
Claims (1)
- Предлагаемое изобретение предусматривает способы предотвращения рвоты и лечения половой дисфункции у млекопитающих с использованием некоторых тетрагидробенз [cd] индолов. Изобретение также предлагает фармацевтические препараты, пригодные для использования в таких способах лечения.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US7519893A | 1993-06-10 | 1993-06-10 | |
US08/075,198 | 1993-06-10 |
Related Child Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
RU99117174/14A Division RU99117174A (ru) | 1993-06-10 | 1999-08-05 | Применение тетрагидробенз [cd] индол-6-карбоксамидов для лечения половой дисфункции, фармацевтическая композиция |
Publications (2)
Publication Number | Publication Date |
---|---|
RU94020717A true RU94020717A (ru) | 1996-08-27 |
RU2154476C2 RU2154476C2 (ru) | 2000-08-20 |
Family
ID=22124191
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
RU94020717/14A RU2154476C2 (ru) | 1993-06-10 | 1994-06-09 | ПРИМЕНЕНИЕ ТЕТРАГИДРОБЕНЗ /cd/ИНДОЛ-6-КАРБОКСАМИДОВ ДЛЯ ПРЕДОТВРАЩЕНИЯ РВОТЫ, ФАРМАЦЕВТИЧЕСКИЕ ПРЕПАРАТЫ НА ИХ ОСНОВЕ |
Country Status (17)
Country | Link |
---|---|
US (1) | US5703112A (ru) |
EP (2) | EP1166783A3 (ru) |
JP (1) | JPH0748254A (ru) |
KR (2) | KR100367792B1 (ru) |
CN (2) | CN1072932C (ru) |
AU (1) | AU677317B2 (ru) |
CA (1) | CA2125088A1 (ru) |
CZ (2) | CZ285762B6 (ru) |
HK (1) | HK1043322B (ru) |
HU (1) | HUT71464A (ru) |
IL (1) | IL109872A (ru) |
NO (4) | NO321500B1 (ru) |
NZ (2) | NZ260667A (ru) |
RU (1) | RU2154476C2 (ru) |
TW (1) | TW258660B (ru) |
UA (2) | UA29415C2 (ru) |
ZA (1) | ZA943862B (ru) |
Families Citing this family (13)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
AU4663100A (en) | 1999-04-30 | 2000-11-17 | Lilly Icos Llc | Treatment of female arousal disorder |
GB0106446D0 (en) * | 2001-03-15 | 2001-05-02 | Vernalis Res Ltd | Chemical compounds |
AU2006254899B2 (en) | 2005-06-08 | 2011-11-24 | Sk Biopharmaceuticals Co., Ltd. | Treatment of sleep-wake disorders |
CA2612672C (en) * | 2005-06-22 | 2014-10-14 | Janssen Pharmaceutica, N.V. | Treatment for sexual dysfunction |
US8741950B2 (en) | 2009-06-22 | 2014-06-03 | Sk Biopharmaceuticals Co., Ltd. | Methods for treating or preventing fatigue |
MX2012005258A (es) | 2009-11-06 | 2012-06-19 | Sk Biopharmaceuticals Co Ltd | El uso de un compuesto de carbamoilo para el tratamiento del trastorno de deficit de atencion/hiperactividad. |
AU2010316172B2 (en) | 2009-11-06 | 2015-11-12 | Sk Biopharmaceuticals Co., Ltd. | Methods for treating fibromyalgia syndrome |
US9610274B2 (en) | 2010-06-30 | 2017-04-04 | Sk Biopharmaceuticals Co., Ltd. | Methods for treating bipolar disorder |
DK2968208T3 (da) | 2013-03-13 | 2022-08-22 | Jazz Pharmaceuticals Ireland Ltd | Behandling af kataplexi |
CN110638804A (zh) | 2013-07-18 | 2020-01-03 | 爵士制药国际Iii有限公司 | 治疗肥胖 |
US10195151B2 (en) | 2016-09-06 | 2019-02-05 | Jazz Pharmaceuticals International Iii Limited | Formulations of (R)-2-amino-3-phenylpropyl carbamate |
KR20200016889A (ko) | 2017-06-02 | 2020-02-17 | 재즈 파마슈티칼즈 아일랜드 리미티드 | 과다 졸림증을 치료하기 위한 방법 및 조성물 |
US10940133B1 (en) | 2020-03-19 | 2021-03-09 | Jazz Pharmaceuticals Ireland Limited | Methods of providing solriamfetol therapy to subjects with impaired renal function |
Family Cites Families (16)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4110339A (en) * | 1977-11-25 | 1978-08-29 | Eli Lilly And Company | 4-(Di-n-propyl)amino-1,3,4,5-tetrahydrobenz[cd]indole |
US4521421A (en) * | 1983-09-26 | 1985-06-04 | Eli Lilly And Company | Treatment of sexual dysfunction |
US4576959A (en) * | 1984-02-06 | 1986-03-18 | Eli Lilly And Company | 6-Substituted-4-dialkylaminotetrahydrobenz[c,d]indoles |
CA1266482A1 (en) * | 1984-05-24 | 1990-03-06 | Carl Kaiser | 6-oxygenated-1,3,4,5-tetrahydrobenz(cd)indol-4-amines |
US4745126A (en) * | 1987-03-12 | 1988-05-17 | Eli Lilly And Company | Method of treating anxiety with tetrahydrobenz[c,d]indole-6-carboxamides |
US4943428A (en) * | 1987-07-10 | 1990-07-24 | Wright State University | Stimulation of serotonin-1A receptors in mammals to alleviate motion sickness and emesis induced by chemical agents |
DE3809155A1 (de) * | 1988-03-18 | 1989-09-28 | Bayer Ag | 1,3,4,5-tetrahydrobenz-(c,d)-indole |
US5204340A (en) * | 1989-04-11 | 1993-04-20 | Eli Lilly And Company | Tetrahydrobenz(c,d)indole serotonin agonists |
KR0151699B1 (ko) * | 1989-07-13 | 1998-10-15 | 로버트 에이. 아미테이지 | (1,2n) 및 (3,2n)-카보사이클릭-2-아미노테트랄린 유도체 |
IL97308A (en) * | 1990-02-26 | 1996-10-31 | Lilly Co Eli | Xahydrobenz [DC] Induced indoles in position 6, their preparation process and pharmaceutical preparations containing them |
US5302612A (en) * | 1990-02-26 | 1994-04-12 | Eli Lilly And Company | 6-substituted-hexahydrobenz[cd]indoles |
WO1991013872A1 (en) * | 1990-03-15 | 1991-09-19 | The Upjohn Company | Therapeutically useful heterocyclic indole compounds |
US5258379A (en) * | 1990-05-04 | 1993-11-02 | Eli Lilly And Company | Method of inhibiting gastric acid secretion with n-arylpiperazines |
US5096908A (en) * | 1990-05-04 | 1992-03-17 | Eli Lilly And Company | Method of inhibiting gastric acid secretion |
US5229409A (en) * | 1990-08-15 | 1993-07-20 | Eli Lilly And Company | 6-substituted-tetrahydrobenz[cd]indoles |
US5244912A (en) * | 1991-03-28 | 1993-09-14 | Eli Lilly And Company | 6-heterocyclic-4-amino-1,3,4,5-tetrahydrobenz(cd)indoles and pharmaceutical use thereof |
-
1994
- 1994-06-02 NZ NZ260667A patent/NZ260667A/en unknown
- 1994-06-02 CZ CZ941354A patent/CZ285762B6/cs not_active IP Right Cessation
- 1994-06-02 NZ NZ314570A patent/NZ314570A/xx unknown
- 1994-06-02 IL IL10987294A patent/IL109872A/xx not_active IP Right Cessation
- 1994-06-02 ZA ZA943862A patent/ZA943862B/xx unknown
- 1994-06-02 CZ CZ982818A patent/CZ285829B6/cs not_active IP Right Cessation
- 1994-06-03 CA CA002125088A patent/CA2125088A1/en not_active Abandoned
- 1994-06-04 TW TW083105103A patent/TW258660B/zh active
- 1994-06-06 UA UA94005243A patent/UA29415C2/ru unknown
- 1994-06-07 EP EP01201582A patent/EP1166783A3/en not_active Withdrawn
- 1994-06-07 EP EP94304103A patent/EP0633023A3/en not_active Withdrawn
- 1994-06-08 AU AU64607/94A patent/AU677317B2/en not_active Ceased
- 1994-06-08 KR KR1019940012778A patent/KR100367792B1/ko not_active IP Right Cessation
- 1994-06-09 CN CN94106467A patent/CN1072932C/zh not_active Expired - Fee Related
- 1994-06-09 HU HU9401730A patent/HUT71464A/hu unknown
- 1994-06-09 JP JP6127646A patent/JPH0748254A/ja active Pending
- 1994-06-09 RU RU94020717/14A patent/RU2154476C2/ru not_active IP Right Cessation
- 1994-06-09 NO NO19942143A patent/NO321500B1/no unknown
-
1995
- 1995-11-17 US US08/560,174 patent/US5703112A/en not_active Expired - Fee Related
-
1999
- 1999-03-30 NO NO991551A patent/NO991551D0/no unknown
- 1999-07-14 NO NO993461A patent/NO308693B1/no unknown
-
2000
- 2000-06-27 UA UA2000063803A patent/UA37311C2/ru unknown
- 2000-10-31 CN CNB00132828XA patent/CN1170536C/zh not_active Expired - Fee Related
-
2001
- 2001-11-28 NO NO20015806A patent/NO20015806D0/no unknown
-
2002
- 2002-07-12 HK HK02105194.1A patent/HK1043322B/zh not_active IP Right Cessation
- 2002-08-31 KR KR1020020052257A patent/KR100367791B1/ko not_active IP Right Cessation
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
MM4A | The patent is invalid due to non-payment of fees |
Effective date: 20070610 |