RU2636147C1 - Производные 1,6-диазабицикло[3,2,1]октан-7-она и их применение при лечении бактериальных инфекционных болезней - Google Patents

Производные 1,6-диазабицикло[3,2,1]октан-7-она и их применение при лечении бактериальных инфекционных болезней Download PDF

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RU2636147C1
RU2636147C1 RU2016106633A RU2016106633A RU2636147C1 RU 2636147 C1 RU2636147 C1 RU 2636147C1 RU 2016106633 A RU2016106633 A RU 2016106633A RU 2016106633 A RU2016106633 A RU 2016106633A RU 2636147 C1 RU2636147 C1 RU 2636147C1
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pharmaceutically acceptable
diazabicyclo
oxo
trans
subject
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RU2016106633A
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Russian (ru)
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Махеш Витхалбхай Пател
Прасад Кешав Дешпанде
Сатиш БХАВСАР
Сачин БХАГВАТ
Мохаммад Алам ДЖАФРИ
Амит МИШРА
Лаксмикант ПАВАСЕ
Сунил Гупта
Раджеш КАЛЕ
Санджив ДЖОШИ
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Вокхардт Лимитед
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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/5375—1,4-Oxazines, e.g. morpholine
    • A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
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    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
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    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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    • A61K31/425—Thiazoles
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    • A61K31/425—Thiazoles
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    • A61K31/43—Compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula, e.g. penicillins, penems
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    • A61K31/54—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
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    • A61K31/545—Compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins, cefaclor, or cephalexine
    • A61K31/546—Compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins, cefaclor, or cephalexine containing further heterocyclic rings, e.g. cephalothin
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RU2016106633A 2011-08-27 2012-08-24 Производные 1,6-диазабицикло[3,2,1]октан-7-она и их применение при лечении бактериальных инфекционных болезней RU2636147C1 (ru)

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IN2412MU2011 2011-08-27

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RU2013155902/04A RU2578370C2 (ru) 2011-08-27 2012-08-24 Производные 1,6- диазабицикло [3,2,1] октан-7-она и их применение при лечении бактериальных инфекционных болезней

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US (5) US8822450B2 (OSRAM)
EP (1) EP2748165B1 (OSRAM)
JP (1) JP5666743B2 (OSRAM)
KR (1) KR101512738B1 (OSRAM)
CN (1) CN103619843B (OSRAM)
AU (1) AU2012303691B2 (OSRAM)
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