RU2572214C2 - Способ получения цинковых комплексов инсулина - Google Patents
Способ получения цинковых комплексов инсулина Download PDFInfo
- Publication number
- RU2572214C2 RU2572214C2 RU2012148821/15A RU2012148821A RU2572214C2 RU 2572214 C2 RU2572214 C2 RU 2572214C2 RU 2012148821/15 A RU2012148821/15 A RU 2012148821/15A RU 2012148821 A RU2012148821 A RU 2012148821A RU 2572214 C2 RU2572214 C2 RU 2572214C2
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- Russia
- Prior art keywords
- insulin
- cooh
- chain
- amino acid
- group
- Prior art date
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- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Chemistry (AREA)
- Inorganic Chemistry (AREA)
- Hematology (AREA)
- Emergency Medicine (AREA)
- Obesity (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Peptides Or Proteins (AREA)
- Medicinal Preparation (AREA)
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP10162368 | 2010-05-10 | ||
| EP10162368.4 | 2010-05-10 | ||
| US33349710P | 2010-05-11 | 2010-05-11 | |
| US61/333,497 | 2010-05-11 | ||
| PCT/EP2011/057388 WO2011141407A1 (en) | 2010-05-10 | 2011-05-09 | Process for the preparation of insulin-zinc complexes |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| RU2012148821A RU2012148821A (ru) | 2014-06-20 |
| RU2572214C2 true RU2572214C2 (ru) | 2015-12-27 |
Family
ID=42732779
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| RU2012148821/15A RU2572214C2 (ru) | 2010-05-10 | 2011-05-09 | Способ получения цинковых комплексов инсулина |
Country Status (12)
| Country | Link |
|---|---|
| US (5) | US20130143803A1 (enExample) |
| EP (1) | EP2569002B1 (enExample) |
| JP (2) | JP6249773B2 (enExample) |
| KR (2) | KR20160105979A (enExample) |
| CN (2) | CN102883743A (enExample) |
| AU (1) | AU2011252127B2 (enExample) |
| BR (1) | BR112012028766A2 (enExample) |
| CA (1) | CA2795091A1 (enExample) |
| ES (1) | ES2612468T3 (enExample) |
| MX (1) | MX2012012943A (enExample) |
| RU (1) | RU2572214C2 (enExample) |
| WO (1) | WO2011141407A1 (enExample) |
Families Citing this family (22)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2006082204A1 (en) | 2005-02-02 | 2006-08-10 | Novo Nordisk A/S | Insulin derivatives |
| EP1969004B1 (en) | 2005-12-28 | 2011-08-10 | Novo Nordisk A/S | Compositions comprising an acylated insulin and zinc and method of making the said compositions |
| JP5202338B2 (ja) | 2006-02-27 | 2013-06-05 | ノボ・ノルデイスク・エー／エス | 新規インシュリン誘導体 |
| AU2007247109B2 (en) | 2006-05-09 | 2012-03-15 | Novo Nordisk A/S | Insulin derivative |
| WO2007128815A1 (en) | 2006-05-09 | 2007-11-15 | Novo Nordisk A/S | Insulin derivative |
| JP5552046B2 (ja) | 2007-06-13 | 2014-07-16 | ノボ・ノルデイスク・エー／エス | インスリン誘導体を含有する薬学的製剤 |
| ES2543393T3 (es) | 2007-11-08 | 2015-08-18 | Novo Nordisk A/S | Derivado de insulina |
| CN102202683A (zh) | 2008-10-30 | 2011-09-28 | 诺沃-诺迪斯克有限公司 | 用少于每日一次的注射频率注射胰岛素来治疗糖尿病 |
| DK2632478T3 (da) | 2010-10-27 | 2019-10-07 | Novo Nordisk As | Behandling af diabetes melitus under anvendelse af insulinindsprøjtninger indgivet med varierende indsprøjtningsintervaller |
| US20160296602A1 (en) * | 2013-03-20 | 2016-10-13 | Novo Nordisk A/S | Dosing Regimen |
| EP2991672A1 (en) | 2013-04-30 | 2016-03-09 | Novo Nordisk A/S | Novel administration regime |
| CA2926701A1 (en) * | 2013-10-07 | 2015-04-16 | Novo Nordisk A/S | Novel derivative of an insulin analogue |
| AR099569A1 (es) | 2014-02-28 | 2016-08-03 | Novo Nordisk As | Derivados de insulina y los usos médicos de estos |
| DK3006045T3 (en) | 2014-10-07 | 2017-07-17 | Cyprumed Gmbh | Pharmaceutical formulations for oral administration of peptide or protein drugs |
| EP3740195A1 (fr) * | 2017-12-07 | 2020-11-25 | Adocia | Compositions sous forme d'une solution aqueuse injectable comprenant de l'amyline, un agoniste au recepteur de l'amyline ou un analogue d'amyline et un co-polyaminoacide |
| IL275146B2 (en) | 2017-12-07 | 2025-01-01 | Adocia | Preparations in the form of an aqueous solution for injection comprising amylin, an amylin receptor agonist or an amylin analog and a copolyamino acid |
| WO2019149245A1 (zh) * | 2018-02-01 | 2019-08-08 | 江苏恒瑞医药股份有限公司 | 含人胰岛素类似物的酰化衍生物的药物组合物及其制备方法 |
| KR20210016400A (ko) | 2018-05-24 | 2021-02-15 | 지앙수 헨그루이 메디슨 컴퍼니 리미티드 | 재조합 인간 인슐린 또는 그 유사체의 전구체를 제조하는 방법 |
| US10335464B1 (en) | 2018-06-26 | 2019-07-02 | Novo Nordisk A/S | Device for titrating basal insulin |
| TW202039437A (zh) | 2018-12-11 | 2020-11-01 | 法商賽諾菲公司 | 肽黏合劑 |
| CN114096269B (zh) | 2019-07-12 | 2024-06-11 | 诺和诺德股份有限公司 | 高浓度胰岛素制剂 |
| CN115300639A (zh) * | 2021-05-06 | 2022-11-08 | 南京汉欣医药科技有限公司 | 一种含有德谷胰岛素的缓释药物组合物及其制备方法 |
Citations (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3868358A (en) * | 1971-04-30 | 1975-02-25 | Lilly Co Eli | Protamine-insulin product |
| EP0214826A2 (en) * | 1985-08-30 | 1987-03-18 | Novo Nordisk A/S | Insulin analogues and method of preparing the same |
| US20090312236A1 (en) * | 2008-06-13 | 2009-12-17 | John Michael Beals | Pegylated insulin lispro compounds |
Family Cites Families (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE1212679B (de) * | 1957-08-03 | 1966-03-17 | Novo Terapeutisk Labor As | Verfahren zur Herstellung von Insulinloesungen |
| GB1042194A (en) * | 1962-04-30 | 1966-09-14 | Olin Mathieson | Insulin preparations |
| DK113585D0 (da) * | 1985-03-12 | 1985-03-12 | Novo Industri As | Nye peptider |
| US4764592A (en) * | 1987-04-23 | 1988-08-16 | Eli Lilly And Company | Crystalline human proinsulin and process for its production |
| HUT56857A (en) | 1988-12-23 | 1991-10-28 | Novo Nordisk As | Human insulin analogues |
| IL93282A (en) | 1989-02-09 | 1995-08-31 | Lilly Co Eli | Insulin analogues |
| NZ273285A (en) * | 1993-09-17 | 1997-10-24 | Novo Nordisk As | Insulin derivatives and compositions thereof |
| US7097845B2 (en) * | 1997-04-23 | 2006-08-29 | Jacob Sten Petersen | Combinations of antigen and mucosal binding component for inducing specific immunological tolerance |
| ES2472421T3 (es) * | 2003-08-05 | 2014-07-01 | Novo Nordisk A/S | Nuevos derivados de insulina |
| AU2004261353B2 (en) | 2003-08-05 | 2009-12-10 | Novo Nordisk A/S | Novel insulin derivatives |
| EP1969004B1 (en) | 2005-12-28 | 2011-08-10 | Novo Nordisk A/S | Compositions comprising an acylated insulin and zinc and method of making the said compositions |
| JP5552046B2 (ja) * | 2007-06-13 | 2014-07-16 | ノボ・ノルデイスク・エー／エス | インスリン誘導体を含有する薬学的製剤 |
-
2011
- 2011-05-09 AU AU2011252127A patent/AU2011252127B2/en not_active Ceased
- 2011-05-09 EP EP11718398.8A patent/EP2569002B1/en active Active
- 2011-05-09 ES ES11718398.8T patent/ES2612468T3/es active Active
- 2011-05-09 CA CA2795091A patent/CA2795091A1/en not_active Withdrawn
- 2011-05-09 KR KR1020167023293A patent/KR20160105979A/ko not_active Ceased
- 2011-05-09 RU RU2012148821/15A patent/RU2572214C2/ru not_active IP Right Cessation
- 2011-05-09 BR BR112012028766A patent/BR112012028766A2/pt not_active Application Discontinuation
- 2011-05-09 CN CN201180023303XA patent/CN102883743A/zh active Pending
- 2011-05-09 JP JP2013509525A patent/JP6249773B2/ja active Active
- 2011-05-09 WO PCT/EP2011/057388 patent/WO2011141407A1/en not_active Ceased
- 2011-05-09 KR KR1020127029547A patent/KR20130092972A/ko not_active Ceased
- 2011-05-09 MX MX2012012943A patent/MX2012012943A/es active IP Right Grant
- 2011-05-09 US US13/696,897 patent/US20130143803A1/en not_active Abandoned
- 2011-05-09 CN CN201611166272.4A patent/CN107029212A/zh active Pending
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2015
- 2015-03-19 US US14/662,874 patent/US20150250857A1/en not_active Abandoned
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2017
- 2017-02-28 US US15/445,305 patent/US20170165327A1/en not_active Abandoned
- 2017-08-16 JP JP2017157054A patent/JP2017203042A/ja not_active Withdrawn
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2020
- 2020-08-12 US US16/991,803 patent/US20210060132A1/en not_active Abandoned
-
2024
- 2024-05-24 US US18/674,042 patent/US20240307503A1/en active Pending
Patent Citations (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3868358A (en) * | 1971-04-30 | 1975-02-25 | Lilly Co Eli | Protamine-insulin product |
| EP0214826A2 (en) * | 1985-08-30 | 1987-03-18 | Novo Nordisk A/S | Insulin analogues and method of preparing the same |
| US20090312236A1 (en) * | 2008-06-13 | 2009-12-17 | John Michael Beals | Pegylated insulin lispro compounds |
Also Published As
| Publication number | Publication date |
|---|---|
| CA2795091A1 (en) | 2011-11-17 |
| US20210060132A1 (en) | 2021-03-04 |
| EP2569002B1 (en) | 2016-10-26 |
| US20130143803A1 (en) | 2013-06-06 |
| KR20160105979A (ko) | 2016-09-08 |
| JP2017203042A (ja) | 2017-11-16 |
| CN107029212A (zh) | 2017-08-11 |
| AU2011252127B2 (en) | 2014-02-20 |
| ES2612468T3 (es) | 2017-05-17 |
| JP6249773B2 (ja) | 2017-12-20 |
| US20240307503A1 (en) | 2024-09-19 |
| AU2011252127A1 (en) | 2012-11-01 |
| US20150250857A1 (en) | 2015-09-10 |
| KR20130092972A (ko) | 2013-08-21 |
| MX2012012943A (es) | 2012-11-29 |
| US20170165327A1 (en) | 2017-06-15 |
| WO2011141407A1 (en) | 2011-11-17 |
| BR112012028766A2 (pt) | 2017-06-13 |
| CN102883743A (zh) | 2013-01-16 |
| JP2013526501A (ja) | 2013-06-24 |
| EP2569002A1 (en) | 2013-03-20 |
| RU2012148821A (ru) | 2014-06-20 |
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| HE9A | Changing address for correspondence with an applicant | ||
| MM4A | The patent is invalid due to non-payment of fees |
Effective date: 20190510 |