RU2228170C2 - Устройства для доставки лекарственных средств, обладающих антипрогестиновыми свойствами - Google Patents

Устройства для доставки лекарственных средств, обладающих антипрогестиновыми свойствами Download PDF

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RU2228170C2
RU2228170C2 RU2002119587/15A RU2002119587A RU2228170C2 RU 2228170 C2 RU2228170 C2 RU 2228170C2 RU 2002119587/15 A RU2002119587/15 A RU 2002119587/15A RU 2002119587 A RU2002119587 A RU 2002119587A RU 2228170 C2 RU2228170 C2 RU 2228170C2
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Russia
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beta
groups
hydroxy
poly
alkylene oxide
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RU2002119587/15A
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Russian (ru)
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RU2002119587A (ru
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Харри ЮКАРАЙНЕН (FI)
Харри Юкарайнен
Томми МАРККУЛА (GB)
Томми МАРККУЛА
Юха АЛА-СОРВАРИ (FI)
Юха АЛА-СОРВАРИ
Матти ЛЕХТИНЕН (FI)
Матти ЛЕХТИНЕН
Яркко РУОХОНЕН (FI)
Яркко РУОХОНЕН
Тимо ХААПАКУМПУ (FI)
Тимо ХААПАКУМПУ
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Шеринг Ой
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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0019—Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
    • A61K9/0024—Solid, semi-solid or solidifying implants, which are implanted or injected in body tissue
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61K31/12—Ketones
    • A61K31/122—Ketones having the oxygen directly attached to a ring, e.g. quinones, vitamin K1, anthralin
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    • A61K31/275—Nitriles; Isonitriles
    • A61K31/277—Nitriles; Isonitriles having a ring, e.g. verapamil
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4418—Non condensed pyridines; Hydrogenated derivatives thereof having a carbocyclic group directly attached to the heterocyclic ring, e.g. cyproheptadine
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/50—Pyridazines; Hydrogenated pyridazines
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    • A61K31/50—Pyridazines; Hydrogenated pyridazines
    • A61K31/502—Pyridazines; Hydrogenated pyridazines ortho- or peri-condensed with carbocyclic ring systems, e.g. cinnoline, phthalazine
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    • A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
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    • A61K31/575—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of three or more carbon atoms, e.g. cholane, cholestane, ergosterol, sitosterol
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    • C08L—COMPOSITIONS OF MACROMOLECULAR COMPOUNDS
    • C08L83/00—Compositions of macromolecular compounds obtained by reactions forming in the main chain of the macromolecule a linkage containing silicon with or without sulfur, nitrogen, oxygen or carbon only; Compositions of derivatives of such polymers
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  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Reproductive Health (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Endocrinology (AREA)
  • Gynecology & Obstetrics (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Polymers & Plastics (AREA)
  • Diabetes (AREA)
  • Rheumatology (AREA)
  • Pregnancy & Childbirth (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Dermatology (AREA)
  • Urology & Nephrology (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Steroid Compounds (AREA)
RU2002119587/15A 1999-12-23 2000-11-21 Устройства для доставки лекарственных средств, обладающих антипрогестиновыми свойствами RU2228170C2 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US09/472,126 1999-12-23
US09/472,126 US6476079B1 (en) 1999-12-23 1999-12-23 Devices for the delivery of drugs having antiprogestinic properties

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RU2002119587A RU2002119587A (ru) 2004-02-27
RU2228170C2 true RU2228170C2 (ru) 2004-05-10

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US (1) US6476079B1 (enExample)
EP (1) EP1239829B1 (enExample)
JP (1) JP4895150B2 (enExample)
KR (1) KR100850548B1 (enExample)
CN (1) CN100346772C (enExample)
AR (1) AR026647A1 (enExample)
AT (1) ATE401859T1 (enExample)
AU (1) AU781555B2 (enExample)
BR (1) BR0016697A (enExample)
CA (1) CA2395226C (enExample)
CO (1) CO5261571A1 (enExample)
CZ (1) CZ301865B6 (enExample)
DE (2) DE60039626D1 (enExample)
DK (1) DK1239829T3 (enExample)
EE (1) EE05123B1 (enExample)
ES (1) ES2310526T3 (enExample)
HK (1) HK1047235B (enExample)
HU (1) HU229438B1 (enExample)
IL (2) IL149663A0 (enExample)
MX (1) MXPA02006174A (enExample)
NO (1) NO332261B1 (enExample)
NZ (1) NZ519876A (enExample)
PE (1) PE20010801A1 (enExample)
PL (1) PL201216B1 (enExample)
PT (1) PT1239829E (enExample)
RU (1) RU2228170C2 (enExample)
SK (1) SK287229B6 (enExample)
TW (1) TWI248367B (enExample)
UA (1) UA70401C2 (enExample)
WO (1) WO2001047490A1 (enExample)
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Cited By (5)

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Publication number Priority date Publication date Assignee Title
RU2488369C2 (ru) * 2007-09-21 2013-07-27 Мсд Осс Б.В. Система доставки лекарственных веществ
RU2503431C2 (ru) * 2007-11-07 2014-01-10 Мерк Шарт и Доум Б.В. Носитель для внутриматочного размещения
RU2529477C2 (ru) * 2009-05-04 2014-09-27 Мерк Шарп и Доум Б.В. Внутриматочная система для лечебного использования
RU2539995C2 (ru) * 2008-11-06 2015-01-27 Ново Нордиск А/С Устройство для ввода лекарства со вспомогательной электронной системой
RU2607179C2 (ru) * 2011-07-20 2017-01-10 Патрик Ф. КАЙЗЕР Интравагинальные устройства для доставки лекарственных средсв

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US6794464B2 (en) 1998-06-30 2004-09-21 Schering Oy Membrane or matrix for controlling the permeation rate of drugs
AU2002210580A1 (en) * 2000-10-20 2002-04-29 Leiras Oy Drug delivery system
CN1289064C (zh) * 2001-08-31 2006-12-13 先灵有限责任公司 药物输送体系
EP1438942A1 (en) * 2003-01-17 2004-07-21 Schering Oy An otorhinological drug delivery device
PL1696822T3 (pl) * 2003-11-13 2010-08-31 Psivida Inc Wstrzykiwane implanty o opóźnionym wydzielaniu mające matrycę rdzenia i powłokę podatne na erozję biologiczną
RU2283637C1 (ru) * 2005-03-22 2006-09-20 Общество с ограниченной ответственностью "Производственно-коммерческая фирма "Две линии" Пластырь
US7862552B2 (en) 2005-05-09 2011-01-04 Boston Scientific Scimed, Inc. Medical devices for treating urological and uterine conditions
JP5137841B2 (ja) 2005-10-13 2013-02-06 シンセス ゲーエムベーハー 薬物含浸容器
US20070149916A1 (en) * 2005-12-22 2007-06-28 Alza Corporation Dry matrices as drug reservoirs in electrotransport applications
EP1862468A1 (de) * 2006-06-02 2007-12-05 Bayer Schering Pharma Aktiengesellschaft Kristallines 11beta-(4-Acetylphenyl)-20,20,21,21,21-pentafluor-17-hydroxy-19-nor-17alpha-pregna-4,9-dien-3-on
US20080261929A1 (en) * 2007-04-23 2008-10-23 Jens Hoffmann Combination of progesterone-receptor antagonist together with an aromatase inhibitor for use in brca mediated diseases
DE102007032468A1 (de) * 2007-07-10 2009-01-15 Brätter, Christian, Dr. Transdermale Therapeutische Systeme, welche den Wirkstoff Anastrozol enthalten
TW200927141A (en) * 2007-11-22 2009-07-01 Bayer Schering Pharma Oy Vaginal delivery system
RU2494706C2 (ru) 2008-09-17 2013-10-10 Байер Ой Устройство для введения
US11992431B2 (en) 2008-09-17 2024-05-28 Bayer Oy Inserter
FI20080523A0 (fi) * 2008-09-17 2008-09-17 Bayer Schering Pharma Oy Insertteri
US8822610B2 (en) 2008-12-22 2014-09-02 ATRP Solutions, Inc. Control over controlled radical polymerization processes
US8815971B2 (en) 2008-12-22 2014-08-26 ATRP Solutions, Inc. Control over controlled radical polymerization processes
US8173750B2 (en) 2009-04-23 2012-05-08 ATRP Solutions, Inc. Star macromolecules for personal and home care
US9783628B2 (en) 2009-04-23 2017-10-10 ATRP Solutions, Inc. Dual-mechanism thickening agents for hydraulic fracturing fluids
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