RU2195450C2 - Новые способы и промежуточные соединения - Google Patents
Новые способы и промежуточные соединения Download PDFInfo
- Publication number
- RU2195450C2 RU2195450C2 RU2000115273/04A RU2000115273A RU2195450C2 RU 2195450 C2 RU2195450 C2 RU 2195450C2 RU 2000115273/04 A RU2000115273/04 A RU 2000115273/04A RU 2000115273 A RU2000115273 A RU 2000115273A RU 2195450 C2 RU2195450 C2 RU 2195450C2
- Authority
- RU
- Russia
- Prior art keywords
- compound
- formula
- mixture
- organic layer
- sequentially
- Prior art date
Links
- 0 *C([C@@]1[C@@](*)C(O)OCC1)C(C(*1)=Cc2c1ccc(N)c2)=O Chemical compound *C([C@@]1[C@@](*)C(O)OCC1)C(C(*1)=Cc2c1ccc(N)c2)=O 0.000 description 1
- OLSFUYVRFNCMSF-IUYQGCFVSA-O CC[C@@H]([C@H](C(O)=[OH+])O)N Chemical compound CC[C@@H]([C@H](C(O)=[OH+])O)N OLSFUYVRFNCMSF-IUYQGCFVSA-O 0.000 description 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C229/00—Compounds containing amino and carboxyl groups bound to the same carbon skeleton
- C07C229/02—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton
- C07C229/34—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton containing six-membered aromatic rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/10—Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
- C07D209/12—Radicals substituted by oxygen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/30—Indoles; Hydrogenated indoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to carbon atoms of the hetero ring
- C07D209/42—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B2200/00—Indexing scheme relating to specific properties of organic compounds
- C07B2200/07—Optical isomers
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Indole Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Preparation Of Compounds By Using Micro-Organisms (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US13999799P | 1999-06-18 | 1999-06-18 | |
| US60/139,997 | 1999-06-18 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| RU2000115273A RU2000115273A (ru) | 2002-06-10 |
| RU2195450C2 true RU2195450C2 (ru) | 2002-12-27 |
Family
ID=22489263
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| RU2000115273/04A RU2195450C2 (ru) | 1999-06-18 | 2000-06-16 | Новые способы и промежуточные соединения |
Country Status (18)
| Country | Link |
|---|---|
| US (1) | US6410750B1 (enExample) |
| EP (1) | EP1061074A1 (enExample) |
| JP (1) | JP3342471B2 (enExample) |
| KR (1) | KR20010049559A (enExample) |
| CN (1) | CN1283615A (enExample) |
| AU (1) | AU4089200A (enExample) |
| BR (1) | BR0002686A (enExample) |
| CA (1) | CA2311872A1 (enExample) |
| CZ (1) | CZ20002242A3 (enExample) |
| HU (1) | HUP0002285A3 (enExample) |
| ID (1) | ID26385A (enExample) |
| IL (1) | IL136726A0 (enExample) |
| IN (1) | IN188853B (enExample) |
| PL (1) | PL340866A1 (enExample) |
| RU (1) | RU2195450C2 (enExample) |
| TR (1) | TR200001781A2 (enExample) |
| YU (1) | YU38000A (enExample) |
| ZA (1) | ZA200002987B (enExample) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AR052864A1 (es) * | 2005-01-06 | 2007-04-11 | Schering Corp | Preparacion de cetoamidas |
| EP2714660B1 (en) * | 2011-05-31 | 2018-09-26 | Theravance Biopharma R&D IP, LLC | Neprilysin inhibitors |
Citations (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO1996039385A1 (en) * | 1995-06-06 | 1996-12-12 | Pfizer Inc. | Substituted n-(indole-2-carbonyl-) amides and derivatives as glycogen phosphorylase inhibitors |
| WO1996039384A1 (en) * | 1995-06-06 | 1996-12-12 | Pfizer, Inc. | Substituted n-(indole-2-carbonyl)-glycinamides and derivatives as glycogen phosphorylase inhibitors |
-
2000
- 2000-05-05 US US09/565,523 patent/US6410750B1/en not_active Expired - Fee Related
- 2000-06-12 IL IL13672600A patent/IL136726A0/xx unknown
- 2000-06-14 ZA ZA200002987A patent/ZA200002987B/xx unknown
- 2000-06-14 IN IN552MU2000 patent/IN188853B/en unknown
- 2000-06-14 EP EP00305048A patent/EP1061074A1/en not_active Withdrawn
- 2000-06-15 JP JP2000179880A patent/JP3342471B2/ja not_active Expired - Fee Related
- 2000-06-16 TR TR2000/01781A patent/TR200001781A2/xx unknown
- 2000-06-16 YU YU38000A patent/YU38000A/sh unknown
- 2000-06-16 CN CN00118397A patent/CN1283615A/zh active Pending
- 2000-06-16 KR KR1020000033140A patent/KR20010049559A/ko not_active Ceased
- 2000-06-16 ID IDP20000495D patent/ID26385A/id unknown
- 2000-06-16 HU HU0002285A patent/HUP0002285A3/hu unknown
- 2000-06-16 CA CA002311872A patent/CA2311872A1/en not_active Abandoned
- 2000-06-16 AU AU40892/00A patent/AU4089200A/en not_active Abandoned
- 2000-06-16 CZ CZ20002242A patent/CZ20002242A3/cs unknown
- 2000-06-16 RU RU2000115273/04A patent/RU2195450C2/ru not_active IP Right Cessation
- 2000-06-19 BR BR0002686-7A patent/BR0002686A/pt not_active IP Right Cessation
- 2000-06-19 PL PL00340866A patent/PL340866A1/xx not_active Application Discontinuation
Patent Citations (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO1996039385A1 (en) * | 1995-06-06 | 1996-12-12 | Pfizer Inc. | Substituted n-(indole-2-carbonyl-) amides and derivatives as glycogen phosphorylase inhibitors |
| WO1996039384A1 (en) * | 1995-06-06 | 1996-12-12 | Pfizer, Inc. | Substituted n-(indole-2-carbonyl)-glycinamides and derivatives as glycogen phosphorylase inhibitors |
Also Published As
| Publication number | Publication date |
|---|---|
| ID26385A (id) | 2000-12-21 |
| HUP0002285A2 (en) | 2001-03-28 |
| HU0002285D0 (en) | 2000-08-28 |
| IL136726A0 (en) | 2001-06-14 |
| TR200001781A2 (tr) | 2001-01-22 |
| CN1283615A (zh) | 2001-02-14 |
| CZ20002242A3 (cs) | 2002-01-16 |
| IN188853B (enExample) | 2002-11-16 |
| PL340866A1 (en) | 2001-01-02 |
| JP3342471B2 (ja) | 2002-11-11 |
| ZA200002987B (en) | 2001-12-14 |
| KR20010049559A (ko) | 2001-06-15 |
| CA2311872A1 (en) | 2000-12-18 |
| AU4089200A (en) | 2000-12-21 |
| YU38000A (sh) | 2003-02-28 |
| EP1061074A1 (en) | 2000-12-20 |
| US6410750B1 (en) | 2002-06-25 |
| BR0002686A (pt) | 2001-08-21 |
| HUP0002285A3 (en) | 2002-09-30 |
| JP2001039949A (ja) | 2001-02-13 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| MM4A | The patent is invalid due to non-payment of fees |
Effective date: 20030617 |