HUP0002285A3 - Process for preparing 3(s)[(5-chloro-1h-indole-2-carbonyl)-amino]-2(r)-hydroxy-4-phenyl-butyric acid and intermediates - Google Patents

Process for preparing 3(s)[(5-chloro-1h-indole-2-carbonyl)-amino]-2(r)-hydroxy-4-phenyl-butyric acid and intermediates

Info

Publication number
HUP0002285A3
HUP0002285A3 HU0002285A HUP0002285A HUP0002285A3 HU P0002285 A3 HUP0002285 A3 HU P0002285A3 HU 0002285 A HU0002285 A HU 0002285A HU P0002285 A HUP0002285 A HU P0002285A HU P0002285 A3 HUP0002285 A3 HU P0002285A3
Authority
HU
Hungary
Prior art keywords
indole
intermediates
carbonyl
chloro
hydroxy
Prior art date
Application number
HU0002285A
Other languages
English (en)
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Publication of HU0002285D0 publication Critical patent/HU0002285D0/hu
Publication of HUP0002285A2 publication Critical patent/HUP0002285A2/hu
Publication of HUP0002285A3 publication Critical patent/HUP0002285A3/hu

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04—Indoles; Hydrogenated indoles
    • C07D209/10—Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
    • C07D209/12—Radicals substituted by oxygen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C229/00—Compounds containing amino and carboxyl groups bound to the same carbon skeleton
    • C07C229/02—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton
    • C07C229/34—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton containing six-membered aromatic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04—Indoles; Hydrogenated indoles
    • C07D209/30—Indoles; Hydrogenated indoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to carbon atoms of the hetero ring
    • C07D209/42—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00—Indexing scheme relating to specific properties of organic compounds
    • C07B2200/07—Optical isomers

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Indole Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
HU0002285A 1999-06-18 2000-06-16 Process for preparing 3(s)[(5-chloro-1h-indole-2-carbonyl)-amino]-2(r)-hydroxy-4-phenyl-butyric acid and intermediates HUP0002285A3 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US13999799P 1999-06-18 1999-06-18

Publications (3)

Publication Number Publication Date
HU0002285D0 HU0002285D0 (en) 2000-08-28
HUP0002285A2 HUP0002285A2 (en) 2001-03-28
HUP0002285A3 true HUP0002285A3 (en) 2002-09-30

Family

ID=22489263

Family Applications (1)

Application Number Title Priority Date Filing Date
HU0002285A HUP0002285A3 (en) 1999-06-18 2000-06-16 Process for preparing 3(s)[(5-chloro-1h-indole-2-carbonyl)-amino]-2(r)-hydroxy-4-phenyl-butyric acid and intermediates

Country Status (18)

Country Link
US (1) US6410750B1 (hu)
EP (1) EP1061074A1 (hu)
JP (1) JP3342471B2 (hu)
KR (1) KR20010049559A (hu)
CN (1) CN1283615A (hu)
AU (1) AU4089200A (hu)
BR (1) BR0002686A (hu)
CA (1) CA2311872A1 (hu)
CZ (1) CZ20002242A3 (hu)
HU (1) HUP0002285A3 (hu)
ID (1) ID26385A (hu)
IL (1) IL136726A0 (hu)
IN (1) IN188853B (hu)
PL (1) PL340866A1 (hu)
RU (1) RU2195450C2 (hu)
TR (1) TR200001781A2 (hu)
YU (1) YU38000A (hu)
ZA (1) ZA200002987B (hu)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7759487B2 (en) * 2005-01-06 2010-07-20 Schering Corporation Preparation of ketone amides
EP2714660B1 (en) * 2011-05-31 2018-09-26 Theravance Biopharma R&D IP, LLC Neprilysin inhibitors

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2223625C (en) 1995-06-06 2003-06-03 Pfizer Inc. Substituted n-(indole-2-carbonyl-) amides and derivatives as glycogen phosphorylase inhibitors
CA2224062C (en) 1995-06-06 2001-09-04 Pfizer Limited Substituted n-(indole-2-carbonyl)-glycinamides and derivatives as glycogen phosphorylase inhibitors

Also Published As

Publication number Publication date
TR200001781A2 (tr) 2001-01-22
HU0002285D0 (en) 2000-08-28
EP1061074A1 (en) 2000-12-20
KR20010049559A (ko) 2001-06-15
IN188853B (hu) 2002-11-16
CA2311872A1 (en) 2000-12-18
ZA200002987B (en) 2001-12-14
CZ20002242A3 (cs) 2002-01-16
RU2195450C2 (ru) 2002-12-27
HUP0002285A2 (en) 2001-03-28
BR0002686A (pt) 2001-08-21
JP3342471B2 (ja) 2002-11-11
CN1283615A (zh) 2001-02-14
IL136726A0 (en) 2001-06-14
US6410750B1 (en) 2002-06-25
PL340866A1 (en) 2001-01-02
JP2001039949A (ja) 2001-02-13
ID26385A (id) 2000-12-21
AU4089200A (en) 2000-12-21
YU38000A (sh) 2003-02-28

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