RU2019110821A - Антагонисты trpv4 - Google Patents

Антагонисты trpv4 Download PDF

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Publication number
RU2019110821A
RU2019110821A RU2019110821A RU2019110821A RU2019110821A RU 2019110821 A RU2019110821 A RU 2019110821A RU 2019110821 A RU2019110821 A RU 2019110821A RU 2019110821 A RU2019110821 A RU 2019110821A RU 2019110821 A RU2019110821 A RU 2019110821A
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RU
Russia
Prior art keywords
sulfonyl
hydroxymethyl
pyrrolidin
hydroxy
benzonitrile
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RU2019110821A
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English (en)
Russian (ru)
Inventor
Эдвард Дж. БРНАРДИК
Карл А. БРУКС
Брайан Гриффин Лоухорн
Пэн ЛИ
Джей М. Мэттьюз
Джон Джеффри МАКЭЙТИ
Мэттью Роберт СЕНДЕР
Ламонт Роско ТЕРРЕЛЛ
Джозеф Е. ПЕРО
Дэвид Дж. БЕХМ
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Глэксосмитклайн Интеллекчуал Проперти (Но.2) Лимитед
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Publication of RU2019110821A publication Critical patent/RU2019110821A/ru

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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
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    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
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RU2019110821A 2016-09-20 2017-09-20 Антагонисты trpv4 RU2019110821A (ru)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US201662397008P 2016-09-20 2016-09-20
US62/397,008 2016-09-20
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