RU2015152566A - Ингибиторы кетогексокиназы на растительной основе для поддержания управления весом - Google Patents

Ингибиторы кетогексокиназы на растительной основе для поддержания управления весом Download PDF

Info

Publication number
RU2015152566A
RU2015152566A RU2015152566A RU2015152566A RU2015152566A RU 2015152566 A RU2015152566 A RU 2015152566A RU 2015152566 A RU2015152566 A RU 2015152566A RU 2015152566 A RU2015152566 A RU 2015152566A RU 2015152566 A RU2015152566 A RU 2015152566A
Authority
RU
Russia
Prior art keywords
composition
plant extract
plant
group
subject
Prior art date
Application number
RU2015152566A
Other languages
English (en)
Russian (ru)
Inventor
Ятиндер РАНА
Русселл Кеит РАНДОЛФ
Джеффрей ЩОЛТЕН
Мыфуонг Тхи ЛЕ
Ричард Дж. ДЖОНСОН
Гарсиа Мигуел Ангел ЛАНАСПА
Original Assignee
Ассесс Бузинесс Груп Интернэшнл Ллс
Де Регентс Оф Де Юниверсити Оф Колорадо, А Боды Корпорейт
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ассесс Бузинесс Груп Интернэшнл Ллс, Де Регентс Оф Де Юниверсити Оф Колорадо, А Боды Корпорейт filed Critical Ассесс Бузинесс Груп Интернэшнл Ллс
Publication of RU2015152566A publication Critical patent/RU2015152566A/ru

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K36/00Medicinal preparations of undetermined constitution containing material from algae, lichens, fungi or plants, or derivatives thereof, e.g. traditional herbal medicines
    • A61K36/18Magnoliophyta (angiosperms)
    • A61K36/185Magnoliopsida (dicotyledons)
    • A61K36/73Rosaceae (Rose family), e.g. strawberry, chokeberry, blackberry, pear or firethorn
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K36/00Medicinal preparations of undetermined constitution containing material from algae, lichens, fungi or plants, or derivatives thereof, e.g. traditional herbal medicines
    • A61K36/11Pteridophyta or Filicophyta (ferns)
    • A61K36/12Filicopsida or Pteridopsida
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K36/00Medicinal preparations of undetermined constitution containing material from algae, lichens, fungi or plants, or derivatives thereof, e.g. traditional herbal medicines
    • A61K36/18Magnoliophyta (angiosperms)
    • A61K36/185Magnoliopsida (dicotyledons)
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K36/00Medicinal preparations of undetermined constitution containing material from algae, lichens, fungi or plants, or derivatives thereof, e.g. traditional herbal medicines
    • A61K36/18Magnoliophyta (angiosperms)
    • A61K36/185Magnoliopsida (dicotyledons)
    • A61K36/19Acanthaceae (Acanthus family)
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K36/00Medicinal preparations of undetermined constitution containing material from algae, lichens, fungi or plants, or derivatives thereof, e.g. traditional herbal medicines
    • A61K36/18Magnoliophyta (angiosperms)
    • A61K36/185Magnoliopsida (dicotyledons)
    • A61K36/23Apiaceae or Umbelliferae (Carrot family), e.g. dill, chervil, coriander or cumin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K36/00Medicinal preparations of undetermined constitution containing material from algae, lichens, fungi or plants, or derivatives thereof, e.g. traditional herbal medicines
    • A61K36/18Magnoliophyta (angiosperms)
    • A61K36/185Magnoliopsida (dicotyledons)
    • A61K36/23Apiaceae or Umbelliferae (Carrot family), e.g. dill, chervil, coriander or cumin
    • A61K36/232Angelica
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K36/00Medicinal preparations of undetermined constitution containing material from algae, lichens, fungi or plants, or derivatives thereof, e.g. traditional herbal medicines
    • A61K36/18Magnoliophyta (angiosperms)
    • A61K36/185Magnoliopsida (dicotyledons)
    • A61K36/38Clusiaceae, Hypericaceae or Guttiferae (Hypericum or Mangosteen family), e.g. common St. Johnswort
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K36/00Medicinal preparations of undetermined constitution containing material from algae, lichens, fungi or plants, or derivatives thereof, e.g. traditional herbal medicines
    • A61K36/18Magnoliophyta (angiosperms)
    • A61K36/185Magnoliopsida (dicotyledons)
    • A61K36/44Ebenaceae (Ebony family), e.g. persimmon
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K36/00Medicinal preparations of undetermined constitution containing material from algae, lichens, fungi or plants, or derivatives thereof, e.g. traditional herbal medicines
    • A61K36/18Magnoliophyta (angiosperms)
    • A61K36/185Magnoliopsida (dicotyledons)
    • A61K36/48Fabaceae or Leguminosae (Pea or Legume family); Caesalpiniaceae; Mimosaceae; Papilionaceae
    • A61K36/487Psoralea
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K36/00Medicinal preparations of undetermined constitution containing material from algae, lichens, fungi or plants, or derivatives thereof, e.g. traditional herbal medicines
    • A61K36/18Magnoliophyta (angiosperms)
    • A61K36/185Magnoliopsida (dicotyledons)
    • A61K36/53Lamiaceae or Labiatae (Mint family), e.g. thyme, rosemary or lavender
    • A61K36/539Scutellaria (skullcap)
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K36/00Medicinal preparations of undetermined constitution containing material from algae, lichens, fungi or plants, or derivatives thereof, e.g. traditional herbal medicines
    • A61K36/18Magnoliophyta (angiosperms)
    • A61K36/185Magnoliopsida (dicotyledons)
    • A61K36/60Moraceae (Mulberry family), e.g. breadfruit or fig
    • A61K36/605Morus (mulberry)
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K36/00Medicinal preparations of undetermined constitution containing material from algae, lichens, fungi or plants, or derivatives thereof, e.g. traditional herbal medicines
    • A61K36/18Magnoliophyta (angiosperms)
    • A61K36/185Magnoliopsida (dicotyledons)
    • A61K36/62Nymphaeaceae (Water-lily family)
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K36/00Medicinal preparations of undetermined constitution containing material from algae, lichens, fungi or plants, or derivatives thereof, e.g. traditional herbal medicines
    • A61K36/18Magnoliophyta (angiosperms)
    • A61K36/185Magnoliopsida (dicotyledons)
    • A61K36/75Rutaceae (Rue family)
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/04Anorexiants; Antiobesity agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Natural Medicines & Medicinal Plants (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Epidemiology (AREA)
  • Medical Informatics (AREA)
  • Microbiology (AREA)
  • Mycology (AREA)
  • Botany (AREA)
  • Biotechnology (AREA)
  • Alternative & Traditional Medicine (AREA)
  • Diabetes (AREA)
  • Organic Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Neurosurgery (AREA)
  • Emergency Medicine (AREA)
  • Endocrinology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Medicines Containing Plant Substances (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
RU2015152566A 2013-06-19 2014-06-16 Ингибиторы кетогексокиназы на растительной основе для поддержания управления весом RU2015152566A (ru)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201361836843P 2013-06-19 2013-06-19
US61/836,843 2013-06-19
PCT/US2014/042534 WO2014204853A1 (en) 2013-06-19 2014-06-16 Plant-based inhibitors of ketohexokinase for the support of weight management

Publications (1)

Publication Number Publication Date
RU2015152566A true RU2015152566A (ru) 2017-07-20

Family

ID=51136839

Family Applications (1)

Application Number Title Priority Date Filing Date
RU2015152566A RU2015152566A (ru) 2013-06-19 2014-06-16 Ингибиторы кетогексокиназы на растительной основе для поддержания управления весом

Country Status (10)

Country Link
US (1) US20140377386A1 (https=)
EP (1) EP3010520A1 (https=)
JP (1) JP2016522255A (https=)
KR (1) KR20160020472A (https=)
CN (1) CN105555287A (https=)
AU (1) AU2014281768A1 (https=)
HK (1) HK1224201A1 (https=)
RU (1) RU2015152566A (https=)
TW (1) TW201534315A (https=)
WO (1) WO2014204853A1 (https=)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN107375256A (zh) * 2017-09-13 2017-11-24 上海壹志医药科技有限公司 根皮素的药物用途
WO2020166494A1 (ja) * 2019-02-15 2020-08-20 国立大学法人信州大学 血圧低下作用を有するナス由来組成物
CN110025603A (zh) * 2019-05-15 2019-07-19 大连天星本草生物科技有限公司 补骨脂查尔酮类化合物在制备治疗肥胖症的药物中的应用

Family Cites Families (26)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5282710A (en) * 1975-12-29 1977-07-11 Nippon Shinyaku Co Ltd Extraction of effective drug component from mulberry
JP2001513571A (ja) * 1997-08-29 2001-09-04 ザ リセックス カンパニー インコーポレイテッド 糖尿病、高血糖症及び低血糖症の治療法
ATE369868T1 (de) * 2000-06-27 2007-09-15 Qualilife Pharmaceuticals Inc Zusammensetzungen und verfahren zur behandlung der weiblichen sexuellen reaktion
JP2002138045A (ja) * 2000-10-30 2002-05-14 Ichimaru Pharcos Co Ltd 前駆脂肪細胞分化誘導剤
WO2005009351A2 (en) * 2003-07-17 2005-02-03 Santé International, Inc. Dietary supplement for promoting control of blood-sugar levels and associated pathology in type 2 diabetics
CN1921872A (zh) * 2004-02-03 2007-02-28 智利南方大学 用于激活PPR-γ受体而治疗自身免疫性疾病和阿尔茨海默病的提取自穿心莲的半日花烷型二萜类组合物
JP2006273788A (ja) * 2005-03-30 2006-10-12 Kaneka Corp Pparリガンド活性を有する植物由来の組成物
KR101802415B1 (ko) * 2005-05-09 2017-11-28 유니젠, 인크. 바쿠치올의 조성물 및 그것의 제조방법
JP2008133192A (ja) * 2005-09-29 2008-06-12 Kureha Corp 抗糖尿病剤
CN101835480B (zh) * 2007-10-24 2013-06-12 三得利控股株式会社 单子山楂乙醇提取物在制备预防及/或改善肥胖的组合物中的用途
JP5450952B2 (ja) * 2007-11-27 2014-03-26 安幸 城田 健康飲食物及び薬剤
US20090252758A1 (en) * 2008-04-07 2009-10-08 Mazed Mohammad A Nutritional supplement for the prevention of cardiovascular disease, alzheimer's disease, diabetes, and regulation and reduction of blood sugar and insulin resistance
JP2009298742A (ja) * 2008-06-16 2009-12-24 Toyobo Co Ltd 生活習慣病改善剤
US20100055247A1 (en) * 2008-08-29 2010-03-04 Tirrito Salvatore J Nutritional Compositions for Athletes
JP2010083838A (ja) * 2008-10-02 2010-04-15 Ichimaru Pharcos Co Ltd アディポネクチン産生促進剤
US20100215782A1 (en) * 2008-10-22 2010-08-26 Metaproteomics, Llc Novel mitochondrial uncoupling methods and compositions for enhancing adipocyte thermogenesis
KR101746867B1 (ko) * 2009-01-26 2017-06-14 타이페이 메디컬 유니이버시티 당뇨 및 비만을 치료하기 위한 프테로신 화합물의 용도
CA2751227C (en) * 2009-02-02 2021-10-26 Laila Nutraceuticals Composition from sphaeranthus indicus and garcinia mangostana for the control of metabolic syndrome
CN101642477A (zh) * 2009-08-28 2010-02-10 李来杰 中药凤尾草的用途
JP2011079752A (ja) * 2009-10-05 2011-04-21 Kracie Home Products Ltd 膵リパーゼ阻害剤並びにそれを含有する飲食品組成物及び医薬品組成物
JP2011168547A (ja) * 2010-02-19 2011-09-01 Sun Foods Co Ltd α−グルコシダ−ゼ活性阻害剤、及びこれを含有する果実飲料
JP2013525370A (ja) * 2010-04-22 2013-06-20 ヤンセン ファーマシューティカ エヌ.ベー. ケトヘキソキナーゼ阻害剤として有用なインダゾール化合物
CN101856351B (zh) * 2010-05-28 2012-05-30 暨南大学 一种组合物及其在制备rxr受体转录抑制剂中的应用
KR20120031800A (ko) * 2010-09-27 2012-04-04 농업회사법인 주식회사 상로 뽕나무 열매 씨앗 추출물을 함유하는 항산화, 항당뇨 및 항노화 활성 조성물
WO2013085338A2 (ko) * 2011-12-07 2013-06-13 한국생명공학연구원 수련뿌리 추출물, 이의 분획물 또는 이로부터 분리된 폴리페놀계 화합물을 유효성분으로 함유하는 대사성 질환 예방 및 치료용 약학적 조성물
EP3549587A1 (de) * 2012-06-30 2019-10-09 BioActive Food GmbH Zusammensetzung zur behandlung von hyperglykämischen erkrankungen

Also Published As

Publication number Publication date
AU2014281768A1 (en) 2015-12-24
EP3010520A1 (en) 2016-04-27
WO2014204853A1 (en) 2014-12-24
KR20160020472A (ko) 2016-02-23
TW201534315A (zh) 2015-09-16
JP2016522255A (ja) 2016-07-28
US20140377386A1 (en) 2014-12-25
CN105555287A (zh) 2016-05-04
HK1224201A1 (zh) 2017-08-18

Similar Documents

Publication Publication Date Title
JP2023133599A (ja) 皮膚障害改善用組成物
JPWO2012096276A1 (ja) 経皮吸収促進剤及び皮膚外用剤
EA201490396A1 (ru) Ингибиторы репликации вирусов гриппа
HRP20191285T1 (hr) Predlijekovi karbidopa i l-dopa te njihova uporaba za liječenje parkinsonove bolesti
MX361350B (es) Compuestos heterocíclicos fusionados como moduladores del canal de sodio.
RU2015152566A (ru) Ингибиторы кетогексокиназы на растительной основе для поддержания управления весом
CN110946948A (zh) 化风丹在制备抗乳腺癌药物中的应用
EA201000340A1 (ru) Аминобензилзамещенные циклические сульфоны, полезные в качестве ингибиторов васе
de Molon Therapeutic potential of tanshinones in osteolytic diseases: from molecular and cellular pathways to preclinical models
NO20090067L (no) Farmasoytiske kombinasjoner for behandling av respiratoriske sykdommer
CN103304607B (zh) 从窄叶鲜卑花降脂减肥有效部位得到的单萜苷化合物及其应用
RU2015113031A (ru) Использование 3-n-бутил изоиндолин кетонов при приготовлении лекарственных средств для профилактики и лечения церебрального инфаркта
JP2010132632A (ja) タンパク質糖化抑制剤
CN119564682A (zh) 一种锌离子螯合剂在唑类药物抗白念珠菌生物膜中的应用
CA2884644A1 (en) Tetrandrine pharmaceutical formulations and method
Gayathiri et al. In silico and in vitro approaches to evaluate the bioactivities of Chaetomorpha linum
JP2016522255A5 (https=)
EA201300882A1 (ru) Способ лечения констипации и/или уплотнения фекальных масс, водный раствор для лечения констипации и/или уплотнения фекальных масс (варианты), набор и лекарственное средство
US20250082658A1 (en) Cell proliferation retardant, cosmetic containing same, and cell proliferation retardation method
JP6272814B2 (ja) ヒアルロン酸産生促進剤
JP5716173B2 (ja) 病原性因子産生抑制剤
CN101385737A (zh) 一种抗菌有效成分及其应用
BRPI0409790A (pt) 7-azaindóis e seu uso como terapêuticos
BRPI0409793A (pt) 4-,6- ou 7-hidroxiindóis com grupos n-óxido e sua aplicação como produtos terapêuticos
EA201491995A1 (ru) Пероральная лекарственная форма