RU2004111359A - Комбинированные агенты для лечения глаукомы - Google Patents

Комбинированные агенты для лечения глаукомы Download PDF

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Publication number
RU2004111359A
RU2004111359A RU2004111359/15A RU2004111359A RU2004111359A RU 2004111359 A RU2004111359 A RU 2004111359A RU 2004111359/15 A RU2004111359/15 A RU 2004111359/15A RU 2004111359 A RU2004111359 A RU 2004111359A RU 2004111359 A RU2004111359 A RU 2004111359A
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Russia
Prior art keywords
treatment
glaucoma
prevention
active ingredients
combination
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RU2004111359/15A
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English (en)
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Томихиса ЙОКОЯМА (JP)
Томихиса ЙОКОЯМА
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Санкио Компани, Лимитед (Jp)
Санкио Компани, Лимитед
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Application filed by Санкио Компани, Лимитед (Jp), Санкио Компани, Лимитед filed Critical Санкио Компани, Лимитед (Jp)
Publication of RU2004111359A publication Critical patent/RU2004111359A/ru

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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/415—1,2-Diazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/557—Eicosanoids, e.g. leukotrienes or prostaglandins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A61P27/06—Antiglaucoma agents or miotics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives

Landscapes

  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Ophthalmology & Optometry (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
  • Saccharide Compounds (AREA)

Claims (3)

1. Комбинация для профилактики или лечения глаукомы, которая включает антагонист ангиотензина II и тимолол малеат в качестве активных ингредиентов, для одновременного, раздельного или последовательного использования указанных активных ингредиентов, где антагонист ангиотензина II представляет собой соединение формулы (I) или его фармакологически приемлемую соль, сложный эфир или другое производное:
Figure 00000001
где R1 представляет группу, имеющую структурную формулу (Ia):
Figure 00000002
2. Комбинация для профилактики или лечения глаукомы по п. 1, которая находится в форме, удобной для местного нанесения в глаза.
3. Способ профилактики или лечения глаукомы, который включает введение пациенту комбинации для профилактики или лечения глаукомы по п.1 или 2.
RU2004111359/15A 1999-12-01 2004-04-13 Комбинированные агенты для лечения глаукомы RU2004111359A (ru)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
JP11/341524 1999-12-01
JP34152499 1999-12-01
JP2000078769 2000-03-21
JP2000-78769 2000-03-21

Related Parent Applications (1)

Application Number Title Priority Date Filing Date
RU2002114335/15A Division RU2002114335A (ru) 1999-12-01 2000-12-01 Комбинированные агенты для лечения глаукомы

Publications (1)

Publication Number Publication Date
RU2004111359A true RU2004111359A (ru) 2005-09-20

Family

ID=26576988

Family Applications (4)

Application Number Title Priority Date Filing Date
RU2002114335/15A RU2002114335A (ru) 1999-12-01 2000-12-01 Комбинированные агенты для лечения глаукомы
RU2004111357/15A RU2299067C2 (ru) 1999-12-01 2004-04-13 Комбинированные агенты для лечения глаукомы
RU2004111359/15A RU2004111359A (ru) 1999-12-01 2004-04-13 Комбинированные агенты для лечения глаукомы
RU2004111358/15A RU2004111358A (ru) 1999-12-01 2004-04-13 Комбинированные агенты для лечения глаукомы

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RU2004111357/15A RU2299067C2 (ru) 1999-12-01 2004-04-13 Комбинированные агенты для лечения глаукомы

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US (4) US7307096B2 (ru)
EP (3) EP1344535A3 (ru)
JP (1) JP4000505B2 (ru)
KR (3) KR20040045028A (ru)
CN (3) CN1615879A (ru)
AT (1) ATE332145T1 (ru)
AU (1) AU773110B2 (ru)
BR (1) BR0015980A (ru)
CA (1) CA2392804C (ru)
CZ (1) CZ20021829A3 (ru)
DE (1) DE60029242T2 (ru)
ES (1) ES2267586T3 (ru)
HK (1) HK1047239B (ru)
HU (1) HUP0204049A3 (ru)
IL (2) IL149444A0 (ru)
MX (1) MXPA02005505A (ru)
NO (1) NO20022584L (ru)
NZ (1) NZ518930A (ru)
PL (1) PL201783B1 (ru)
RU (4) RU2002114335A (ru)
TW (1) TWI290470B (ru)
WO (1) WO2001039805A1 (ru)

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Publication number Publication date
ATE332145T1 (de) 2006-07-15
HK1047239B (zh) 2006-12-08
DE60029242T2 (de) 2007-07-05
EP1344534A2 (en) 2003-09-17
EP1234582B1 (en) 2006-07-05
HUP0204049A3 (en) 2006-07-28
NO20022584L (no) 2002-07-29
EP1344535A3 (en) 2004-01-28
RU2004111357A (ru) 2005-09-20
NZ518930A (en) 2003-09-26
KR20040045029A (ko) 2004-05-31
CN1407903A (zh) 2003-04-02
TWI290470B (en) 2007-12-01
US20080221184A1 (en) 2008-09-11
IL149444A0 (en) 2002-11-10
CZ20021829A3 (cs) 2002-08-14
CN1615880A (zh) 2005-05-18
KR100607430B1 (ko) 2006-08-02
HUP0204049A2 (hu) 2003-04-28
BR0015980A (pt) 2002-11-12
RU2004111358A (ru) 2005-09-20
AU1557501A (en) 2001-06-12
CA2392804A1 (en) 2001-06-07
ES2267586T3 (es) 2007-03-16
EP1234582A1 (en) 2002-08-28
CA2392804C (en) 2009-02-03
EP1234582A4 (en) 2003-05-07
KR20040045028A (ko) 2004-05-31
DE60029242D1 (de) 2006-08-17
RU2299067C2 (ru) 2007-05-20
RU2002114335A (ru) 2004-01-10
EP1344535A2 (en) 2003-09-17
PL201783B1 (pl) 2009-05-29
US20050014808A1 (en) 2005-01-20
US20050043383A1 (en) 2005-02-24
AU773110B2 (en) 2004-05-20
JP4000505B2 (ja) 2007-10-31
HK1047239A1 (en) 2003-02-14
WO2001039805A1 (fr) 2001-06-07
JP2001335511A (ja) 2001-12-04
CN1615879A (zh) 2005-05-18
IL149444A (en) 2007-06-17
MXPA02005505A (es) 2002-09-02
NO20022584D0 (no) 2002-05-31
CN1263512C (zh) 2006-07-12
US7307096B2 (en) 2007-12-11
EP1344534A3 (en) 2004-01-02
PL355431A1 (en) 2004-04-19
KR20020058034A (ko) 2002-07-12
US20030040529A1 (en) 2003-02-27

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