RS20050931A - Novel lincomycin derivatives possessing antimicro bial activity - Google Patents

Novel lincomycin derivatives possessing antimicro bial activity

Info

Publication number
RS20050931A
RS20050931A YUP-2005/0931A YUP20050931A RS20050931A RS 20050931 A RS20050931 A RS 20050931A YU P20050931 A YUP20050931 A YU P20050931A RS 20050931 A RS20050931 A RS 20050931A
Authority
RS
Serbia
Prior art keywords
lincomycin derivatives
derivatives possessing
novel
novel lincomycin
activity
Prior art date
Application number
YUP-2005/0931A
Other languages
English (en)
Serbian (sr)
Inventor
Mikhail Gordeev
Jason Lewis
Sampath Anandan
Hardwin O'Dowd
Original Assignee
Vicuron Pharmaceuticals Inc.,
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US10/642,807 external-priority patent/US7164011B2/en
Priority claimed from US10/777,455 external-priority patent/US7199105B2/en
Application filed by Vicuron Pharmaceuticals Inc., filed Critical Vicuron Pharmaceuticals Inc.,
Publication of RS20050931A publication Critical patent/RS20050931A/sr

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/70—Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7042—Compounds having saccharide radicals and heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/70—Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7042—Compounds having saccharide radicals and heterocyclic rings
    • A61K31/7052—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/02—Acyclic radicals, not substituted by cyclic structures
    • C07H15/14—Acyclic radicals, not substituted by cyclic structures attached to a sulfur, selenium or tellurium atom of a saccharide radical
    • C07H15/16—Lincomycin; Derivatives thereof
YUP-2005/0931A 2003-06-17 2004-06-17 Novel lincomycin derivatives possessing antimicro bial activity RS20050931A (en)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US47929603P 2003-06-17 2003-06-17
US47950203P 2003-06-17 2003-06-17
US10/642,807 US7164011B2 (en) 2002-08-15 2003-08-15 Lincomycin derivatives possessing antibacterial activity
US10/777,455 US7199105B2 (en) 2002-08-15 2004-02-11 Lincomycin derivatives possessing antibacterial activity
PCT/US2004/019689 WO2005012320A2 (en) 2003-06-17 2004-06-17 Novel lincomycin derivatives possessing antimicrobial activity

Publications (1)

Publication Number Publication Date
RS20050931A true RS20050931A (en) 2008-04-04

Family

ID=40203032

Family Applications (1)

Application Number Title Priority Date Filing Date
YUP-2005/0931A RS20050931A (en) 2003-06-17 2004-06-17 Novel lincomycin derivatives possessing antimicro bial activity

Country Status (17)

Country Link
EP (1) EP1644393A2 (ja)
JP (1) JP2007516172A (ja)
KR (1) KR20060091050A (ja)
AU (1) AU2004261550A1 (ja)
BR (1) BRPI0411534A (ja)
CA (1) CA2528592A1 (ja)
EC (1) ECSP056233A (ja)
GE (1) GEP20084437B (ja)
HK (1) HK1090061A1 (ja)
IL (1) IL172183A0 (ja)
IS (1) IS8147A (ja)
MA (1) MA27860A1 (ja)
MX (1) MXPA05013915A (ja)
NO (1) NO20055893L (ja)
OA (1) OA13179A (ja)
RS (1) RS20050931A (ja)
WO (1) WO2005012320A2 (ja)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7199105B2 (en) 2002-08-15 2007-04-03 Vicuron Pharmaceuticals, Inc. Lincomycin derivatives possessing antibacterial activity
EA200500353A1 (ru) 2002-08-15 2006-06-30 Вайкьюрон Фармасьютикалз, Инк. Производные линкомицина, обладающие антибактериальной активностью
US7199106B2 (en) 2003-06-17 2007-04-03 Vicuron Pharmaceuticals, Inc. Lincomycin derivatives possessing antimicrobial activity
WO2005007665A2 (en) * 2003-06-17 2005-01-27 Vicuron Pharmaceuticals Inc. Lincomycin derivatives possessing antibacterial activity
US7256177B2 (en) 2003-06-17 2007-08-14 Vicuron Pharmaceuticals, Inc. Lincomycin derivatives possessing antibacterial activity
US7361743B2 (en) 2004-02-11 2008-04-22 Pfizer Inc Lincomycin derivatives possessing antibacterial activity
CN101291916A (zh) * 2005-08-31 2008-10-22 惠氏公司 甘氨酰环素的9-氨基羰基取代衍生物
JP5064237B2 (ja) 2005-12-09 2012-10-31 Ｍｅｉｊｉ Ｓｅｉｋａファルマ株式会社 リンコマイシン誘導体およびこれを有効成分とする抗菌剤
US7867980B2 (en) 2007-05-31 2011-01-11 Meiji Seika Kaisha, Ltd. Lincosamide derivatives and antimicrobial agents comprising the same as active ingredient
EP2151447A4 (en) * 2007-05-31 2012-09-05 Meiji Seika Kaisha LINCOMYCIN DERIVATIVES AND ANTIBACTERIAL AGENTS CONTAINING SAME AS ACTIVE INGREDIENTS
US20130267699A1 (en) 2011-06-24 2013-10-10 California Institute Of Technology Quaternary heteroatom containing compounds
US8822679B2 (en) * 2011-06-24 2014-09-02 California Institute Of Technology Quaternary heteroatom containing compounds
US10421696B2 (en) 2014-12-18 2019-09-24 California Institute Of Technology Enantioselective synthesis of α-quaternary mannich adducts by palladium-catalyzed allylic alkylation
EP3274342B1 (en) 2015-03-27 2022-05-04 California Institute of Technology Asymmetric catalytic decarboxylative alkyl alkylation using low catalyst concentrations and a robust precatalyst
WO2017156239A1 (en) 2016-03-11 2017-09-14 California Institute Of Technology Compositions and methods for acylating lactams
EP3480190B1 (en) 2017-11-01 2023-01-04 California Institute of Technology Methods for enantioselective allylic alkylation of esters, lactones, and lactams with unactivated allylic alcohols
EP3699173A1 (en) 2018-10-18 2020-08-26 California Institute of Technology Gem-disubstituted pyrrolidines, piperazines, and diazepanes, and compositions and methods of making the same
CN110357839A (zh) * 2019-08-29 2019-10-22 重庆经致制药技术开发有限公司 布瓦西坦手性中间体的制备方法

Family Cites Families (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3268556A (en) * 1964-04-13 1966-08-23 Upjohn Co Novel lincomycin derivatives
NL128232C (ja) * 1964-04-13
NL146501C (ja) * 1964-07-01
US3282917A (en) * 1964-08-17 1966-11-01 Upjohn Co Methyl n-(1-alkyl-4-alkoxy-prolyl)-alpha-thiolincosaminide compounds and process therefor
US3496163A (en) * 1965-02-08 1970-02-17 Upjohn Co 7-halo-7-deoxylincomycins and process for preparing the same
NL140527B (nl) * 1965-02-08 1973-12-17 Upjohn Co Werkwijze ter bereiding van aan lincomycine verwante verbindingen.
US3555007A (en) * 1968-07-22 1971-01-12 Upjohn Co 7-deoxy-7-halo lincomycin d derivatives
US3549615A (en) * 1968-10-17 1970-12-22 Upjohn Co Lincomycin derivatives and process for producing the same
DE2118636A1 (de) * 1970-04-20 1971-11-04 The Upjohn Co., Kalamazoo, Mich. (V.StA.) 3-Nucleotide von Lincomycin und deren Analogen, Verfahren zu ihrer Herstellung und ihre Verwendung in therapeutischen Präparaten
US3787390A (en) * 1971-06-23 1974-01-22 Upjohn Co Analogs of lincomycin and process
US3849396A (en) * 1973-01-08 1974-11-19 Upjohn Co Lincomycin and clindamycin 1-o-ethers
US3923602A (en) * 1973-10-25 1975-12-02 Upjohn Co Composition of matter and process
JPS5641239A (en) * 1979-09-13 1981-04-17 Hitachi Cable Ltd Flame-retardant composition
US4278789A (en) * 1979-11-23 1981-07-14 The Upjohn Company Lincomycin compounds
EA200500353A1 (ru) * 2002-08-15 2006-06-30 Вайкьюрон Фармасьютикалз, Инк. Производные линкомицина, обладающие антибактериальной активностью
BRPI0411537A (pt) * 2003-06-17 2006-08-01 Vicuron Pharm Inc derivados de lincomicina que possuem atividade antibacteriana

Also Published As

Publication number Publication date
EP1644393A2 (en) 2006-04-12
GEP20084437B (en) 2008-07-25
ECSP056233A (es) 2006-04-19
HK1090061A1 (en) 2006-12-15
BRPI0411534A (pt) 2006-08-22
MA27860A1 (fr) 2006-04-03
WO2005012320A3 (en) 2005-10-20
NO20055893L (no) 2006-03-14
MXPA05013915A (es) 2006-07-03
JP2007516172A (ja) 2007-06-21
WO2005012320A2 (en) 2005-02-10
AU2004261550A1 (en) 2005-02-10
CA2528592A1 (en) 2005-02-10
IS8147A (is) 2005-11-24
OA13179A (en) 2006-12-13
IL172183A0 (en) 2011-08-01
KR20060091050A (ko) 2006-08-17

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