UY28542A1 - Amidas macrocíclicas antibacterianas - Google Patents
Amidas macrocíclicas antibacterianasInfo
- Publication number
- UY28542A1 UY28542A1 UY28542A UY28542A UY28542A1 UY 28542 A1 UY28542 A1 UY 28542A1 UY 28542 A UY28542 A UY 28542A UY 28542 A UY28542 A UY 28542A UY 28542 A1 UY28542 A1 UY 28542A1
- Authority
- UY
- Uruguay
- Prior art keywords
- amides
- antibacterial
- macrocyclic amides
- antibacterial macrocyclic
- prophylaxis
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/08—Tripeptides
- C07K5/0802—Tripeptides with the first amino acid being neutral
- C07K5/0812—Tripeptides with the first amino acid being neutral and aromatic or cycloaliphatic
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/02—Drugs for disorders of the endocrine system of the hypothalamic hormones, e.g. TRH, GnRH, CRH, GRH, somatostatin
- A61P5/04—Drugs for disorders of the endocrine system of the hypothalamic hormones, e.g. TRH, GnRH, CRH, GRH, somatostatin for decreasing, blocking or antagonising the activity of the hypothalamic hormones
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Animal Behavior & Ethology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Molecular Biology (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
- Genetics & Genomics (AREA)
- Biophysics (AREA)
- Biochemistry (AREA)
- Endocrinology (AREA)
- Diabetes (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Peptides Or Proteins (AREA)
Abstract
La invención se refiere a amidas macrocíclicas antivacterianas y a procedimientos para su preparación, a su uso para el tratamiento y/o la profilaxis de enfermedades, así comoa su uso para la preparación de medicamentos para el tratamiento y/o la profilaxis de enfermedades, especialmente de infecciones bacterianas.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE10345724 | 2003-10-01 | ||
DE10358822A DE10358822A1 (de) | 2003-10-01 | 2003-12-16 | Antibakterielle Amid-Makrozyklen |
Publications (1)
Publication Number | Publication Date |
---|---|
UY28542A1 true UY28542A1 (es) | 2005-04-29 |
Family
ID=34424312
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
UY28542A UY28542A1 (es) | 2003-10-01 | 2004-09-30 | Amidas macrocíclicas antibacterianas |
Country Status (5)
Country | Link |
---|---|
US (1) | US20050256037A1 (es) |
JP (1) | JP2008502583A (es) |
CA (1) | CA2540646A1 (es) |
UY (1) | UY28542A1 (es) |
WO (1) | WO2005033129A1 (es) |
Families Citing this family (14)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE10226921A1 (de) * | 2002-06-17 | 2003-12-24 | Bayer Ag | Antibakterielle Amid-Makrozyklen |
DE10358824A1 (de) | 2003-12-16 | 2005-07-21 | Bayer Healthcare Ag | Antibakterielle Makrozyklen mit substituiertem Biphenyl |
DE102005014240A1 (de) * | 2004-09-24 | 2006-03-30 | Bayer Healthcare Ag | Antibakterielle Amid-Makrozyklen IV |
DE102005014247A1 (de) * | 2005-03-30 | 2006-10-05 | Aicuris Gmbh & Co. Kg | Antibakterielle Amid-Makrozyklen VI |
DE102005014245A1 (de) * | 2005-03-30 | 2006-10-05 | Aicuris Gmbh & Co. Kg | Antibakterielle Amid-Makrozyklen V |
DE102005032781A1 (de) * | 2005-07-14 | 2007-01-18 | Aicuris Gmbh & Co. Kg | Antibakterielle Amid-Markozyklen VII |
WO2007089335A2 (en) * | 2005-12-29 | 2007-08-09 | Lexicon Pharmaceutical Inc. | Multicyclic amino acid derivatives and methods of their use |
CA2848238C (en) * | 2006-10-03 | 2016-07-19 | Tekmira Pharmaceuticals Corporation | Lipid containing formulations |
MX2010007823A (es) * | 2008-01-18 | 2010-08-10 | Merck Sharp & Dohme | Inhibidores de beta-lactamasa. |
PT3368544T (pt) | 2015-10-27 | 2020-08-20 | Hoffmann La Roche | Péptidos macrocíclicos contra acinetobacter baumannii |
EP3388444A1 (en) | 2017-04-10 | 2018-10-17 | F. Hoffmann-La Roche AG | Anti-bacterial peptide macrocycles and use thereof |
US11505573B2 (en) | 2018-03-28 | 2022-11-22 | Hoffmann-La Roche Inc. | Peptide macrocycles against Acinetobacter baumannii |
US11819532B2 (en) | 2018-04-23 | 2023-11-21 | Hoffmann-La Roche Inc. | Peptide macrocycles against Acinetobacter baumannii |
TWI797784B (zh) * | 2020-10-22 | 2023-04-01 | 美商恩特葛瑞斯股份有限公司 | 環戊二烯的選擇性烷基化 |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3452136A (en) * | 1968-04-17 | 1969-06-24 | American Cyanamid Co | Antibiotic af283 and production thereof |
DE10226921A1 (de) * | 2002-06-17 | 2003-12-24 | Bayer Ag | Antibakterielle Amid-Makrozyklen |
-
2004
- 2004-09-22 CA CA002540646A patent/CA2540646A1/en not_active Abandoned
- 2004-09-22 JP JP2006530002A patent/JP2008502583A/ja not_active Ceased
- 2004-09-22 WO PCT/EP2004/010605 patent/WO2005033129A1/de active Application Filing
- 2004-09-30 UY UY28542A patent/UY28542A1/es not_active Application Discontinuation
- 2004-10-01 US US10/957,489 patent/US20050256037A1/en not_active Abandoned
Also Published As
Publication number | Publication date |
---|---|
CA2540646A1 (en) | 2005-04-14 |
WO2005033129A1 (de) | 2005-04-14 |
JP2008502583A (ja) | 2008-01-31 |
US20050256037A1 (en) | 2005-11-17 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
NO20050210L (no) | Antibakterielle amid-makrocykluser | |
ECSP056138A (es) | Dihidroquinazolinas sustituidas | |
DOP2002000429A (es) | Imidazotriazinas | |
MY150958A (en) | Compounds for the treatment of multi-drug resistant bacterial infections | |
UY29170A1 (es) | Adeninas sustituidas y usos de las mismas | |
UY28313A1 (es) | Nonadepsipeptidos acilados | |
UY28542A1 (es) | Amidas macrocíclicas antibacterianas | |
UY29189A1 (es) | Nonadepsipeptidos acilados ii | |
ATE495186T1 (de) | Antibakterielle amid-makrozyklen iv | |
ATE510845T1 (de) | Antibakterielle makrozyklen mit substituiertem biphenyl | |
WO2005118613A3 (de) | Antibakterielle amid-makrozyklen | |
ATE433459T1 (de) | Desoxo-nonadepsipeptide | |
CL2004000710A1 (es) | Composicion antimicrobiana y antiparasitaria formada por un antibiotico derivado del cloranfenicol o tianfenicol, un endectocida y por lo menos un vehiculo aceptable, y su uso para tratar enfermedades respiratorias y parasitarias de los bovinos. | |
ATE455789T1 (de) | Substituierte nonadepsipeptide | |
DE502005005652D1 (de) | Heterocyclyl-substituierte nonadepsipeptide | |
ATE524488T1 (de) | Lysobactinamide | |
DOP2001000140A (es) | Aril y heteroarilsulfonatos | |
DOP2004001003A (es) | Amidas macrociclicas antibacterianas | |
WO2005121160A3 (en) | 11, 12 cyclic thiocarbamate macrolide antibacterial agents | |
GT200400196A (es) | Amidas macrociclicas antibacterianas | |
UY26945A1 (es) | Alcanosulfonatos de fenoxifenilo | |
DOP2004000891A (es) | Nonadepsipeptidos acilados | |
DOP2005000223A (es) | Nonadepsipeptidos acilados ii | |
ATE554079T1 (de) | Neue makrolidverbindungen mit antibiotischen und antineoplastischen eigenschaften | |
WO2007006548A3 (de) | Antibakterielle amid-makrozyklen vii |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
109 | Application deemed to be withdrawn |
Effective date: 20150526 |