HK1090061A1 - Novel lincomycin derivatives possessing antimicrobial activity - Google Patents
Novel lincomycin derivatives possessing antimicrobial activityInfo
- Publication number
- HK1090061A1 HK1090061A1 HK06110528.4A HK06110528A HK1090061A1 HK 1090061 A1 HK1090061 A1 HK 1090061A1 HK 06110528 A HK06110528 A HK 06110528A HK 1090061 A1 HK1090061 A1 HK 1090061A1
- Authority
- HK
- Hong Kong
- Prior art keywords
- antimicrobial activity
- derivatives possessing
- lincomycin derivatives
- possessing antimicrobial
- novel lincomycin
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/70—Carbohydrates; Sugars; Derivatives thereof
- A61K31/7042—Compounds having saccharide radicals and heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/70—Carbohydrates; Sugars; Derivatives thereof
- A61K31/7042—Compounds having saccharide radicals and heterocyclic rings
- A61K31/7052—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
- C07H15/02—Acyclic radicals, not substituted by cyclic structures
- C07H15/14—Acyclic radicals, not substituted by cyclic structures attached to a sulfur, selenium or tellurium atom of a saccharide radical
- C07H15/16—Lincomycin; Derivatives thereof
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US47950203P | 2003-06-17 | 2003-06-17 | |
| US47929603P | 2003-06-17 | 2003-06-17 | |
| US10/642,807 US7164011B2 (en) | 2002-08-15 | 2003-08-15 | Lincomycin derivatives possessing antibacterial activity |
| US10/777,455 US7199105B2 (en) | 2002-08-15 | 2004-02-11 | Lincomycin derivatives possessing antibacterial activity |
| PCT/US2004/019689 WO2005012320A2 (en) | 2003-06-17 | 2004-06-17 | Novel lincomycin derivatives possessing antimicrobial activity |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| HK1090061A1 true HK1090061A1 (en) | 2006-12-15 |
Family
ID=40203032
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| HK06110528.4A HK1090061A1 (en) | 2003-06-17 | 2006-09-21 | Novel lincomycin derivatives possessing antimicrobial activity |
Country Status (17)
| Country | Link |
|---|---|
| EP (1) | EP1644393A2 (en) |
| JP (1) | JP2007516172A (en) |
| KR (1) | KR20060091050A (en) |
| AU (1) | AU2004261550A1 (en) |
| BR (1) | BRPI0411534A (en) |
| CA (1) | CA2528592A1 (en) |
| EC (1) | ECSP056233A (en) |
| GE (1) | GEP20084437B (en) |
| HK (1) | HK1090061A1 (en) |
| IL (1) | IL172183A0 (en) |
| IS (1) | IS8147A (en) |
| MA (1) | MA27860A1 (en) |
| MX (1) | MXPA05013915A (en) |
| NO (1) | NO20055893L (en) |
| OA (1) | OA13179A (en) |
| RS (1) | RS20050931A (en) |
| WO (1) | WO2005012320A2 (en) |
Families Citing this family (18)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ZA200501012B (en) | 2002-08-15 | 2006-10-25 | Vicuron Pharm Inc | Lincomycin derivatives possessing antibacterial activity |
| US7199105B2 (en) | 2002-08-15 | 2007-04-03 | Vicuron Pharmaceuticals, Inc. | Lincomycin derivatives possessing antibacterial activity |
| US7256177B2 (en) | 2003-06-17 | 2007-08-14 | Vicuron Pharmaceuticals, Inc. | Lincomycin derivatives possessing antibacterial activity |
| EP1654268A2 (en) * | 2003-06-17 | 2006-05-10 | Vicuron Pharmaceuticals, Inc. | Lincomycin derivatives possessing antibacterial activity |
| US7199106B2 (en) | 2003-06-17 | 2007-04-03 | Vicuron Pharmaceuticals, Inc. | Lincomycin derivatives possessing antimicrobial activity |
| US7361743B2 (en) * | 2004-02-11 | 2008-04-22 | Pfizer Inc | Lincomycin derivatives possessing antibacterial activity |
| BRPI0615300A2 (en) * | 2005-08-31 | 2009-07-14 | Wyeth Corp | compound; pharmaceutical composition; method for the preparation, treatment or control of bacterial infections in warm-blooded animals; use of a compound; and method for preparing compounds represented by formula (i) |
| US7871982B2 (en) | 2005-12-09 | 2011-01-18 | Meiji Seika Kaisha, Ltd. | Lincomycin derivatives and antimicrobial agents comprising the same as active ingredient |
| WO2008146917A1 (en) * | 2007-05-31 | 2008-12-04 | Meiji Seika Kaisha, Ltd. | Lincomycin derivatives and antibacterial agents containing the same as the active ingredient |
| WO2008146919A1 (en) | 2007-05-31 | 2008-12-04 | Meiji Seika Kaisha, Ltd. | Lincosamide derivative, and antibacterial agent comprising the same as active ingredient |
| US20130267699A1 (en) | 2011-06-24 | 2013-10-10 | California Institute Of Technology | Quaternary heteroatom containing compounds |
| US8822679B2 (en) * | 2011-06-24 | 2014-09-02 | California Institute Of Technology | Quaternary heteroatom containing compounds |
| US10421696B2 (en) | 2014-12-18 | 2019-09-24 | California Institute Of Technology | Enantioselective synthesis of α-quaternary mannich adducts by palladium-catalyzed allylic alkylation |
| CN107922373A (en) | 2015-03-27 | 2018-04-17 | 加利福尼亚技术学院 | Use low catalyst concentration and the asymmetry catalysis decarboxylation alkyl-alkyl for the pre-catalyst stablized |
| WO2017156239A1 (en) | 2016-03-11 | 2017-09-14 | California Institute Of Technology | Compositions and methods for acylating lactams |
| US10358422B2 (en) | 2017-11-01 | 2019-07-23 | California Institute Of Technology | Methods for enantioselective allylic alkylation of esters, lactones, and lactams with unactivated allylic alcohols |
| EP3699173A1 (en) | 2018-10-18 | 2020-08-26 | California Institute of Technology | Gem-disubstituted pyrrolidines, piperazines, and diazepanes, and compositions and methods of making the same |
| CN110357839A (en) * | 2019-08-29 | 2019-10-22 | 重庆经致制药技术开发有限公司 | The preparation method of Bu Waxitan chiral intermediate |
Family Cites Families (16)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3268556A (en) * | 1964-04-13 | 1966-08-23 | Upjohn Co | Novel lincomycin derivatives |
| NL128232C (en) * | 1964-04-13 | |||
| NL146501C (en) * | 1964-07-01 | |||
| US3282917A (en) * | 1964-08-17 | 1966-11-01 | Upjohn Co | Methyl n-(1-alkyl-4-alkoxy-prolyl)-alpha-thiolincosaminide compounds and process therefor |
| NL140527B (en) * | 1965-02-08 | 1973-12-17 | Upjohn Co | PROCESS FOR PREPARING LINCOMYCIN RELATED COMPOUNDS. |
| US3496163A (en) * | 1965-02-08 | 1970-02-17 | Upjohn Co | 7-halo-7-deoxylincomycins and process for preparing the same |
| US3555007A (en) * | 1968-07-22 | 1971-01-12 | Upjohn Co | 7-deoxy-7-halo lincomycin d derivatives |
| US3549615A (en) * | 1968-10-17 | 1970-12-22 | Upjohn Co | Lincomycin derivatives and process for producing the same |
| DE2118636A1 (en) * | 1970-04-20 | 1971-11-04 | The Upjohn Co., Kalamazoo, Mich. (V.StA.) | 3-nucleotides of lincomycin and their analogues, processes for their preparation and their use in therapeutic preparations |
| US3787390A (en) * | 1971-06-23 | 1974-01-22 | Upjohn Co | Analogs of lincomycin and process |
| US3849396A (en) * | 1973-01-08 | 1974-11-19 | Upjohn Co | Lincomycin and clindamycin 1-o-ethers |
| US3923602A (en) * | 1973-10-25 | 1975-12-02 | Upjohn Co | Composition of matter and process |
| JPS5641239A (en) * | 1979-09-13 | 1981-04-17 | Hitachi Cable Ltd | Flame-retardant composition |
| US4278789A (en) * | 1979-11-23 | 1981-07-14 | The Upjohn Company | Lincomycin compounds |
| ZA200501012B (en) * | 2002-08-15 | 2006-10-25 | Vicuron Pharm Inc | Lincomycin derivatives possessing antibacterial activity |
| JP2007528360A (en) * | 2003-06-17 | 2007-10-11 | ビキュロン・ファーマシューティカルズ・インコーポレイテッド | Lincomycin derivatives with antibacterial activity |
-
2004
- 2004-06-17 KR KR1020057024291A patent/KR20060091050A/en active Search and Examination
- 2004-06-17 EP EP04776816A patent/EP1644393A2/en not_active Withdrawn
- 2004-06-17 WO PCT/US2004/019689 patent/WO2005012320A2/en active Application Filing
- 2004-06-17 GE GEAP20049117A patent/GEP20084437B/en unknown
- 2004-06-17 JP JP2006517464A patent/JP2007516172A/en active Pending
- 2004-06-17 AU AU2004261550A patent/AU2004261550A1/en not_active Abandoned
- 2004-06-17 OA OA1200500364A patent/OA13179A/en unknown
- 2004-06-17 BR BRPI0411534-1A patent/BRPI0411534A/en not_active IP Right Cessation
- 2004-06-17 RS YUP-2005/0931A patent/RS20050931A/en unknown
- 2004-06-17 MX MXPA05013915A patent/MXPA05013915A/en unknown
- 2004-06-17 CA CA002528592A patent/CA2528592A1/en not_active Abandoned
-
2005
- 2005-11-24 IS IS8147A patent/IS8147A/en unknown
- 2005-11-24 IL IL172183A patent/IL172183A0/en unknown
- 2005-12-12 NO NO20055893A patent/NO20055893L/en not_active Application Discontinuation
- 2005-12-16 MA MA28672A patent/MA27860A1/en unknown
- 2005-12-16 EC EC2005006233A patent/ECSP056233A/en unknown
-
2006
- 2006-09-21 HK HK06110528.4A patent/HK1090061A1/en not_active IP Right Cessation
Also Published As
| Publication number | Publication date |
|---|---|
| OA13179A (en) | 2006-12-13 |
| NO20055893L (en) | 2006-03-14 |
| AU2004261550A1 (en) | 2005-02-10 |
| KR20060091050A (en) | 2006-08-17 |
| IS8147A (en) | 2005-11-24 |
| EP1644393A2 (en) | 2006-04-12 |
| WO2005012320A2 (en) | 2005-02-10 |
| MXPA05013915A (en) | 2006-07-03 |
| BRPI0411534A (en) | 2006-08-22 |
| MA27860A1 (en) | 2006-04-03 |
| WO2005012320A3 (en) | 2005-10-20 |
| JP2007516172A (en) | 2007-06-21 |
| ECSP056233A (en) | 2006-04-19 |
| IL172183A0 (en) | 2011-08-01 |
| CA2528592A1 (en) | 2005-02-10 |
| RS20050931A (en) | 2008-04-04 |
| GEP20084437B (en) | 2008-07-25 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| PC | Patent ceased (i.e. patent has lapsed due to the failure to pay the renewal fee) |
Effective date: 20140617 |