PT94645A - Processo para a preparacao de derivados de aminopirimidina com actividade fungicida e de composicoes fungicidas que os contem - Google Patents
Processo para a preparacao de derivados de aminopirimidina com actividade fungicida e de composicoes fungicidas que os contemInfo
- Publication number
- PT94645A PT94645A PT94645A PT9464590A PT94645A PT 94645 A PT94645 A PT 94645A PT 94645 A PT94645 A PT 94645A PT 9464590 A PT9464590 A PT 9464590A PT 94645 A PT94645 A PT 94645A
- Authority
- PT
- Portugal
- Prior art keywords
- fungicid
- activity
- preparation
- compositions containing
- aminopyrimidine derivatives
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
- A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Agronomy & Crop Science (AREA)
- Pest Control & Pesticides (AREA)
- Plant Pathology (AREA)
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Dentistry (AREA)
- General Health & Medical Sciences (AREA)
- Wood Science & Technology (AREA)
- Zoology (AREA)
- Environmental Sciences (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE3922735A DE3922735A1 (de) | 1989-07-11 | 1989-07-11 | Aminopyrimidin-derivate, verfahren zu ihrer herstellung, sie enthaltende mittel und ihre verwendung als fungizide |
Publications (2)
Publication Number | Publication Date |
---|---|
PT94645A true PT94645A (pt) | 1991-03-20 |
PT94645B PT94645B (pt) | 1997-02-28 |
Family
ID=6384711
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
PT94645A PT94645B (pt) | 1989-07-11 | 1990-07-10 | Processo para a preparacao de derivados de aminopirimidina com actividade fungicida e de composicoes fungicidas que os contem |
Country Status (5)
Country | Link |
---|---|
US (1) | US5250530A (pt) |
EP (1) | EP0407899B1 (pt) |
DE (2) | DE3922735A1 (pt) |
HU (1) | HUT54280A (pt) |
PT (1) | PT94645B (pt) |
Families Citing this family (71)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CA2091986C (en) * | 1990-10-09 | 1995-11-28 | Andrew Thurkauf | Certain cycloalkyl and azacycloalkyl pyrrolopyrimidines; a new class of gaba brain receptor ligands |
GB9024873D0 (en) * | 1990-11-15 | 1991-01-02 | Ici Plc | Fungicidal compounds |
WO1992010490A1 (de) * | 1990-12-05 | 1992-06-25 | Hoechst Aktiengesellschaft | Pyridyl-pyrimidin-derivate, verfahren zu ihrer herstellung, sie enthaltende mittel und ihre verwendung als fungizide |
DE4117560A1 (de) * | 1991-05-29 | 1992-12-03 | Bayer Ag | Verwendung von pyridinylpyrimidin-derivaten zum schutz technischer materialien |
US5593996A (en) * | 1991-12-30 | 1997-01-14 | American Cyanamid Company | Triazolopyrimidine derivatives |
DE4206148A1 (de) * | 1992-02-28 | 1993-09-02 | Bayer Ag | Substituierte pyridylpyrimidine |
JP2657760B2 (ja) * | 1992-07-15 | 1997-09-24 | 小野薬品工業株式会社 | 4−アミノキナゾリン誘導体およびそれを含有する医薬品 |
ATE163647T1 (de) * | 1993-08-26 | 1998-03-15 | Ono Pharmaceutical Co | 4-aminopyrimidin derivate |
US6410729B1 (en) | 1996-12-05 | 2002-06-25 | Amgen Inc. | Substituted pyrimidine compounds and methods of use |
JPH11199564A (ja) * | 1997-09-12 | 1999-07-27 | American Cyanamid Co | 除草性2−アジニル−6−アリールオキシピリ(ミ)ジン |
US6174901B1 (en) | 1998-12-18 | 2001-01-16 | Amgen Inc. | Substituted pyridine and pyridazine compounds and methods of use |
DE19904710A1 (de) * | 1999-02-05 | 2000-08-10 | Aventis Pharma Gmbh | Substituierte 4-Amino-2-aryl-tetrahydrochinazoline, ihre Herstellung, ihre Verwendung und sie enthaltende pharmazeutische Präparate |
US6906067B2 (en) * | 1999-12-28 | 2005-06-14 | Bristol-Myers Squibb Company | N-heterocyclic inhibitors of TNF-α expression |
FR2803592A1 (fr) * | 2000-01-06 | 2001-07-13 | Aventis Cropscience Sa | Nouveaux derives de l'acide 3-hydroxypicolinique, leur procede de preparation et compositions fongicides les contenant. |
US6716851B2 (en) | 2000-12-12 | 2004-04-06 | Cytovia, Inc. | Substituted 2-aryl-4-arylaminopyrimidines and analogs as activators or caspases and inducers of apoptosis and the use thereof |
EP1373222A2 (de) | 2001-03-15 | 2004-01-02 | Basf Aktiengesellschaft | 5-phenylpyrimidine, verfahren und zwischenprodukte zu ihrer herstellung und ihre verwendung zur bekaempfung von schadpilzen |
ES2242839T3 (es) * | 2001-04-20 | 2005-11-16 | Ciba Specialty Chemicals Holding Inc. | 4-amino-2- (piridin-2-il)pirimidina como sustancias activas microbicidas. |
EP1254903B1 (en) * | 2001-04-20 | 2005-06-08 | Ciba SC Holding AG | 4-Amino-2-(pyridin-2-yl)pyrimidine as microbicidal active substances |
CA2345853A1 (en) | 2001-04-30 | 2002-10-30 | Minoru Katayama | Skiing facilities capable of changing shape of surface of ski slope and method for changing shape of surface of ski slope of skiing facilities |
CA2467683C (en) | 2001-11-19 | 2011-09-27 | Basf Aktiengesellschaft | 5-phenylpyrimidines, agents comprising the same, method for production and use thereof |
ATE428705T1 (de) * | 2002-02-21 | 2009-05-15 | Basf Se | 2-(2-pyridyl)-5-phenyl-6-aminopyrimidine, verfahren und zwischenprodukte zu ihrer herstellung und ihre verwendung zur bekämpfung von schadpilzen |
CN1642422A (zh) * | 2002-03-15 | 2005-07-20 | 西巴特殊化学品控股有限公司 | 4-氨基嘧啶及其在表面抗菌处理中的应用 |
WO2004013124A1 (en) * | 2002-07-31 | 2004-02-12 | Ciba Specialty Chemicals Holding Inc. | Pyridyl-triazine derivatives as microbicidal active substances |
US7759336B2 (en) * | 2002-12-10 | 2010-07-20 | Ono Pharmaceutical Co., Ltd. | Nitrogen-containing heterocyclic compounds and medicinal use thereof |
CN100357297C (zh) * | 2003-02-06 | 2007-12-26 | 巴斯福股份公司 | 嘧啶、其生产方法及其用途 |
US20040254178A1 (en) * | 2003-04-16 | 2004-12-16 | Amgen Inc. | Substituted heterocyclic compounds and methods of use |
TWI312272B (en) * | 2003-05-12 | 2009-07-21 | Sumitomo Chemical Co | Pyrimidine compound and pests controlling composition containing the same |
JP4595381B2 (ja) * | 2003-05-12 | 2010-12-08 | 住友化学株式会社 | ピリミジン化合物及びその有害生物防除用途 |
MXPA06001494A (es) * | 2003-08-05 | 2007-05-11 | Vertex Pharma | Compuestos de piramidina condensados como inhibidores de canales ionicos gatillados por tension. |
US6818631B1 (en) * | 2003-08-15 | 2004-11-16 | Nippon Soda Co. Ltd. | Fungicidal pyrimidine derivatives |
US20050038041A1 (en) * | 2003-08-15 | 2005-02-17 | Yuki Nakagawa | Fungicidal pyrimidine derivatives |
ES2234433B1 (es) * | 2003-12-15 | 2006-11-01 | Almirall Prodesfarma, S.A. | 4-aminopirimidinas como antagonistas de receptores de adenosina. |
DE102004003428A1 (de) * | 2004-01-23 | 2005-08-11 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | Neue langwirksame Beta-2-Agonisten, und deren Verwendung als Arzneimittel |
JP2005232081A (ja) * | 2004-02-19 | 2005-09-02 | Bayer Cropscience Ag | ベンジルピリミジン誘導体の農園芸用殺菌剤としての利用 |
TW200538180A (en) * | 2004-02-20 | 2005-12-01 | Astrazeneca Ab | New compounds |
WO2006000358A1 (de) * | 2004-06-25 | 2006-01-05 | Basf Aktiengesellschaft | 2, 4, 5, 6-substituierte pyridine, verfahren zu ihrer herstellung und ihre verwendung zur bekämpfung von schadpilzen |
EP1768972A1 (de) * | 2004-07-14 | 2007-04-04 | Basf Aktiengesellschaft | 2-substituierte pyrimidine, verfahren zu ihrer herstellung und ihre verwendung zur bekämpfung von schadpilzen |
JP2008513401A (ja) * | 2004-09-17 | 2008-05-01 | ビーエーエスエフ ソシエタス・ヨーロピア | 植物の線虫病に対処するための2−置換ピリミジンの使用 |
EP1793676A1 (en) * | 2004-09-23 | 2007-06-13 | Basf Aktiengesellschaft | Use of 2-substituted pyrimidines for combating nematode of plants |
JP2006188462A (ja) * | 2005-01-07 | 2006-07-20 | Ube Ind Ltd | 4−(ホモ)ピペラジニルピリミジン誘導体及び抗菌剤 |
US20060178388A1 (en) * | 2005-02-04 | 2006-08-10 | Wrobleski Stephen T | Phenyl-substituted pyrimidine compounds useful as kinase inhibitors |
US20080176744A1 (en) * | 2005-03-10 | 2008-07-24 | Basf Aktiengesellschaft | Use of 4-Aminopyrimidines for Controlling Harmful Fungi, Novel 4-Aminopyrimidines, Processes for Their Preparation and Compositions Comprising Them |
EP1956009A1 (en) * | 2005-12-02 | 2008-08-13 | Mitsubishi Tanabe Pharma Corporation | Aromatic compound |
KR20080083188A (ko) * | 2006-01-11 | 2008-09-16 | 아스트라제네카 아베 | 모르폴리노 피리미딘 유도체 및 요법에서의 그 유도체의용도 |
WO2008023180A1 (en) * | 2006-08-24 | 2008-02-28 | Astrazeneca Ab | Morpholino pyrimidine derivatives useful in the treatment of proliferative disorders |
MX2009002046A (es) | 2006-08-24 | 2009-03-06 | Astrazeneca Ab | Derivados de morfolino pirimidina utiles en el tratamiento de trastornos proliferativos. |
WO2008028935A2 (en) * | 2006-09-07 | 2008-03-13 | Neurosearch A/S | Pyridinyl-pyrimidine derivatives useful as potassium channel modulating agents |
JP2010511727A (ja) * | 2006-12-04 | 2010-04-15 | ニューロクライン バイオサイエンシーズ,インコーポレイテッド | アデノシン受容体アンタゴニストとしての置換ピリミジン |
US20100249084A1 (en) * | 2007-03-21 | 2010-09-30 | Youngsheng Chen | Substituted pyrimidines as adenosine receptor antagonists |
US20100227858A1 (en) * | 2007-07-09 | 2010-09-09 | Astrazeneca Ab | Trisubstituted pyrimidine derivatives for the treatment of proliferative diseases |
AU2008273891B2 (en) | 2007-07-09 | 2012-01-12 | Astrazeneca Ab | Morpholino pyrimidine derivatives used in diseases linked to mTOR kinase and/or PI3K |
US20100261723A1 (en) * | 2007-07-09 | 2010-10-14 | Astrazeneca Ab | Trisubstituted pyrimidine derivatives for the treatment of proliferative diseases |
AU2008273889B2 (en) * | 2007-07-09 | 2012-03-08 | Astrazeneca Ab | Trisubstituted pyrimidine derivatives for the treatment of proliferative diseases |
WO2009019099A1 (en) * | 2007-08-09 | 2009-02-12 | Basf Se | Tetrasubstituted pyrimidine derivatives for controlling phytopathogenic fungi |
PL2432767T3 (pl) * | 2009-05-19 | 2013-11-29 | Dow Agrosciences Llc | Związki i sposoby zwalczania grzybów |
DE102010002558A1 (de) | 2009-11-20 | 2011-06-01 | Symrise Ag | Verwendung physiologischer Kühlwirkstoffe und Mittel enthaltend solche Wirkstoffe |
KR101467858B1 (ko) * | 2009-12-28 | 2014-12-02 | 재단법인 생물기술개발중심 | mTOR 및 PI3K 억제제로서의 신규 피리미딘 화합물 |
US9315491B2 (en) | 2009-12-28 | 2016-04-19 | Development Center For Biotechnology | Pyrimidine compounds as mTOR and PI3K inhibitors |
SA111320519B1 (ar) | 2010-06-11 | 2014-07-02 | Astrazeneca Ab | مركبات بيريميدينيل للاستخدام كمثبطات atr |
WO2012035421A2 (en) | 2010-09-17 | 2012-03-22 | Purdue Pharma L.P. | Pyridine compounds and the uses thereof |
WO2015003360A2 (en) * | 2013-07-11 | 2015-01-15 | Agios Pharmaceuticals, Inc. | Therapeutically active compounds and their methods of use |
EP3278873B1 (en) * | 2015-03-30 | 2020-02-05 | Nippon Shokubai Co., Ltd. | Particulate water-absorbing agent |
BR112018012914B1 (pt) | 2015-12-22 | 2023-04-18 | SHY Therapeutics LLC | Composto, uso de um composto e composição farmacêutica |
US10774064B2 (en) | 2016-06-02 | 2020-09-15 | Cadent Therapeutics, Inc. | Potassium channel modulators |
SI3571193T1 (sl) | 2017-01-23 | 2022-04-29 | Cadent Therapeutics, Inc. | Modulatorji kalijevega kanalčka |
KR20200041294A (ko) | 2017-06-21 | 2020-04-21 | 샤이 테라퓨틱스 엘엘씨 | 암, 염증성 질환, 신경발달질환 및 섬유증 질환의 치료를 위하여 Ras 수퍼패밀리와 상호작용하는 화합물 |
JP2022508945A (ja) | 2018-10-22 | 2022-01-19 | カデント セラピューティクス,インコーポレーテッド | カリウムチャネルモジュレーターの結晶形態 |
US11746100B2 (en) | 2020-04-28 | 2023-09-05 | Global Blood Therapeutics, Inc. | Cycloalkyl pyrimidines as ferroportin inhibitors |
JP7471407B2 (ja) * | 2020-05-19 | 2024-04-19 | ユニマテック株式会社 | 含フッ素ピリミジン化合物および含フッ素ピリミジノン化合物 |
WO2022239808A1 (ja) * | 2021-05-11 | 2022-11-17 | 国立研究開発法人理化学研究所 | 抗寄生虫活性を有する化合物 |
WO2023085142A1 (ja) * | 2021-11-12 | 2023-05-19 | ユニマテック株式会社 | 含フッ素ピリミジン化合物、有害菌類防除剤および含フッ素ピリミジン化合物の製造方法 |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4109092A (en) * | 1976-10-07 | 1978-08-22 | Sterling Drug Inc. | Preparation of 2-(pyridinyl)-4-pyrimidinamines |
DE3675197D1 (de) * | 1985-12-03 | 1990-11-29 | Sumitomo Chemical Co | Pyridinylpyrimidin-derivate, verfahren zu deren herstellung und diese als wirksamen stoff enthaltende pflanzenkrankheiten-schutzmittel. |
PH23565A (en) * | 1986-09-05 | 1989-08-25 | Sumitomo Chemical Co | Novel pyrimidinylpyrimidine derivatives and a plant disease protectant containing them as the active ingredient |
CA1288433C (en) * | 1986-12-03 | 1991-09-03 | Tsuguhiro Katoh | Pyridinylpyrimidine derivatives, method for production thereof and a fungicide containing them as the active ingredient |
-
1989
- 1989-07-11 DE DE3922735A patent/DE3922735A1/de not_active Withdrawn
-
1990
- 1990-07-06 EP EP90112903A patent/EP0407899B1/de not_active Expired - Lifetime
- 1990-07-06 DE DE59008571T patent/DE59008571D1/de not_active Expired - Fee Related
- 1990-07-09 US US07/549,764 patent/US5250530A/en not_active Expired - Fee Related
- 1990-07-10 HU HU904151A patent/HUT54280A/hu unknown
- 1990-07-10 PT PT94645A patent/PT94645B/pt not_active IP Right Cessation
Also Published As
Publication number | Publication date |
---|---|
EP0407899A3 (en) | 1991-07-24 |
DE59008571D1 (de) | 1995-04-06 |
EP0407899A2 (de) | 1991-01-16 |
HU904151D0 (pt) | 1990-12-28 |
PT94645B (pt) | 1997-02-28 |
US5250530A (en) | 1993-10-05 |
HUT54280A (en) | 1991-02-28 |
EP0407899B1 (de) | 1995-03-01 |
DE3922735A1 (de) | 1991-01-24 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
BB1A | Laying open of patent application |
Effective date: 19901011 |
|
FG3A | Patent granted, date of granting |
Effective date: 19961129 |
|
MM3A | Annulment or lapse |
Free format text: LAPSE DUE TO NON-PAYMENT OF FEES Effective date: 19980531 |