PT89353A - Processo para a preparacao de derivados de cefalosporina com actividade antimicrobiana e de composicoes farmaceuticas que os contem - Google Patents

Processo para a preparacao de derivados de cefalosporina com actividade antimicrobiana e de composicoes farmaceuticas que os contem

Info

Publication number
PT89353A
PT89353A PT89353A PT8935388A PT89353A PT 89353 A PT89353 A PT 89353A PT 89353 A PT89353 A PT 89353A PT 8935388 A PT8935388 A PT 8935388A PT 89353 A PT89353 A PT 89353A
Authority
PT
Portugal
Prior art keywords
cefalosporine
derivatives
preparation
pharmaceutical compositions
compositions containing
Prior art date
Application number
PT89353A
Other languages
English (en)
Inventor
Dennis Dalton Keith
Ka-Kong Chan
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of PT89353A publication Critical patent/PT89353A/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D501/00Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/14Compounds having a nitrogen atom directly attached in position 7
    • C07D501/16Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
    • C07D501/207-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids
    • C07D501/247-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids with hydrocarbon radicals, substituted by hetero atoms or hetero rings, attached in position 3
    • C07D501/36Methylene radicals, substituted by sulfur atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D519/00Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Cephalosporin Compounds (AREA)
PT89353A 1987-12-28 1988-12-28 Processo para a preparacao de derivados de cefalosporina com actividade antimicrobiana e de composicoes farmaceuticas que os contem PT89353A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US13841087A 1987-12-28 1987-12-28
US25500488A 1988-10-07 1988-10-07

Publications (1)

Publication Number Publication Date
PT89353A true PT89353A (pt) 1989-12-29

Family

ID=26836174

Family Applications (1)

Application Number Title Priority Date Filing Date
PT89353A PT89353A (pt) 1987-12-28 1988-12-28 Processo para a preparacao de derivados de cefalosporina com actividade antimicrobiana e de composicoes farmaceuticas que os contem

Country Status (13)

Country Link
EP (1) EP0322810A3 (pt)
JP (1) JPH01203395A (pt)
KR (1) KR890009942A (pt)
AU (1) AU621328B2 (pt)
DK (1) DK722988A (pt)
FI (1) FI885988A (pt)
HU (1) HU205361B (pt)
IL (1) IL88775A0 (pt)
MC (1) MC2000A1 (pt)
NO (1) NO885780L (pt)
NZ (1) NZ227470A (pt)
PT (1) PT89353A (pt)
YU (2) YU234688A (pt)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ZA874696B (en) * 1986-07-03 1988-01-04 F. Hoffmann-La Roche & Co. Aktiengesellschaft Acyl derivatives
EP0366193A3 (en) * 1988-10-24 1992-01-08 Norwich Eaton Pharmaceuticals, Inc. Novel antimicrobial quinolonyl lactams
CA2001203C (en) * 1988-10-24 2001-02-13 Thomas P. Demuth, Jr. Novel antimicrobial dithiocarbamoyl quinolones
EP0997466A1 (en) * 1988-10-24 2000-05-03 PROCTER & GAMBLE PHARMACEUTICALS, INC. Novel antimicrobial lactam-quinolones
US5328908A (en) * 1988-10-24 1994-07-12 Procter & Gamble Pharmaceuticals, Inc. Antimicrobial quinolone thioureas
SG54293A1 (en) * 1988-10-24 1998-11-16 Procter & Gamble Pharma Novel antimicrobial fluoroquinolonyl cephems
EP0525057B1 (en) * 1990-04-18 2000-06-14 Procter & Gamble Pharmaceuticals, Inc. Antimicrobial quinolonyl lactams
US5066800A (en) * 1990-04-27 1991-11-19 Hoffmann-La Roche Inc. Qunoline intermediates useful therein for synthesizing antibacterial compounds
DE4234330A1 (de) * 1992-10-12 1994-04-14 Bayer Ag Chinoloncarbonsäuren

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2479229B1 (fr) * 1980-03-26 1986-01-17 Clin Midy Nouveaux derives des cephalosporines, leur procede de preparation et les medicaments utilisables comme antibiotiques qui contiennent lesdits derives
US4396620A (en) * 1981-09-08 1983-08-02 Eli Lilly And Company Cephalosporin quinolinium betaines
KR920004820B1 (ko) * 1984-02-23 1992-06-18 메이지제과 주식회사 새로운 세팔로스포린 유도체의 제조방법
FR2570702B1 (fr) * 1984-09-27 1987-01-09 Sanofi Sa Derives des cephalosporines, procedes d'obtention et leur application a titre d'antibiotiques
ZA874696B (en) * 1986-07-03 1988-01-04 F. Hoffmann-La Roche & Co. Aktiengesellschaft Acyl derivatives
CA2005787A1 (en) * 1988-12-29 1990-06-29 Masao Wada Cephalosporin compounds

Also Published As

Publication number Publication date
NO885780L (no) 1989-06-29
HUT48896A (en) 1989-07-28
YU219789A (en) 1991-06-30
MC2000A1 (fr) 1990-01-26
EP0322810A3 (de) 1989-12-13
EP0322810A2 (de) 1989-07-05
JPH01203395A (ja) 1989-08-16
KR890009942A (ko) 1989-08-05
YU234688A (en) 1990-04-30
DK722988D0 (da) 1988-12-23
DK722988A (da) 1989-06-29
NZ227470A (en) 1991-06-25
HU205361B (en) 1992-04-28
AU621328B2 (en) 1992-03-12
AU2755488A (en) 1989-06-29
FI885988A (fi) 1989-06-29
NO885780D0 (no) 1988-12-27
IL88775A0 (en) 1989-07-31

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Legal Events

Date Code Title Description
FC3A Refusal

Effective date: 19940217