PT94042A - Processo para a preparacao de compostos antagonistas de aminoacidos estimulantes do complexo de receptores do acido n-metil-d-aspartico (nmda) e de composicoes farmaceuticas que os contem - Google Patents
Processo para a preparacao de compostos antagonistas de aminoacidos estimulantes do complexo de receptores do acido n-metil-d-aspartico (nmda) e de composicoes farmaceuticas que os contemInfo
- Publication number
- PT94042A PT94042A PT94042A PT9404290A PT94042A PT 94042 A PT94042 A PT 94042A PT 94042 A PT94042 A PT 94042A PT 9404290 A PT9404290 A PT 9404290A PT 94042 A PT94042 A PT 94042A
- Authority
- PT
- Portugal
- Prior art keywords
- aminoacides
- nmda
- receptors
- methyl
- contain
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D495/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
- C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
- C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D215/48—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Pain & Pain Management (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Vascular Medicine (AREA)
- Anesthesiology (AREA)
- Urology & Nephrology (AREA)
- Psychiatry (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pyridine Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Quinoline Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Plural Heterocyclic Compounds (AREA)
- Peptides Or Proteins (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US35242389A | 1989-05-16 | 1989-05-16 |
Publications (2)
Publication Number | Publication Date |
---|---|
PT94042A true PT94042A (pt) | 1991-01-08 |
PT94042B PT94042B (pt) | 1997-05-28 |
Family
ID=23385074
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
PT94042A PT94042B (pt) | 1989-05-16 | 1990-05-15 | Processo para a preparacao de compostos antagonistas de aminoacidos estimulantes do complexo de receptores do acido n-metil-d-aspartico (nmda) e de composicoes farmaceuticas que os contem |
Country Status (19)
Country | Link |
---|---|
EP (1) | EP0398283B1 (pt) |
JP (1) | JP3014001B2 (pt) |
KR (1) | KR0169107B1 (pt) |
CN (1) | CN1027369C (pt) |
AT (1) | ATE113597T1 (pt) |
AU (1) | AU626418B2 (pt) |
DE (1) | DE69013750T2 (pt) |
DK (1) | DK0398283T3 (pt) |
ES (1) | ES2066035T3 (pt) |
FI (1) | FI95795C (pt) |
GR (1) | GR3014893T3 (pt) |
HU (1) | HU214322B (pt) |
IE (1) | IE64671B1 (pt) |
IL (1) | IL94377A (pt) |
NO (1) | NO177141C (pt) |
NZ (1) | NZ233641A (pt) |
PT (1) | PT94042B (pt) |
TW (1) | TW207950B (pt) |
ZA (1) | ZA903588B (pt) |
Families Citing this family (17)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5028707A (en) * | 1989-11-20 | 1991-07-02 | Board Of Regents, University Of Texas | 4-hydroxyquinaldic acid derivatives |
DK101290D0 (da) * | 1990-04-24 | 1990-04-24 | Novo Nordisk As | Heterocykliske forbindelser, deres fremstilling og anvendelse |
US5606063A (en) * | 1991-02-27 | 1997-02-25 | Merrell Pharmaceuticals Inc. | NMDA antagonists |
AU660969B2 (en) * | 1991-02-27 | 1995-07-13 | Merrell Pharmaceuticals Inc. | NMDA antagonists |
GB9200781D0 (en) * | 1992-01-15 | 1992-03-11 | Merck Sharp & Dohme | Therapeutic agents |
US5464843A (en) * | 1992-06-23 | 1995-11-07 | G.D. Searle & Co. | Imidazo[1,2-a]pyridinyldiacid compounds for cognitive enhancement and for treatment of cognitive disorders and neutrotoxic injury |
FR2722786B1 (fr) * | 1994-07-20 | 1996-08-23 | Rhone Poulenc Rorer Sa | Derives de 4-hydroxy-3-phenyl-indeno(1,2-b)pyridine-2(1h)- one, leur preparation et les medicaments les contenant |
DE4444815A1 (de) * | 1994-12-15 | 1996-06-20 | Merck Patent Gmbh | Thienopyridone |
WO1997037999A1 (en) * | 1996-04-04 | 1997-10-16 | University Of Nebraska Board Of Regents | Synthetic triple helix-forming compounds |
DE60022906T2 (de) | 1999-12-28 | 2006-07-06 | Eisai Co., Ltd. | Heterozyklische verbindungen mit sulfonamid-gruppen |
DE50207103D1 (en) * | 2001-03-14 | 2006-07-20 | Gruenenthal Gmbh | Substituierte pyrazolo- und thiazolopyrimidine als analgetika |
FR2864535B1 (fr) * | 2003-12-24 | 2006-12-22 | Merck Sante Sas | Derives acides de quinoline et leurs applications en therapeutique |
GB0420719D0 (en) * | 2004-09-17 | 2004-10-20 | Addex Pharmaceuticals Sa | Novel allosteric modulators |
NZ589136A (en) | 2008-04-11 | 2012-06-29 | Merck Patent Gmbh | Thienopyridone derivatives as amp-activated protein kinase (ampk) activators |
DE102008019838A1 (de) * | 2008-04-19 | 2009-12-10 | Boehringer Ingelheim International Gmbh | Neue Arylsulfonylglycin-Derivate, deren Herstellung und deren Verwendung als Arzneimittel |
WO2017121308A1 (en) * | 2016-01-11 | 2017-07-20 | Chongqing Fochon Pharmaceutical Co., Ltd. | Fused pyridine compounds, compositions and methods of use |
WO2018202039A1 (zh) * | 2017-05-03 | 2018-11-08 | 成都海创药业有限公司 | 杂环化合物及其制备方法 |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2563831B1 (fr) * | 1984-05-04 | 1986-11-21 | Sanofi Sa | Nouveaux derives de thienopyridinone, leur procede de preparation et compositions pharmaceutiques les contenant |
GB8627698D0 (en) * | 1986-11-20 | 1986-12-17 | Boots Co Plc | Therapeutic agents |
GB8804448D0 (en) * | 1988-02-25 | 1988-03-23 | Smithkline Beckman Intercredit | Compounds |
EP0403885A1 (de) * | 1989-06-20 | 1990-12-27 | Bayer Ag | Verwendung von 3-Hydroxybenzothiophenen zur Bekämpfung von Endoparasiten, neue 3-Hydroxybenzothiophene und Verfahren zu ihrer Herstellung |
EP0446604A3 (en) * | 1990-03-16 | 1992-02-19 | American Cyanamid Company | Pyridine and related aza heterocycle derivatives as cardiovascular agents |
-
1990
- 1990-05-10 AU AU54914/90A patent/AU626418B2/en not_active Ceased
- 1990-05-10 NZ NZ233641A patent/NZ233641A/en unknown
- 1990-05-10 ZA ZA903588A patent/ZA903588B/xx unknown
- 1990-05-11 TW TW079103840A patent/TW207950B/zh active
- 1990-05-14 HU HU903031A patent/HU214322B/hu not_active IP Right Cessation
- 1990-05-14 IL IL9437790A patent/IL94377A/xx not_active IP Right Cessation
- 1990-05-15 JP JP2123258A patent/JP3014001B2/ja not_active Expired - Fee Related
- 1990-05-15 PT PT94042A patent/PT94042B/pt not_active IP Right Cessation
- 1990-05-15 CN CN90103522A patent/CN1027369C/zh not_active Expired - Fee Related
- 1990-05-15 FI FI902416A patent/FI95795C/fi not_active IP Right Cessation
- 1990-05-15 IE IE175090A patent/IE64671B1/en not_active IP Right Cessation
- 1990-05-15 KR KR1019900006897A patent/KR0169107B1/ko not_active IP Right Cessation
- 1990-05-15 NO NO902179A patent/NO177141C/no not_active IP Right Cessation
- 1990-05-16 ES ES90109226T patent/ES2066035T3/es not_active Expired - Lifetime
- 1990-05-16 DK DK90109226.2T patent/DK0398283T3/da active
- 1990-05-16 EP EP90109226A patent/EP0398283B1/en not_active Expired - Lifetime
- 1990-05-16 DE DE69013750T patent/DE69013750T2/de not_active Expired - Fee Related
- 1990-05-16 AT AT90109226T patent/ATE113597T1/de not_active IP Right Cessation
-
1995
- 1995-02-01 GR GR940403551T patent/GR3014893T3/el unknown
Also Published As
Publication number | Publication date |
---|---|
DK0398283T3 (da) | 1994-11-28 |
KR900018112A (ko) | 1990-12-20 |
FI95795C (fi) | 1996-03-25 |
NO902179D0 (no) | 1990-05-15 |
NO177141B (no) | 1995-04-18 |
FI95795B (fi) | 1995-12-15 |
TW207950B (pt) | 1993-06-21 |
ATE113597T1 (de) | 1994-11-15 |
HUT54657A (en) | 1991-03-28 |
DE69013750T2 (de) | 1995-05-24 |
EP0398283A1 (en) | 1990-11-22 |
ES2066035T3 (es) | 1995-03-01 |
CN1027369C (zh) | 1995-01-11 |
CN1047292A (zh) | 1990-11-28 |
AU5491490A (en) | 1990-11-22 |
KR0169107B1 (ko) | 1999-01-15 |
DE69013750D1 (de) | 1994-12-08 |
AU626418B2 (en) | 1992-07-30 |
JPH0311067A (ja) | 1991-01-18 |
IL94377A0 (en) | 1991-03-10 |
FI902416A0 (fi) | 1990-05-15 |
GR3014893T3 (en) | 1995-05-31 |
NO177141C (no) | 1995-07-26 |
NO902179L (no) | 1990-11-19 |
HU903031D0 (en) | 1990-09-28 |
JP3014001B2 (ja) | 2000-02-28 |
NZ233641A (en) | 1992-07-28 |
IE64671B1 (en) | 1995-08-23 |
EP0398283B1 (en) | 1994-11-02 |
HU214322B (hu) | 1998-03-02 |
IE901750L (en) | 1990-11-16 |
IL94377A (en) | 1997-01-10 |
PT94042B (pt) | 1997-05-28 |
ZA903588B (en) | 1991-02-27 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FG3A | Patent granted, date of granting |
Effective date: 19970226 |
|
MM3A | Annulment or lapse |
Free format text: LAPSE DUE TO NON-PAYMENT OF FEES Effective date: 20040826 |