PT84064B - Processo para a preparacao de novos derivados de aminoacidos e de composicoes farmaceuticas que os contem - Google Patents

Processo para a preparacao de novos derivados de aminoacidos e de composicoes farmaceuticas que os contem

Info

Publication number
PT84064B
PT84064B PT84064A PT8406487A PT84064B PT 84064 B PT84064 B PT 84064B PT 84064 A PT84064 A PT 84064A PT 8406487 A PT8406487 A PT 8406487A PT 84064 B PT84064 B PT 84064B
Authority
PT
Portugal
Prior art keywords
amino acid
pharmaceutical compositions
compositions containing
acid derivatives
new amino
Prior art date
Application number
PT84064A
Other languages
English (en)
Other versions
PT84064A (en
Inventor
Ursula Sonnewald
Original Assignee
Novo Industri As
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from DK5186A external-priority patent/DK5186D0/da
Priority claimed from DK95686A external-priority patent/DK95686D0/da
Application filed by Novo Industri As filed Critical Novo Industri As
Publication of PT84064A publication Critical patent/PT84064A/pt
Publication of PT84064B publication Critical patent/PT84064B/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/08Antiepileptics; Anticonvulsants
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/06Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D409/00Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/06Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pain & Pain Management (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
PT84064A 1986-01-07 1987-01-06 Processo para a preparacao de novos derivados de aminoacidos e de composicoes farmaceuticas que os contem PT84064B (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DK5186A DK5186D0 (da) 1986-01-07 1986-01-07 Aminosyrer
DK95686A DK95686D0 (pt) 1986-03-03 1986-03-03

Publications (2)

Publication Number Publication Date
PT84064A PT84064A (en) 1987-02-01
PT84064B true PT84064B (pt) 1989-07-31

Family

ID=26063196

Family Applications (1)

Application Number Title Priority Date Filing Date
PT84064A PT84064B (pt) 1986-01-07 1987-01-06 Processo para a preparacao de novos derivados de aminoacidos e de composicoes farmaceuticas que os contem

Country Status (12)

Country Link
US (1) US4931450A (pt)
EP (1) EP0231996B1 (pt)
JP (1) JPH0791289B2 (pt)
AU (1) AU600248B2 (pt)
CA (1) CA1297105C (pt)
DE (1) DE3787657T2 (pt)
DK (1) DK165692C (pt)
ES (1) ES2059360T3 (pt)
FI (1) FI89481C (pt)
IL (1) IL81179A (pt)
NO (1) NO170976C (pt)
PT (1) PT84064B (pt)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DK704488D0 (da) * 1988-12-19 1988-12-19 Novo Industri As Nye n-substituerede azaheterocykliske carboxylsyrer
DK288385D0 (da) * 1985-06-26 1985-06-26 Novo Industri As Aminosyrederivater
DK270488D0 (da) * 1988-05-18 1988-05-18 Novo Industri As Hidtil ukendte o-substituerede ketoximer
DK588189D0 (da) * 1989-11-22 1989-11-22 Novo Nordisk As Nye heterocykliske carboxylsyrer
US5112980A (en) * 1989-12-27 1992-05-12 Monsanto Company Process of preparing substituted pyridine compounds
US5962449A (en) 1995-04-07 1999-10-05 Novo Nordisk A/S Tricyclic compounds in treating hyperalgesic conditions and NIDDM
US6191165B1 (en) 1996-05-31 2001-02-20 Allelix Neuroscience Inc. Pharmaceutical for treatment of neurological and neuropsychiatric disorders
WO1997049403A1 (en) * 1996-06-27 1997-12-31 University College Dublin Use of nipecotic acid or guvacine derivatives for the manufacture of a medicament for the treatment of postischemic neurodegenerative disorders
US6503926B2 (en) 1998-09-04 2003-01-07 Millennium Pharmaceuticals, Inc. Chemokine receptor antagonists and methods of use therefor
US6288083B1 (en) 1998-09-04 2001-09-11 Millennium Pharmaceuticals, Inc. Chemokine receptor antagonists and methods of use therefor
DE19840611A1 (de) * 1998-09-05 2000-03-09 Klaus Wanner GABA-uptake-Inhibitoren mit Pyrrolidinstruktur
CZ20032503A3 (cs) 2001-02-16 2004-02-18 Allelix Neuroscience, Inc. Inhibitory GlyT - 1
US7189757B2 (en) * 2001-10-16 2007-03-13 Hypnion, Inc. Treatment of sleep disorders using CNS target modulators
US7355042B2 (en) * 2001-10-16 2008-04-08 Hypnion, Inc. Treatment of CNS disorders using CNS target modulators
US20050009730A1 (en) * 2001-10-16 2005-01-13 Dale Edgar Treatment of cns disorders using cns target modulators
CN1382441A (zh) * 2002-05-21 2002-12-04 中国科学院上海生命科学研究院 γ-氨基丁酸转运蛋白抑制剂在制备镇痛药物中的应用

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU552050B2 (en) * 1981-05-26 1986-05-22 Smithkline Beckman Corporation N-substituted azeheterocyclic carboxylic acids and their esters
US4383999A (en) * 1981-05-26 1983-05-17 Smithkline Beckman Corporation Inhibition of GABA uptake by N-substituted azaheterocyclic carboxylic acids and their esters
US4681884A (en) * 1983-09-01 1987-07-21 Boehringer Ingelheim Pharmaceuticals, Inc. Diazine-ethenylphenyl oxamic acids and esters and salts thereof

Also Published As

Publication number Publication date
FI870059A (fi) 1987-07-08
JPH0791289B2 (ja) 1995-10-04
NO170976B (no) 1992-09-28
FI89481B (fi) 1993-06-30
DE3787657T2 (de) 1994-02-03
AU6719387A (en) 1987-07-09
EP0231996A3 (en) 1988-10-19
DE3787657D1 (de) 1993-11-11
US4931450A (en) 1990-06-05
EP0231996B1 (en) 1993-10-06
FI870059A0 (fi) 1987-01-07
EP0231996A2 (en) 1987-08-12
IL81179A0 (en) 1987-08-31
JPS62228073A (ja) 1987-10-06
DK165692C (da) 1993-11-08
IL81179A (en) 1992-02-16
AU600248B2 (en) 1990-08-09
ES2059360T3 (es) 1994-11-16
DK165692B (da) 1993-01-04
NO870049L (no) 1987-07-08
PT84064A (en) 1987-02-01
DK3887D0 (pt) 1987-01-06
DK3887A (pt) 1987-09-17
CA1297105C (en) 1992-03-10
FI89481C (fi) 1993-10-11
NO870049D0 (no) 1987-01-06
NO170976C (no) 1993-01-06

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Legal Events

Date Code Title Description
PD3A Change of proprietorship
MM3A Annulment or lapse

Free format text: LAPSE DUE TO NON-PAYMENT OF FEES

Effective date: 20000731