ES2059360T3 - Nuevos derivados de aminoacidos. - Google Patents

Nuevos derivados de aminoacidos.

Info

Publication number
ES2059360T3
ES2059360T3 ES87300064T ES87300064T ES2059360T3 ES 2059360 T3 ES2059360 T3 ES 2059360T3 ES 87300064 T ES87300064 T ES 87300064T ES 87300064 T ES87300064 T ES 87300064T ES 2059360 T3 ES2059360 T3 ES 2059360T3
Authority
ES
Spain
Prior art keywords
amino acid
acid derivatives
new amino
derivatives
imidazolito
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
ES87300064T
Other languages
English (en)
Inventor
Ursula Sonnewald
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Novo Nordisk AS
Original Assignee
Novo Nordisk AS
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from DK5186A external-priority patent/DK5186D0/da
Priority claimed from DK95686A external-priority patent/DK95686D0/da
Application filed by Novo Nordisk AS filed Critical Novo Nordisk AS
Application granted granted Critical
Publication of ES2059360T3 publication Critical patent/ES2059360T3/es
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/08—Antiepileptics; Anticonvulsants
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/06—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pain & Pain Management (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biomedical Technology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

DERIVADOS DE FENILBUTENO QUE TIENEN, OPCIONALMENTE GRUPOS SUSTITUIDOS FENILO Y PIRROLILO, FURANILO, PIRIDILO, PIRAZILO, IMIDAZOLITO, PIRAZOLILO, TETRAHIDROFURANILO, PIPERIDINILO, PIPERAZINILO O ALQUILTIENILO EN LA POSICION 4 Y 3-CARBOXIPIPERIDIN-1ILO, 3-CARBOXITETRAHIDROPIRIDIN-1-ILO O 3-CARBOXIMETILPIRROLIDIN-1-ILO EN LA POSICION 1. POTENCIAN LA NEUROTRANSMISION GABA-ERGICA.
ES87300064T 1986-01-07 1987-01-06 Nuevos derivados de aminoacidos. Expired - Lifetime ES2059360T3 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DK5186A DK5186D0 (da) 1986-01-07 1986-01-07 Aminosyrer
DK95686A DK95686D0 (es) 1986-03-03 1986-03-03

Publications (1)

Publication Number Publication Date
ES2059360T3 true ES2059360T3 (es) 1994-11-16

Family

ID=26063196

Family Applications (1)

Application Number Title Priority Date Filing Date
ES87300064T Expired - Lifetime ES2059360T3 (es) 1986-01-07 1987-01-06 Nuevos derivados de aminoacidos.

Country Status (12)

Country Link
US (1) US4931450A (es)
EP (1) EP0231996B1 (es)
JP (1) JPH0791289B2 (es)
AU (1) AU600248B2 (es)
CA (1) CA1297105C (es)
DE (1) DE3787657T2 (es)
DK (1) DK165692C (es)
ES (1) ES2059360T3 (es)
FI (1) FI89481C (es)
IL (1) IL81179A (es)
NO (1) NO170976C (es)
PT (1) PT84064B (es)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DK704488D0 (da) * 1988-12-19 1988-12-19 Novo Industri As Nye n-substituerede azaheterocykliske carboxylsyrer
DK288385D0 (da) * 1985-06-26 1985-06-26 Novo Industri As Aminosyrederivater
DK270488D0 (da) * 1988-05-18 1988-05-18 Novo Industri As Hidtil ukendte o-substituerede ketoximer
DK588189D0 (da) * 1989-11-22 1989-11-22 Novo Nordisk As Nye heterocykliske carboxylsyrer
US5112980A (en) * 1989-12-27 1992-05-12 Monsanto Company Process of preparing substituted pyridine compounds
US5962449A (en) 1995-04-07 1999-10-05 Novo Nordisk A/S Tricyclic compounds in treating hyperalgesic conditions and NIDDM
US6191165B1 (en) 1996-05-31 2001-02-20 Allelix Neuroscience Inc. Pharmaceutical for treatment of neurological and neuropsychiatric disorders
WO1997049403A1 (en) * 1996-06-27 1997-12-31 University College Dublin Use of nipecotic acid or guvacine derivatives for the manufacture of a medicament for the treatment of postischemic neurodegenerative disorders
US6288083B1 (en) 1998-09-04 2001-09-11 Millennium Pharmaceuticals, Inc. Chemokine receptor antagonists and methods of use therefor
US6503926B2 (en) 1998-09-04 2003-01-07 Millennium Pharmaceuticals, Inc. Chemokine receptor antagonists and methods of use therefor
DE19840611A1 (de) * 1998-09-05 2000-03-09 Klaus Wanner GABA-uptake-Inhibitoren mit Pyrrolidinstruktur
CZ20032503A3 (cs) 2001-02-16 2004-02-18 Allelix Neuroscience, Inc. Inhibitory GlyT - 1
US7189757B2 (en) * 2001-10-16 2007-03-13 Hypnion, Inc. Treatment of sleep disorders using CNS target modulators
EP1443929A4 (en) * 2001-10-16 2008-02-06 Hypnion Inc TREATMENT OF CNS DISTURBANCES WITH CNS TARGET MODULATORS
US7355042B2 (en) * 2001-10-16 2008-04-08 Hypnion, Inc. Treatment of CNS disorders using CNS target modulators
CN1382441A (zh) * 2002-05-21 2002-12-04 中国科学院上海生命科学研究院 γ－氨基丁酸转运蛋白抑制剂在制备镇痛药物中的应用

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU552050B2 (en) * 1981-05-26 1986-05-22 Smithkline Beckman Corporation N-substituted azeheterocyclic carboxylic acids and their esters
US4383999A (en) * 1981-05-26 1983-05-17 Smithkline Beckman Corporation Inhibition of GABA uptake by N-substituted azaheterocyclic carboxylic acids and their esters
US4681884A (en) * 1983-09-01 1987-07-21 Boehringer Ingelheim Pharmaceuticals, Inc. Diazine-ethenylphenyl oxamic acids and esters and salts thereof

Also Published As

Publication number Publication date
FI89481B (fi) 1993-06-30
AU600248B2 (en) 1990-08-09
EP0231996A3 (en) 1988-10-19
NO170976B (no) 1992-09-28
DK165692B (da) 1993-01-04
US4931450A (en) 1990-06-05
DK165692C (da) 1993-11-08
NO870049L (no) 1987-07-08
NO170976C (no) 1993-01-06
EP0231996B1 (en) 1993-10-06
IL81179A0 (en) 1987-08-31
DK3887D0 (es) 1987-01-06
CA1297105C (en) 1992-03-10
FI870059A (fi) 1987-07-08
PT84064B (pt) 1989-07-31
NO870049D0 (no) 1987-01-06
FI89481C (fi) 1993-10-11
JPS62228073A (ja) 1987-10-06
AU6719387A (en) 1987-07-09
PT84064A (en) 1987-02-01
DK3887A (es) 1987-09-17
DE3787657T2 (de) 1994-02-03
FI870059A0 (fi) 1987-01-07
IL81179A (en) 1992-02-16
JPH0791289B2 (ja) 1995-10-04
DE3787657D1 (de) 1993-11-11
EP0231996A2 (en) 1987-08-12

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