PT81659B - Processo para a preparacao de aminoacil-labdanos e de composicoes farmaceuticas que os contem - Google Patents

Processo para a preparacao de aminoacil-labdanos e de composicoes farmaceuticas que os contem

Info

Publication number
PT81659B
PT81659B PT81659A PT8165985A PT81659B PT 81659 B PT81659 B PT 81659B PT 81659 A PT81659 A PT 81659A PT 8165985 A PT8165985 A PT 8165985A PT 81659 B PT81659 B PT 81659B
Authority
PT
Portugal
Prior art keywords
labdans
pharmaceutical compositions
compositions containing
aminoacyl
preparing
Prior art date
Application number
PT81659A
Other languages
English (en)
Other versions
PT81659A (en
Original Assignee
Hoechst Roussel Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoechst Roussel Pharma filed Critical Hoechst Roussel Pharma
Publication of PT81659A publication Critical patent/PT81659A/pt
Publication of PT81659B publication Critical patent/PT81659B/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H13/00Compounds containing saccharide radicals esterified by carbonic acid or derivatives thereof, or by organic acids, e.g. phosphonic acids
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D311/00Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings
    • C07D311/02Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D311/78Ring systems having three or more relevant rings
    • C07D311/92Naphthopyrans; Hydrogenated naphthopyrans
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D493/00Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system
    • C07D493/02Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system in which the condensed system contains two hetero rings
    • C07D493/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D497/00Heterocyclic compounds containing in the condensed system at least one hetero ring having oxygen and sulfur atoms as the only ring hetero atoms
    • C07D497/02Heterocyclic compounds containing in the condensed system at least one hetero ring having oxygen and sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D497/04Ortho-condensed systems
PT81659A 1984-12-14 1985-12-12 Processo para a preparacao de aminoacil-labdanos e de composicoes farmaceuticas que os contem PT81659B (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US68177984A 1984-12-14 1984-12-14

Publications (2)

Publication Number Publication Date
PT81659A PT81659A (en) 1986-01-01
PT81659B true PT81659B (pt) 1988-04-21

Family

ID=24736768

Family Applications (1)

Application Number Title Priority Date Filing Date
PT81659A PT81659B (pt) 1984-12-14 1985-12-12 Processo para a preparacao de aminoacil-labdanos e de composicoes farmaceuticas que os contem

Country Status (19)

Country Link
EP (1) EP0191166B1 (pt)
JP (1) JPS61145178A (pt)
KR (1) KR900007625B1 (pt)
AR (1) AR243877A1 (pt)
AT (1) ATE60767T1 (pt)
AU (2) AU577912B2 (pt)
CA (1) CA1307529C (pt)
DE (1) DE3581725D1 (pt)
DK (1) DK167218B1 (pt)
ES (1) ES8703460A1 (pt)
FI (1) FI87208C (pt)
GR (1) GR852981B (pt)
HU (1) HU201043B (pt)
IE (1) IE58698B1 (pt)
NO (1) NO171064C (pt)
NZ (1) NZ214532A (pt)
PH (1) PH24599A (pt)
PT (1) PT81659B (pt)
ZA (1) ZA859556B (pt)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3678736D1 (de) * 1985-03-01 1991-05-23 Hoechst Roussel Pharma Labdanderivate, verfahren zu deren herstellung und deren verwendung als arzneimittel.
IN163242B (pt) 1985-05-03 1988-08-27 Hoechst India
AU591196B2 (en) * 1985-11-15 1989-11-30 Nippon Kayaku Kabushiki Kaisha Novel forskolin derivatives
JPS6310783A (ja) * 1985-11-15 1988-01-18 Nippon Kayaku Co Ltd 新規フオルスコリン誘導体
US4734513A (en) * 1986-03-31 1988-03-29 Hoechst-Roussel Pharmaceuticals Inc. Method of synthesizing forskolin from 9-deoxyforskolin
US4740522A (en) * 1986-08-28 1988-04-26 Hoechst-Roussel Pharmaceuticals Inc. Oxolabdanes useful as pharmaceuticals for reducing intraocular pressure
US5247097A (en) * 1986-08-28 1993-09-21 Hoechst-Roussel Pharmaceuticals Incorporated Oxolabdanes
US4920146A (en) * 1986-12-29 1990-04-24 Hoechst Roussel Pharmaceuticals Inc. Carbamoyloxylabdane compounds useful in reducing intraocular pressure
US5646175A (en) * 1987-12-28 1997-07-08 Hoechst Marion Roussel, Inc. Carbamoyloxylabdane compounds
NZ223051A (en) * 1986-12-29 1990-06-26 Hoechst Roussel Pharma Carbamoyloxylabdane derivatives and pharmaceutical compositions
US5302730A (en) * 1987-06-29 1994-04-12 Nippon Kayaku Kk Process for the preparation of 6,7-diacyl-7-deacetylforskolin derivatives
US4916204A (en) * 1987-07-31 1990-04-10 Massachusetts Institute Of Technology Pure polyanhydride from dicarboxylic acid and coupling agent
US5846992A (en) * 1987-10-08 1998-12-08 Hoechst Marion Roussel, Inc. Synergistic intraocular pressure lowering combinations
US4902696A (en) * 1987-10-08 1990-02-20 Hoechst-Roussel Pharmaceuticals, Inc. Synergistic intraocular pressure lowering combinations
US4883793A (en) * 1988-05-09 1989-11-28 Hoechst-Roussel Pharmaceuticals Inc. Hydrazinocarbonyloxylabdanes for treating cardiac failure
US5051132A (en) * 1989-06-15 1991-09-24 Nippon Kayaku Kabushiki Kaisha Lyophilized preparation of 6-(3-dimethylaminopropionyl)forskolin

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2654796A1 (de) * 1976-12-03 1978-06-08 Hoechst Ag Polyoxygenierte labdan-derivate
IL59004A0 (en) * 1978-12-30 1980-03-31 Beecham Group Ltd Substituted benzamides their preparation and pharmaceutical compositions containing them
DE3678736D1 (de) * 1985-03-01 1991-05-23 Hoechst Roussel Pharma Labdanderivate, verfahren zu deren herstellung und deren verwendung als arzneimittel.

Also Published As

Publication number Publication date
FI854919A0 (fi) 1985-12-12
FI854919A (fi) 1986-06-15
IE58698B1 (en) 1993-11-03
NO855026L (no) 1986-06-16
AU620421B2 (en) 1992-02-20
EP0191166A2 (en) 1986-08-20
NO171064B (no) 1992-10-12
AU577912B2 (en) 1988-10-06
IE853160L (en) 1986-06-14
DK578585D0 (da) 1985-12-13
EP0191166A3 (en) 1988-03-02
PT81659A (en) 1986-01-01
AU3813289A (en) 1989-10-26
KR860004915A (ko) 1986-07-16
AU5131685A (en) 1986-07-17
ZA859556B (en) 1986-08-27
ES8703460A1 (es) 1987-02-16
ES549860A0 (es) 1987-02-16
FI87208B (fi) 1992-08-31
DK167218B1 (da) 1993-09-20
AR243877A1 (es) 1993-09-30
NO171064C (no) 1993-01-20
EP0191166B1 (en) 1991-02-06
NZ214532A (en) 1989-05-29
PH24599A (en) 1990-08-17
FI87208C (fi) 1992-12-10
GR852981B (pt) 1986-04-08
JPS61145178A (ja) 1986-07-02
DE3581725D1 (de) 1991-03-14
CA1307529C (en) 1992-09-15
ATE60767T1 (de) 1991-02-15
KR900007625B1 (ko) 1990-10-17
HU201043B (en) 1990-09-28
HUT40636A (en) 1987-01-28
DK578585A (da) 1986-06-15

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Effective date: 19950430