PT90591B - Processo aperfeicoado para a preparacao de acidos 5-amino-7-(amino-substituido)-quinolina-3-carboxilicos - Google Patents

Processo aperfeicoado para a preparacao de acidos 5-amino-7-(amino-substituido)-quinolina-3-carboxilicos Download PDF

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Publication number
PT90591B
PT90591B PT90591A PT9059189A PT90591B PT 90591 B PT90591 B PT 90591B PT 90591 A PT90591 A PT 90591A PT 9059189 A PT9059189 A PT 9059189A PT 90591 B PT90591 B PT 90591B
Authority
PT
Portugal
Prior art keywords
process according
group
general formula
hydrogen atom
amino
Prior art date
Application number
PT90591A
Other languages
English (en)
Portuguese (pt)
Other versions
PT90591A (pt
Inventor
James Norton Wemple
Original Assignee
Warner Lambert Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Warner Lambert Co filed Critical Warner Lambert Co
Publication of PT90591A publication Critical patent/PT90591A/pt
Publication of PT90591B publication Critical patent/PT90591B/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/48—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
    • C07D215/54—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3
    • C07D215/56—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3 with oxygen atoms in position 4
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
  • Peptides Or Proteins (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Quinoline Compounds (AREA)
PT90591A 1988-05-18 1989-05-17 Processo aperfeicoado para a preparacao de acidos 5-amino-7-(amino-substituido)-quinolina-3-carboxilicos PT90591B (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US19558088A 1988-05-18 1988-05-18
US33184589A 1989-04-04 1989-04-04

Publications (2)

Publication Number Publication Date
PT90591A PT90591A (pt) 1989-11-30
PT90591B true PT90591B (pt) 1994-09-30

Family

ID=26891107

Family Applications (1)

Application Number Title Priority Date Filing Date
PT90591A PT90591B (pt) 1988-05-18 1989-05-17 Processo aperfeicoado para a preparacao de acidos 5-amino-7-(amino-substituido)-quinolina-3-carboxilicos

Country Status (11)

Country Link
EP (1) EP0342649B1 (ja)
JP (1) JPH0242060A (ja)
KR (1) KR900018069A (ja)
AT (1) ATE114649T1 (ja)
AU (1) AU609974B2 (ja)
DE (1) DE68919531D1 (ja)
DK (1) DK168865B1 (ja)
FI (1) FI892323A (ja)
NO (1) NO891952L (ja)
NZ (1) NZ229140A (ja)
PT (1) PT90591B (ja)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2147721T3 (es) 1990-04-18 2000-10-01 Procter & Gamble Pharma Quinolonil lactamas antimicrobianas.
US5646163A (en) * 1992-10-30 1997-07-08 The Procter & Gamble Company Quinolone 5-(N-heterosubstituted amino) antimicrobials
TW252107B (ja) * 1993-08-27 1995-07-21 Hokuriku Pharmacetical Co Ltd
DE19546249A1 (de) * 1995-12-12 1997-06-19 Bayer Ag Neue Kristallmodifikation des 1-Cyclopropyl-7-([S,S]-2,8-diazabicyclo[4,3,0]non-8-yl)-6-fluor-1,4-dihydro-8-methoxy-4-oxo-3-chinolincarbonsäure Hydrochlorid (CDCH), Verfahren zu dessen Herstellung und diese enthaltende pharmazeutische Zubereitungen

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU594983B2 (en) * 1985-10-29 1990-03-22 Dainippon Pharmaceutical Co. Ltd. Novel quinoline derivatives and processes for preparation thereof
EP0242789A3 (en) * 1986-04-25 1990-09-05 Dainippon Pharmaceutical Co., Ltd. Novel quinoline derivates and processes for preparation thereof
DE3711193A1 (de) * 1987-04-02 1988-10-13 Bayer Ag 5-substituierte chinolon- und naphthyridoncarbonsaeure-derivate
CA1332605C (en) * 1988-10-03 1994-10-18 Yasuhiro Nishitani Pyridonecarboxylic acids

Also Published As

Publication number Publication date
AU3383789A (en) 1989-11-23
NO891952L (no) 1989-11-20
EP0342649A3 (en) 1990-12-19
ATE114649T1 (de) 1994-12-15
AU609974B2 (en) 1991-05-09
FI892323A0 (fi) 1989-05-15
DK239789A (da) 1989-11-19
EP0342649B1 (en) 1994-11-30
NO891952D0 (no) 1989-05-16
DE68919531D1 (de) 1995-01-12
DK168865B1 (da) 1994-06-27
DK239789D0 (da) 1989-05-17
EP0342649A2 (en) 1989-11-23
PT90591A (pt) 1989-11-30
NZ229140A (en) 1990-06-26
FI892323A (fi) 1989-11-19
KR900018069A (ko) 1990-12-20
JPH0242060A (ja) 1990-02-13

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FG3A Patent granted, date of granting

Effective date: 19940315

MM3A Annulment or lapse

Free format text: LAPSE DUE TO NON-PAYMENT OF FEES

Effective date: 19950930