PT2081937E - Moduladores de proteína-cinase de triazolo-piridazina - Google Patents
Moduladores de proteína-cinase de triazolo-piridazina Download PDFInfo
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- PT2081937E PT2081937E PT07854193T PT07854193T PT2081937E PT 2081937 E PT2081937 E PT 2081937E PT 07854193 T PT07854193 T PT 07854193T PT 07854193 T PT07854193 T PT 07854193T PT 2081937 E PT2081937 E PT 2081937E
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Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D519/00—Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US86255206P | 2006-10-23 | 2006-10-23 | |
| US87138406P | 2006-12-21 | 2006-12-21 | |
| US91375207P | 2007-04-24 | 2007-04-24 | |
| US95283307P | 2007-07-30 | 2007-07-30 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| PT2081937E true PT2081937E (pt) | 2012-10-15 |
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| PT07854193T PT2081937E (pt) | 2006-10-23 | 2007-10-18 | Moduladores de proteína-cinase de triazolo-piridazina |
Country Status (16)
| Country | Link |
|---|---|
| US (1) | US8071581B2 (https=) |
| EP (1) | EP2081937B1 (https=) |
| JP (1) | JP2010507577A (https=) |
| KR (1) | KR101083177B1 (https=) |
| AU (1) | AU2007309237B2 (https=) |
| BR (1) | BRPI0717317A2 (https=) |
| CA (1) | CA2667453A1 (https=) |
| DK (1) | DK2081937T3 (https=) |
| EA (1) | EA016527B1 (https=) |
| ES (1) | ES2393132T3 (https=) |
| MX (1) | MX2009004060A (https=) |
| PE (1) | PE20081256A1 (https=) |
| PL (1) | PL2081937T3 (https=) |
| PT (1) | PT2081937E (https=) |
| TW (1) | TW200833692A (https=) |
| WO (1) | WO2008051805A2 (https=) |
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| WO2002083139A1 (en) * | 2001-04-10 | 2002-10-24 | Merck & Co., Inc. | Inhibitors of akt activity |
| WO2002083675A2 (en) | 2001-04-10 | 2002-10-24 | Merck Sharp & Dohme Limited | Inhibitors of akt activity |
| WO2003014649A1 (en) * | 2001-08-10 | 2003-02-20 | Yokohama Tlo Company Ltd. | Heat transfer device |
| HUE030390T2 (en) * | 2005-12-21 | 2017-05-29 | Janssen Pharmaceutica Nv | Triazolopyridazines as tyrosine kinase modulators |
| JP2009538899A (ja) * | 2006-05-30 | 2009-11-12 | ファイザー・プロダクツ・インク | トリアゾロピリダジン誘導体 |
| PE20080403A1 (es) * | 2006-07-14 | 2008-04-25 | Amgen Inc | Derivados heterociclicos fusionados y metodos de uso |
-
2007
- 2007-10-18 CA CA002667453A patent/CA2667453A1/en not_active Abandoned
- 2007-10-18 AU AU2007309237A patent/AU2007309237B2/en not_active Ceased
- 2007-10-18 JP JP2009533536A patent/JP2010507577A/ja not_active Withdrawn
- 2007-10-18 PL PL07854193T patent/PL2081937T3/pl unknown
- 2007-10-18 US US12/442,987 patent/US8071581B2/en not_active Expired - Fee Related
- 2007-10-18 PT PT07854193T patent/PT2081937E/pt unknown
- 2007-10-18 DK DK07854193.5T patent/DK2081937T3/da active
- 2007-10-18 MX MX2009004060A patent/MX2009004060A/es not_active Application Discontinuation
- 2007-10-18 BR BRPI0717317-2A2A patent/BRPI0717317A2/pt not_active IP Right Cessation
- 2007-10-18 ES ES07854193T patent/ES2393132T3/es active Active
- 2007-10-18 EA EA200970402A patent/EA016527B1/ru not_active IP Right Cessation
- 2007-10-18 KR KR1020097007986A patent/KR101083177B1/ko not_active Expired - Fee Related
- 2007-10-18 EP EP07854193A patent/EP2081937B1/en active Active
- 2007-10-18 WO PCT/US2007/081832 patent/WO2008051805A2/en not_active Ceased
- 2007-10-22 TW TW096139481A patent/TW200833692A/zh unknown
- 2007-10-23 PE PE2007001436A patent/PE20081256A1/es not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| US8071581B2 (en) | 2011-12-06 |
| MX2009004060A (es) | 2009-06-19 |
| WO2008051805A3 (en) | 2008-07-10 |
| JP2010507577A (ja) | 2010-03-11 |
| WO2008051805A2 (en) | 2008-05-02 |
| PE20081256A1 (es) | 2008-10-13 |
| US20100120739A1 (en) | 2010-05-13 |
| TW200833692A (en) | 2008-08-16 |
| EP2081937A2 (en) | 2009-07-29 |
| EP2081937B1 (en) | 2012-09-12 |
| PL2081937T3 (pl) | 2013-01-31 |
| BRPI0717317A2 (pt) | 2013-10-22 |
| CA2667453A1 (en) | 2008-05-02 |
| ES2393132T3 (es) | 2012-12-18 |
| DK2081937T3 (da) | 2012-10-01 |
| KR101083177B1 (ko) | 2011-11-11 |
| AU2007309237B2 (en) | 2012-03-22 |
| EA016527B1 (ru) | 2012-05-30 |
| KR20090069303A (ko) | 2009-06-30 |
| EA200970402A1 (ru) | 2009-10-30 |
| AU2007309237A1 (en) | 2008-05-02 |
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