PT1620439E - Novos polimorfos de cloridrato de olanzapina - Google Patents

Novos polimorfos de cloridrato de olanzapina Download PDF

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Publication number
PT1620439E
PT1620439E PT04728854T PT04728854T PT1620439E PT 1620439 E PT1620439 E PT 1620439E PT 04728854 T PT04728854 T PT 04728854T PT 04728854 T PT04728854 T PT 04728854T PT 1620439 E PT1620439 E PT 1620439E
Authority
PT
Portugal
Prior art keywords
new polymorphs
new
hydrochloride
olanzapine
olanzapine hydrochloride
Prior art date
Application number
PT04728854T
Other languages
English (en)
Inventor
Gyula Simig
Janos Petho
Jozsef Barkoczy
Peter Kotay Nagy
Zsuzsa Szent-Kirallyi
Original Assignee
Egis Gyogyszergyar Nyrt
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Egis Gyogyszergyar Nyrt filed Critical Egis Gyogyszergyar Nyrt
Publication of PT1620439E publication Critical patent/PT1620439E/pt

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D495/00Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Neurology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Biomedical Technology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Neurosurgery (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Psychiatry (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
PT04728854T 2003-04-22 2004-04-22 Novos polimorfos de cloridrato de olanzapina PT1620439E (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
HU0301082A HU226410B1 (en) 2003-04-22 2003-04-22 Novel polymorphous forms of olanzapine hydrochlorides, process for producing them, use thereof and pharmaceutical compositions containing them

Publications (1)

Publication Number Publication Date
PT1620439E true PT1620439E (pt) 2008-10-23

Family

ID=89981318

Family Applications (1)

Application Number Title Priority Date Filing Date
PT04728854T PT1620439E (pt) 2003-04-22 2004-04-22 Novos polimorfos de cloridrato de olanzapina

Country Status (24)

Country Link
US (1) US7951798B2 (pt)
EP (1) EP1620439B1 (pt)
JP (1) JP4763594B2 (pt)
KR (1) KR20060004954A (pt)
CN (2) CN101468999B (pt)
AT (1) ATE401332T1 (pt)
AU (1) AU2004232544B2 (pt)
BG (1) BG109361A (pt)
CA (1) CA2522734C (pt)
CZ (1) CZ2005684A3 (pt)
DE (1) DE602004015096D1 (pt)
DK (1) DK1620439T3 (pt)
EA (1) EA008376B1 (pt)
ES (1) ES2310728T3 (pt)
HR (1) HRP20080479T3 (pt)
HU (1) HU226410B1 (pt)
IL (1) IL171522A (pt)
PL (2) PL1620439T3 (pt)
PT (1) PT1620439E (pt)
SI (1) SI1620439T1 (pt)
SK (1) SK50942005A3 (pt)
UA (1) UA80881C2 (pt)
WO (1) WO2004094433A1 (pt)
ZA (1) ZA200508936B (pt)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2003300324A1 (en) * 2002-12-24 2004-07-22 Teva Pharmaceutical Industries Ltd. Novel crystal forms of olanzapine, methods for their preparation and method for the preparation of known olanzapine crystal forms
SI21850A (sl) * 2004-07-28 2006-02-28 Krka, Tovarna Zdravil, D.D., Novo Mesto Soli olanzapina in njihova pretvorba v prosto bazo olanzapina
KR20130030305A (ko) * 2004-11-16 2013-03-26 엘란 파마 인터내셔널 리미티드 주사가능한 나노입자형 올란자핀 제형
HUP0501046A2 (en) 2005-11-11 2007-08-28 Egis Gyogyszergyar Nyilvanosan Process for the preparation of olanzapine
KR20170091770A (ko) * 2006-07-10 2017-08-09 파이온 유케이 리미티드 속효형 벤조디아제핀 염 및 이의 중합체 형태
WO2008151430A1 (en) * 2007-06-14 2008-12-18 Apotex Pharmachem Inc. Novel processes to form-i of olanzapine
WO2009124321A1 (en) * 2008-04-04 2009-10-08 University Of Massachusetts Methods and compositions for improving the production of fuels in microorganisms
EP2450039A1 (en) 2010-11-08 2012-05-09 PAION UK Ltd. Dosing regimen for sedation with CNS 7056 (Remimazolam)
WO2013009517A1 (en) * 2011-07-08 2013-01-17 Eli Lilly And Company (THIENO[2,3-b][1,5]BENZOXAZEPIN-4-YL)PIPERAZIN-1-YL COMPOUNDS AS DUAL ACTIVITY H1 INVERSE AGONISTS/5-HT2A ANTAGONISTS
CN104955827B (zh) * 2013-01-14 2017-06-30 伊莱利利公司 作为双重活性H1反向激动剂/5‑HT2A拮抗剂的(噻吩并[2,3‑b][1,5]苯并氧杂氮杂*‑4‑基)哌嗪‑1‑基化合物
AR094963A1 (es) 2013-03-04 2015-09-09 Ono Pharmaceutical Co Reacción de oxidación excelente en el índice de conversión
KR101489062B1 (ko) * 2013-03-28 2015-02-02 동아에스티 주식회사 고순도의 올란자핀 및 이의 결정형 ii의 제조방법
JP6940866B2 (ja) * 2017-06-21 2021-09-29 国立研究開発法人情報通信研究機構 半導体光デバイス、半導体光源、光集積回路、及び半導体光デバイスの製造方法

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5229382A (en) * 1990-04-25 1993-07-20 Lilly Industries Limited 2-methyl-thieno-benzodiazepine
GB9009229D0 (en) * 1990-04-25 1990-06-20 Lilly Industries Ltd Pharmaceutical compounds
UA73715C2 (en) * 1997-09-30 2005-09-15 Lilly Co Eli Pharmaceutically acceptable formulation of olanzapine pamoate and its use for treatment
PT1468689E (pt) * 1998-09-30 2007-07-09 Lilly Co Eli Formulação de 2-metil-tieno-benzodiazepina.
UA80095C2 (en) * 2001-07-20 2007-08-27 Lilly Co Eli 2 methyl-thieno-benzodiazepine lyophilized formulation and method for the preparation thereof
ATE504588T1 (de) * 2004-01-27 2011-04-15 Synthon Bv Stabile salze von olanzapin

Also Published As

Publication number Publication date
ES2310728T3 (es) 2009-01-16
CN100471859C (zh) 2009-03-25
US7951798B2 (en) 2011-05-31
BG109361A (bg) 2006-09-29
KR20060004954A (ko) 2006-01-16
IL171522A (en) 2010-05-31
DK1620439T3 (da) 2008-11-17
HUP0301082A2 (hu) 2004-12-28
PL378061A1 (pl) 2006-02-20
CN1777613A (zh) 2006-05-24
EP1620439B1 (en) 2008-07-16
JP2006524219A (ja) 2006-10-26
WO2004094433A1 (en) 2004-11-04
CZ2005684A3 (cs) 2006-01-11
ATE401332T1 (de) 2008-08-15
HRP20080479T3 (en) 2008-10-31
CN101468999A (zh) 2009-07-01
US20070004706A1 (en) 2007-01-04
JP4763594B2 (ja) 2011-08-31
EP1620439A1 (en) 2006-02-01
SK50942005A3 (sk) 2006-02-02
DE602004015096D1 (de) 2008-08-28
CA2522734A1 (en) 2004-11-04
AU2004232544B2 (en) 2010-06-03
CN101468999B (zh) 2012-05-09
HU226410B1 (en) 2008-11-28
PL1620439T3 (pl) 2009-02-27
ZA200508936B (en) 2008-07-30
EA008376B1 (ru) 2007-04-27
HU0301082D0 (en) 2003-06-28
CA2522734C (en) 2010-05-25
AU2004232544A1 (en) 2004-11-04
SI1620439T1 (sl) 2009-06-30
UA80881C2 (en) 2007-11-12
EA200501633A1 (ru) 2006-04-28

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