PT1404317E - Derivados de 5-halo-triptamina utilizados como ligandos dos receptores serotoninérgicos 5-ht6 e/ou 5-ht7 - Google Patents
Derivados de 5-halo-triptamina utilizados como ligandos dos receptores serotoninérgicos 5-ht6 e/ou 5-ht7 Download PDFInfo
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- PT1404317E PT1404317E PT02745793T PT02745793T PT1404317E PT 1404317 E PT1404317 E PT 1404317E PT 02745793 T PT02745793 T PT 02745793T PT 02745793 T PT02745793 T PT 02745793T PT 1404317 E PT1404317 E PT 1404317E
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Classifications
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- C—CHEMISTRY; METALLURGY
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- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/10—Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
- C07D209/14—Radicals substituted by nitrogen atoms, not forming part of a nitro radical
- C07D209/16—Tryptamines
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
- A61K31/403—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
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- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
- A61K31/403—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
- A61K31/404—Indoles, e.g. pindolol
- A61K31/405—Indole-alkanecarboxylic acids; Derivatives thereof, e.g. tryptophan, indomethacin
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- A61P9/12—Antihypertensives
Landscapes
- Health & Medical Sciences (AREA)
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- Organic Chemistry (AREA)
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- Anesthesiology (AREA)
- Hospice & Palliative Care (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Indole Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| IT2001RM000356A ITRM20010356A1 (it) | 2001-06-21 | 2001-06-21 | "5-alogeno derivati della triptamina utili come ligandi del recettore5-ht6 e/o 5-ht7 della serotonina. |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| PT1404317E true PT1404317E (pt) | 2009-02-23 |
Family
ID=11455609
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| PT02745793T PT1404317E (pt) | 2001-06-21 | 2002-06-17 | Derivados de 5-halo-triptamina utilizados como ligandos dos receptores serotoninérgicos 5-ht6 e/ou 5-ht7 |
Country Status (21)
| Country | Link |
|---|---|
| US (1) | US7098233B2 (enExample) |
| EP (1) | EP1404317B1 (enExample) |
| JP (2) | JP4683839B2 (enExample) |
| KR (1) | KR100885308B1 (enExample) |
| CN (1) | CN100482223C (enExample) |
| AT (1) | ATE416767T1 (enExample) |
| AU (1) | AU2002317482B2 (enExample) |
| BR (1) | BR0210538A (enExample) |
| CA (1) | CA2455296C (enExample) |
| CY (1) | CY1108879T1 (enExample) |
| CZ (1) | CZ20033314A3 (enExample) |
| DE (1) | DE60230270D1 (enExample) |
| DK (1) | DK1404317T3 (enExample) |
| ES (1) | ES2319107T3 (enExample) |
| HU (1) | HUP0400250A3 (enExample) |
| IT (1) | ITRM20010356A1 (enExample) |
| MX (1) | MXPA03011510A (enExample) |
| PL (1) | PL367618A1 (enExample) |
| PT (1) | PT1404317E (enExample) |
| SK (1) | SK287828B6 (enExample) |
| WO (1) | WO2003000252A1 (enExample) |
Families Citing this family (35)
| Publication number | Priority date | Publication date | Assignee | Title |
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| AR039127A1 (es) * | 2002-03-27 | 2005-02-09 | Glaxo Group Ltd | Compuesto de quinolina, procedimiento para su preparacion, composicion farmaceutica que lo comprende y uso del mismo para la fabricacion de un medicamento |
| NZ544331A (en) | 2003-07-22 | 2010-03-26 | Arena Pharm Inc | Diaryl and arylheteroaryl urea derivatives as modulators of the 5-HT2A serotonin receptor useful for the prophylaxis and treatment of disorders related thereto |
| US8086315B2 (en) | 2004-02-12 | 2011-12-27 | Asap Medical, Inc. | Cardiac stimulation apparatus and method for the control of hypertension |
| CA2557158A1 (en) * | 2004-02-20 | 2005-09-01 | Astellas Pharma Inc. | Prophylactic antimigraine agents |
| US20080171788A1 (en) * | 2005-02-08 | 2008-07-17 | Shinobu Akuzawa | Medicament For Irritable Bowel Syndrome |
| EP1923387B1 (en) | 2005-08-08 | 2011-10-19 | Astellas Pharma Inc. | Acylguanidine derivative or salt thereof |
| WO2007046112A1 (en) * | 2005-10-19 | 2007-04-26 | Suven Life Sciences Inc. | Arylthioether tryptamine derivatives as functional 5-ht6 ligands |
| WO2007097276A1 (ja) * | 2006-02-20 | 2007-08-30 | Astellas Pharma Inc. | ピロール誘導体またはその塩 |
| EP2120950B1 (en) * | 2007-03-21 | 2012-07-04 | Glaxo Group Limited | Use of quinoline derivatives in the treatment of pain |
| EP2209380A4 (en) * | 2007-10-09 | 2011-09-14 | Mark T Hamann | METHOD OF USE OF COMPOSITIONS WITH ANTIDEPRESSIVE EFFICACY, MOOD EFFICACY AND OTHER NEUROLOGICAL EFFECTIVENESS AND COMPOSITIONS THEREOF |
| EP2254564A1 (en) | 2007-12-12 | 2010-12-01 | Glaxo Group Limited | Combinations comprising 3-phenylsulfonyl-8-piperazinyl-1yl-quinoline |
| WO2009123714A2 (en) | 2008-04-02 | 2009-10-08 | Arena Pharmaceuticals, Inc. | Processes for the preparation of pyrazole derivatives useful as modulators of the 5-ht2a serotonin receptor |
| US9126946B2 (en) | 2008-10-28 | 2015-09-08 | Arena Pharmaceuticals, Inc. | Processes useful for the preparation of 1-[3-(4-bromo-2-methyl-2H-pyrazol-3-yl)-4-methoxy-phenyl]-3-(2,4-difluoro-phenyl)urea and crystalline forms related thereto |
| CA2842455A1 (en) * | 2011-08-05 | 2013-02-14 | Sucampo Ag | Method for treating schizophrenia |
| CN102816103B (zh) * | 2012-08-20 | 2014-05-07 | 冉瑞琼 | 硫化天冬氨酸修饰的退黑素衍生物及其应用 |
| US9008769B2 (en) | 2012-12-21 | 2015-04-14 | Backbeat Medical, Inc. | Methods and systems for lowering blood pressure through reduction of ventricle filling |
| US9370662B2 (en) | 2013-12-19 | 2016-06-21 | Backbeat Medical, Inc. | Methods and systems for controlling blood pressure by controlling atrial pressure |
| CN104529865B (zh) * | 2014-12-12 | 2017-02-01 | 广东东阳光药业有限公司 | 苄胺类衍生物及其在药物上的应用 |
| JP2018516992A (ja) | 2015-06-12 | 2018-06-28 | アクソファント サイエンシーズ ゲーエムベーハーＡｘｏｖａｎｔ Ｓｃｉｅｎｃｅｓ Ｇｍｂｈ | レム睡眠行動障害の予防および処置のために有用なジアリールおよびアリールヘテロアリール尿素誘導体 |
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2001
- 2001-06-21 IT IT2001RM000356A patent/ITRM20010356A1/it unknown
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2002
- 2002-06-17 PL PL02367618A patent/PL367618A1/xx not_active IP Right Cessation
- 2002-06-17 CZ CZ20033314A patent/CZ20033314A3/cs unknown
- 2002-06-17 CN CNB02814337XA patent/CN100482223C/zh not_active Expired - Fee Related
- 2002-06-17 AU AU2002317482A patent/AU2002317482B2/en not_active Ceased
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- 2002-06-17 EP EP02745793A patent/EP1404317B1/en not_active Expired - Lifetime
- 2002-06-17 AT AT02745793T patent/ATE416767T1/de active
- 2002-06-17 SK SK38-2004A patent/SK287828B6/sk not_active IP Right Cessation
- 2002-06-17 KR KR1020037016564A patent/KR100885308B1/ko not_active Expired - Fee Related
- 2002-06-17 PT PT02745793T patent/PT1404317E/pt unknown
- 2002-06-17 DE DE60230270T patent/DE60230270D1/de not_active Expired - Lifetime
- 2002-06-17 ES ES02745793T patent/ES2319107T3/es not_active Expired - Lifetime
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- 2002-06-17 JP JP2003506898A patent/JP4683839B2/ja not_active Expired - Fee Related
- 2002-06-17 BR BR0210538-1A patent/BR0210538A/pt not_active Application Discontinuation
- 2002-06-17 HU HU0400250A patent/HUP0400250A3/hu unknown
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| Publication number | Publication date |
|---|---|
| DE60230270D1 (de) | 2009-01-22 |
| BR0210538A (pt) | 2004-06-22 |
| CY1108879T1 (el) | 2014-07-02 |
| KR100885308B1 (ko) | 2009-02-24 |
| AU2002317482B2 (en) | 2007-08-16 |
| ITRM20010356A1 (it) | 2002-12-23 |
| ES2319107T3 (es) | 2009-05-04 |
| CZ20033314A3 (cs) | 2004-08-18 |
| DK1404317T3 (da) | 2009-02-23 |
| HUP0400250A2 (hu) | 2004-08-30 |
| JP2011016835A (ja) | 2011-01-27 |
| CA2455296C (en) | 2010-08-17 |
| WO2003000252A1 (en) | 2003-01-03 |
| JP4683839B2 (ja) | 2011-05-18 |
| MXPA03011510A (es) | 2004-03-18 |
| HK1068792A1 (zh) | 2005-05-06 |
| JP2004534816A (ja) | 2004-11-18 |
| ITRM20010356A0 (it) | 2001-06-21 |
| SK382004A3 (en) | 2004-05-04 |
| CA2455296A1 (en) | 2003-01-03 |
| SK287828B6 (sk) | 2011-11-04 |
| PL367618A1 (en) | 2005-03-07 |
| US7098233B2 (en) | 2006-08-29 |
| EP1404317A1 (en) | 2004-04-07 |
| KR20040032113A (ko) | 2004-04-14 |
| US20040235899A1 (en) | 2004-11-25 |
| CN1535146A (zh) | 2004-10-06 |
| ATE416767T1 (de) | 2008-12-15 |
| EP1404317B1 (en) | 2008-12-10 |
| CN100482223C (zh) | 2009-04-29 |
| HUP0400250A3 (en) | 2008-03-28 |
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