PT1171444E - Pirido-tieno-diazepinas seu processo de preparacao e composicao farmaceuticas que as contem - Google Patents

Pirido-tieno-diazepinas seu processo de preparacao e composicao farmaceuticas que as contem

Info

Publication number
PT1171444E
PT1171444E PT00917149T PT00917149T PT1171444E PT 1171444 E PT1171444 E PT 1171444E PT 00917149 T PT00917149 T PT 00917149T PT 00917149 T PT00917149 T PT 00917149T PT 1171444 E PT1171444 E PT 1171444E
Authority
PT
Portugal
Prior art keywords
pirido
tieno
diazepines
preparation
pharmaceutical composition
Prior art date
Application number
PT00917149T
Other languages
English (en)
Inventor
Dennis Bigg
Anne-Marie Liberatore
Original Assignee
Conseils De R D App Sci S C R
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Conseils De R D App Sci S C R filed Critical Conseils De R D App Sci S C R
Publication of PT1171444E publication Critical patent/PT1171444E/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
    • C07D495/14—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/06—Antipsoriatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
    • A61P19/10—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/02—Drugs for disorders of the endocrine system of the hypothalamic hormones, e.g. TRH, GnRH, CRH, GRH, somatostatin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Diabetes (AREA)
  • Endocrinology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Rheumatology (AREA)
  • Dermatology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Obesity (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Hematology (AREA)
  • Emergency Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
PT00917149T 1999-04-09 2000-04-07 Pirido-tieno-diazepinas seu processo de preparacao e composicao farmaceuticas que as contem PT1171444E (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR9904440A FR2791980B1 (fr) 1999-04-09 1999-04-09 Pyrido-thieno-diazepines, leur procede de preparation, et les compositions pharmaceutiques les contenant

Publications (1)

Publication Number Publication Date
PT1171444E true PT1171444E (pt) 2003-11-28

Family

ID=9544211

Family Applications (1)

Application Number Title Priority Date Filing Date
PT00917149T PT1171444E (pt) 1999-04-09 2000-04-07 Pirido-tieno-diazepinas seu processo de preparacao e composicao farmaceuticas que as contem

Country Status (20)

Country Link
US (1) US6777408B1 (pt)
EP (1) EP1171444B1 (pt)
JP (1) JP4681737B2 (pt)
AR (1) AR028818A1 (pt)
AT (1) ATE244246T1 (pt)
AU (1) AU3825700A (pt)
CA (1) CA2369725C (pt)
CZ (1) CZ302455B6 (pt)
DE (1) DE60003662T2 (pt)
DK (1) DK1171444T3 (pt)
ES (1) ES2202091T3 (pt)
FR (1) FR2791980B1 (pt)
HU (1) HUP0200928A3 (pt)
MY (1) MY120085A (pt)
NO (1) NO20014803L (pt)
PL (1) PL207639B1 (pt)
PT (1) PT1171444E (pt)
RU (1) RU2245883C2 (pt)
TW (1) TW513433B (pt)
WO (1) WO2000061587A1 (pt)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7189856B2 (en) 2001-12-28 2007-03-13 Gideon Shapiro Non-peptide somatostatin receptor ligands
AU2007325315A1 (en) * 2006-11-28 2008-06-05 Kalypsys Inc Heterocyclic modulators of TGR5
WO2012075456A1 (en) 2010-12-02 2012-06-07 Constellation Pharmaceuticals Bromodomain inhibitors and uses thereof
AR084070A1 (es) 2010-12-02 2013-04-17 Constellation Pharmaceuticals Inc Inhibidores del bromodominio y usos de los mismos
US9422292B2 (en) 2011-05-04 2016-08-23 Constellation Pharmaceuticals, Inc. Bromodomain inhibitors and uses thereof
WO2012174487A2 (en) 2011-06-17 2012-12-20 Constellation Pharmaceuticals, Inc. Bromodomain inhibitors and uses thereof
WO2013184878A1 (en) 2012-06-06 2013-12-12 Constellation Pharmaceuticals, Inc. Benzo [b] isoxazoloazepine bromodomain inhibitors and uses thereof
TWI602820B (zh) 2012-06-06 2017-10-21 星宿藥物公司 溴域抑制劑及其用途
CA2952830C (en) 2014-06-20 2022-11-01 Constellation Pharmaceuticals, Inc. Crystalline forms of 2-((4s)-6-(4-chlorophenyl)-1-methyl-4h-benzo[c]isoxazolo[4,5-e]azepin-4-yl)acetamide

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3435974A1 (de) * 1984-10-01 1986-04-10 Boehringer Ingelheim KG, 6507 Ingelheim Diazepine enthaltende pharmazeutische zusammensetzungen mit paf-antagonistischer wirkung
NL9000627A (nl) * 1990-03-29 1991-10-16 Scras Werkwijze ter bereiding van nieuwe thienotriazolo-diazepines.
US5593988A (en) * 1991-10-11 1997-01-14 Yoshitomi Pharmaceutical Industries, Ltd. Therapeutic agent for osteoporosis and diazepine compound
WO1994006802A1 (en) * 1992-09-18 1994-03-31 Yoshitomi Pharmaceutical Industries, Ltd. Thienodiazepine compound and medicinal use thereof
CA2144985A1 (en) * 1992-09-18 1994-03-31 Minoru Moriwaki Thienodiazepine compounds and their pharmaceutical use
DE19636769A1 (de) * 1996-09-10 1998-03-12 Basf Ag 3-Substituierte Pyrido [4',3':4,5]thieno[2,3-d]pyrimidin-Derivate, ihre Herstellung und Verwendung
CZ20004640A3 (cs) * 1999-06-15 2001-06-13 Sod Conseils Rech Applic Nové diazepiny, kompozice s jejich obsahem a léčivo pro léčení patologických stavů nebo onemocnění při kterých působí receptory somatostatinu

Also Published As

Publication number Publication date
WO2000061587A1 (fr) 2000-10-19
CA2369725C (fr) 2011-05-31
DE60003662T2 (de) 2004-06-09
PL350902A1 (en) 2003-02-10
ES2202091T3 (es) 2004-04-01
EP1171444B1 (fr) 2003-07-02
DK1171444T3 (da) 2003-10-27
HUP0200928A3 (en) 2004-07-28
PL207639B1 (pl) 2011-01-31
AR028818A1 (es) 2003-05-28
FR2791980B1 (fr) 2001-07-06
AU3825700A (en) 2000-11-14
US6777408B1 (en) 2004-08-17
JP2002541260A (ja) 2002-12-03
EP1171444A1 (fr) 2002-01-16
NO20014803L (no) 2001-10-04
ATE244246T1 (de) 2003-07-15
CZ302455B6 (cs) 2011-06-01
CZ20013572A3 (cs) 2002-05-15
MY120085A (en) 2005-08-30
CA2369725A1 (fr) 2000-10-19
RU2245883C2 (ru) 2005-02-10
JP4681737B2 (ja) 2011-05-11
DE60003662D1 (de) 2003-08-07
FR2791980A1 (fr) 2000-10-13
NO20014803D0 (no) 2001-10-03
TW513433B (en) 2002-12-11
HUP0200928A2 (hu) 2002-07-29

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