PL361003A1 - Ulepszony sposób wytwarzania rozpuszczalnych w wodzie związków azolowych - Google Patents

Ulepszony sposób wytwarzania rozpuszczalnych w wodzie związków azolowych

Info

Publication number
PL361003A1
PL361003A1 PL01361003A PL36100301A PL361003A1 PL 361003 A1 PL361003 A1 PL 361003A1 PL 01361003 A PL01361003 A PL 01361003A PL 36100301 A PL36100301 A PL 36100301A PL 361003 A1 PL361003 A1 PL 361003A1
Authority
PL
Poland
Prior art keywords
improved process
water soluble
azole compounds
soluble azole
triazole antifungal
Prior art date
Application number
PL01361003A
Other languages
English (en)
Inventor
Chung-Pin Chen
Timothy Paul Connolly
Laxima Reddy Kolla
John D. Matiskella
Richard H. Mueller
Yadagiri Rendri
Dejah T. Petsch
Original Assignee
Bristol-Myers Squibb Company
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bristol-Myers Squibb Company filed Critical Bristol-Myers Squibb Company
Publication of PL361003A1 publication Critical patent/PL361003A1/pl

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02Phosphorus compounds
    • C07F9/06Phosphorus compounds without P—C bonds
    • C07F9/08Esters of oxyacids of phosphorus
    • C07F9/09Esters of phosphoric acids
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02Phosphorus compounds
    • C07F9/547Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/6558Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing at least two different or differently substituted hetero rings neither condensed among themselves nor condensed with a common carbocyclic ring or ring system
    • C07F9/65583Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing at least two different or differently substituted hetero rings neither condensed among themselves nor condensed with a common carbocyclic ring or ring system each of the hetero rings containing nitrogen as ring hetero atom
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02Phosphorus compounds
    • C07F9/547Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/6515Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having three nitrogen atoms as the only ring hetero atoms
    • C07F9/6518Five-membered rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biochemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Preventing Corrosion Or Incrustation Of Metals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
PL01361003A 2000-11-20 2001-10-18 Ulepszony sposób wytwarzania rozpuszczalnych w wodzie związków azolowych PL361003A1 (pl)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US25200100P 2000-11-20 2000-11-20
PCT/US2001/032382 WO2002042283A1 (en) 2000-11-20 2001-10-18 Improved process for water soluble azole compounds

Publications (1)

Publication Number Publication Date
PL361003A1 true PL361003A1 (pl) 2004-09-20

Family

ID=22954236

Family Applications (1)

Application Number Title Priority Date Filing Date
PL01361003A PL361003A1 (pl) 2000-11-20 2001-10-18 Ulepszony sposób wytwarzania rozpuszczalnych w wodzie związków azolowych

Country Status (18)

Country Link
US (1) US6448401B1 (pl)
EP (1) EP1345915B1 (pl)
JP (1) JP4579496B2 (pl)
KR (1) KR100734456B1 (pl)
CN (1) CN1279033C (pl)
AT (1) ATE353079T1 (pl)
AU (2) AU2002213317B2 (pl)
BR (1) BR0115448A (pl)
CA (1) CA2429378C (pl)
CZ (1) CZ20031388A3 (pl)
DE (1) DE60126425T2 (pl)
ES (1) ES2280405T3 (pl)
HU (1) HUP0301917A3 (pl)
IL (2) IL155612A0 (pl)
MX (1) MXPA03004332A (pl)
NO (1) NO20032241D0 (pl)
PL (1) PL361003A1 (pl)
WO (1) WO2002042283A1 (pl)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6362172B2 (en) * 2000-01-20 2002-03-26 Bristol-Myers Squibb Company Water soluble prodrugs of azole compounds
TWI329105B (en) 2002-02-01 2010-08-21 Rigel Pharmaceuticals Inc 2,4-pyrimidinediamine compounds and their uses
PL1656372T3 (pl) 2003-07-30 2013-08-30 Rigel Pharmaceuticals Inc Związki 2,4-pirymidynodiaminy do stosowania w leczeniu lub zapobieganiu chorobom autoimmunologicznym
US20060047135A1 (en) * 2004-08-30 2006-03-02 Chadwick Scott T Process for preparing chloromethyl di-tert-butylphosphate
BRPI0606318B8 (pt) 2005-01-19 2021-05-25 Rigel Pharmaceuticals Inc composto, composição, e, uso de um composto
JO2691B1 (en) * 2005-05-03 2013-03-03 ايساي آر آند دي مانجمنت كو.، ليمتد Monolysine salts for azole compounds
JP4981673B2 (ja) * 2005-09-13 2012-07-25 エーザイ・アール・アンド・ディー・マネジメント株式会社 安定性が改善されたクロロメチルフォスフェイト誘導体を含む組成物およびその製造方法
EP1964843B1 (en) * 2005-12-20 2013-08-28 Eisai R&D Management Co., Ltd. Process for production of water-soluble azole prodrug
DE602007009489D1 (de) * 2006-02-22 2010-11-11 Eisai R&D Man Co Ltd Stabilisierte pharmazeutische zusammensetzung
WO2008108384A1 (ja) 2007-03-06 2008-09-12 Eisai R & D Management Co., Ltd. 安定性が改善されたクロロメチルフォスフェイト誘導体を含む組成物及びその製造方法
FI20070574A0 (fi) * 2007-07-30 2007-07-30 Kuopion Yliopisto Vesiliukoinen propofolin etylideenifosfaatti-aihiolääke
JP6336902B2 (ja) 2011-06-22 2018-06-06 ビョーメ バイオサイエンシズ ピーブイティー.リミテッド コンジュゲートベースの抗真菌性および抗菌性プロドラッグ
EP3525759A1 (en) * 2016-10-14 2019-08-21 Pulmatrix Operating Company, Inc. Antifungal dry powders

Family Cites Families (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2111527C (en) 1992-12-24 2000-07-18 Jerzy Golik Phosphonooxymethyl ethers of taxane derivatives
CA2129288C (en) 1993-08-17 2000-05-16 Jerzy Golik Phosphonooxymethyl esters of taxane derivatives
AU681753B2 (en) 1993-12-21 1997-09-04 Merck Sharp & Dohme Corp. Tetrahydrofuran antifungals
NZ278882A (en) 1994-01-24 1997-06-24 Janssen Pharmaceutica Nv Piperazine-containing azole antifungal compounds
NZ270418A (en) * 1994-02-07 1997-09-22 Eisai Co Ltd Polycyclic triazole & imidazole derivatives, antifungal compositions
ATE240319T1 (de) 1995-06-02 2003-05-15 Schering Corp Antifungale tetrahydrofurane
GB9602080D0 (en) * 1996-02-02 1996-04-03 Pfizer Ltd Pharmaceutical compounds
EP0829478A3 (en) 1996-09-09 1998-03-25 F. Hoffmann-La Roche Ag N-Benzylimidazolium and N-benzyltriazolium derivatives, their preparation and their use as antifungal and antimycotic agents
AU730592B2 (en) 1998-01-29 2001-03-08 Bristol-Myers Squibb Company Phosphate derivatives of diaryl 1,3,4-oxadiazolone
US5883097A (en) 1998-04-16 1999-03-16 Schering Corporation Soluble azole antifungal salt
US6265584B1 (en) 1998-05-22 2001-07-24 Bristol-Myers Squibb Company Water soluble prodrugs of azole compounds
US6204257B1 (en) * 1998-08-07 2001-03-20 Universtiy Of Kansas Water soluble prodrugs of hindered alcohols
AU1915500A (en) * 1998-11-20 2000-06-13 Bristol-Myers Squibb Company Water soluble prodrugs of azole compounds
US6362172B2 (en) * 2000-01-20 2002-03-26 Bristol-Myers Squibb Company Water soluble prodrugs of azole compounds

Also Published As

Publication number Publication date
US20020062028A1 (en) 2002-05-23
NO20032241D0 (no) 2003-05-19
CZ20031388A3 (cs) 2003-08-13
EP1345915A4 (en) 2005-08-03
CA2429378C (en) 2008-03-18
JP2004518640A (ja) 2004-06-24
ATE353079T1 (de) 2007-02-15
WO2002042283A1 (en) 2002-05-30
DE60126425T2 (de) 2007-10-18
CN1279033C (zh) 2006-10-11
MXPA03004332A (es) 2004-05-04
HUP0301917A3 (en) 2005-11-28
CN1474817A (zh) 2004-02-11
AU2002213317B2 (en) 2007-03-15
KR20040020865A (ko) 2004-03-09
HUP0301917A2 (hu) 2003-09-29
US6448401B1 (en) 2002-09-10
KR100734456B1 (ko) 2007-07-03
AU1331702A (en) 2002-06-03
IL155612A (en) 2010-05-31
EP1345915A1 (en) 2003-09-24
ES2280405T3 (es) 2007-09-16
BR0115448A (pt) 2004-02-17
EP1345915B1 (en) 2007-01-31
IL155612A0 (en) 2003-11-23
JP4579496B2 (ja) 2010-11-10
DE60126425D1 (de) 2007-03-22
CA2429378A1 (en) 2002-05-30

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Legal Events

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REFS Decisions on refusal to grant patents (taken after the publication of the particulars of the applications)