PL3222277T3 - Bifenylosulfonamid będący antagonistą receptora endoteliny i angiotensyny ii do leczenia stwardnienia kłębuszków nerkowych i nefropatii wywołanej iga - Google Patents

Bifenylosulfonamid będący antagonistą receptora endoteliny i angiotensyny ii do leczenia stwardnienia kłębuszków nerkowych i nefropatii wywołanej iga

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Publication number
PL3222277T3
PL3222277T3 PL17157697T PL17157697T PL3222277T3 PL 3222277 T3 PL3222277 T3 PL 3222277T3 PL 17157697 T PL17157697 T PL 17157697T PL 17157697 T PL17157697 T PL 17157697T PL 3222277 T3 PL3222277 T3 PL 3222277T3
Authority
PL
Poland
Prior art keywords
endotelin
angiotensin
iga
antagonist
receptor
Prior art date
Application number
PL17157697T
Other languages
English (en)
Inventor
Jinkun Zhang
Zofia E Dziewanowska
Rene Belder
Ian Henderson
Joseph B Bogardus
Zhaoying Zhang
Original Assignee
Ligand Pharmaceuticals Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=42828649&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=PL3222277(T3) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Ligand Pharmaceuticals Inc. filed Critical Ligand Pharmaceuticals Inc.
Publication of PL3222277T3 publication Critical patent/PL3222277T3/pl

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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42—Oxazoles
    • A61K31/422—Oxazoles not condensed and containing further heterocyclic rings
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    • A61K9/2013—Organic compounds, e.g. phospholipids, fats
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  • Hematology (AREA)
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  • Endocrinology (AREA)
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PL17157697T 2009-03-31 2010-03-29 Bifenylosulfonamid będący antagonistą receptora endoteliny i angiotensyny ii do leczenia stwardnienia kłębuszków nerkowych i nefropatii wywołanej iga PL3222277T3 (pl)

Applications Claiming Priority (6)

Application Number Priority Date Filing Date Title
US16541909P 2009-03-31 2009-03-31
US16544709P 2009-03-31 2009-03-31
PCT/US2010/029093 WO2010114801A1 (en) 2009-03-31 2010-03-29 Oral formulations of diphenylsulfonamide endothelin and angiotensin ii receptor agonists to treat elevated blood pressure and diabetic nephropathy
EP17157697.8A EP3222277B1 (en) 2009-03-31 2010-03-29 A biphenylsulfonamide endothelin and angiotensin ii receptor antagonist to treat glomerulosclerosis and iga-induced nephropathy
EP10759268A EP2413930A4 (en) 2009-03-31 2010-03-29 ORAL FORMULATION OF ENDOTHELIN AND ANGIOTENSIN II RECEPTOR AGONISTS BASED ON DIPHENYLSULFONAMIDE TO TREAT HIGH BLOOD PRESSURE AND DIABETIC NEPHROPATHY
EP14155459.2A EP2732818B1 (en) 2009-03-31 2010-03-29 A biphenylsulfonamide endothelin and angiotensin ii receptor antagonist to treat glomerulosclerosis

Publications (1)

Publication Number Publication Date
PL3222277T3 true PL3222277T3 (pl) 2020-08-24

Family

ID=42828649

Family Applications (2)

Application Number Title Priority Date Filing Date
PL14155459T PL2732818T3 (pl) 2009-03-31 2010-03-29 Bifenylosulfonamidowy antagonista receptora endoteliny i angiotensyny II do leczenia stwardnienia kłębków nerkowych
PL17157697T PL3222277T3 (pl) 2009-03-31 2010-03-29 Bifenylosulfonamid będący antagonistą receptora endoteliny i angiotensyny ii do leczenia stwardnienia kłębuszków nerkowych i nefropatii wywołanej iga

Family Applications Before (1)

Application Number Title Priority Date Filing Date
PL14155459T PL2732818T3 (pl) 2009-03-31 2010-03-29 Bifenylosulfonamidowy antagonista receptora endoteliny i angiotensyny II do leczenia stwardnienia kłębków nerkowych

Country Status (18)

Country Link
US (4) US20140142149A1 (pl)
EP (4) EP3708163A1 (pl)
JP (3) JP2012522058A (pl)
CN (2) CN102421434A (pl)
CY (3) CY1119232T1 (pl)
DK (2) DK2732818T3 (pl)
ES (2) ES2811342T3 (pl)
FI (1) FIC20240031I1 (pl)
FR (1) FR24C1038I2 (pl)
HR (2) HRP20171197T1 (pl)
HU (3) HUE049450T2 (pl)
LT (3) LT2732818T (pl)
NL (1) NL301291I2 (pl)
PL (2) PL2732818T3 (pl)
PT (2) PT2732818T (pl)
SI (2) SI3222277T1 (pl)
SM (2) SMT201700416T1 (pl)
WO (1) WO2010114801A1 (pl)

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US20130022551A1 (en) * 2011-07-22 2013-01-24 Trustees Of Boston University DEspR ANTAGONISTS AND AGONISTS AS THERAPEUTICS
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JP6491669B2 (ja) 2014-02-05 2019-03-27 メルク・シャープ・アンド・ドーム・コーポレーションＭｅｒｃｋ Ｓｈａｒｐ ＆ Ｄｏｈｍｅ Ｃｏｒｐ． Ｃｇｒｐ活性化合物の錠剤製剤
CN114181195A (zh) 2014-02-07 2022-03-15 全球血液疗法股份有限公司 一种化合物的结晶多晶型物
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