PL2997021T3 - Nowi agoniści receptora somatostatyny podtypu 4 (SSTR4) - Google Patents

Nowi agoniści receptora somatostatyny podtypu 4 (SSTR4)

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Publication number
PL2997021T3
PL2997021T3 PL14724085T PL14724085T PL2997021T3 PL 2997021 T3 PL2997021 T3 PL 2997021T3 PL 14724085 T PL14724085 T PL 14724085T PL 14724085 T PL14724085 T PL 14724085T PL 2997021 T3 PL2997021 T3 PL 2997021T3
Authority
PL
Poland
Prior art keywords
sstr4
agonists
receptor subtype
somatostatin receptor
new somatostatin
Prior art date
Application number
PL14724085T
Other languages
English (en)
Polish (pl)
Inventor
Riccardo Giovannini
Yunhai Cui
Henri Doods
Marco Ferrara
Stefan Just
Raimund Kuelzer
Iain Lingard
Rocco Mazzaferro
Klaus Rudolf
Original Assignee
Centrexion Therapeutics Corporation
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Centrexion Therapeutics Corporation filed Critical Centrexion Therapeutics Corporation
Publication of PL2997021T3 publication Critical patent/PL2997021T3/pl

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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/403—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/415—1,2-Diazoles
    • A61K31/4155—1,2-Diazoles non condensed and containing further heterocyclic rings
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    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/415—1,2-Diazoles
    • A61K31/416—1,2-Diazoles condensed with carbocyclic ring systems, e.g. indazole
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    • A61K31/423—Oxazoles condensed with carbocyclic rings
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    • A61K31/437—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
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    • A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
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    • A61K31/4965—Non-condensed pyrazines
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    • A61K31/50—Pyridazines; Hydrogenated pyridazines
    • A61K31/501—Pyridazines; Hydrogenated pyridazines not condensed and containing further heterocyclic rings
    • A—HUMAN NECESSITIES
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    • C07D—HETEROCYCLIC COMPOUNDS
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    • C07D—HETEROCYCLIC COMPOUNDS
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    • C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • C07D487/04—Ortho-condensed systems

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  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
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  • Diabetes (AREA)
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  • Hematology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Peptides Or Proteins (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Indole Compounds (AREA)
PL14724085T 2013-05-17 2014-05-15 Nowi agoniści receptora somatostatyny podtypu 4 (SSTR4) PL2997021T3 (pl)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP13168224 2013-05-17
EP14724085.7A EP2997021B1 (en) 2013-05-17 2014-05-15 New somatostatin receptor subtype 4 (sstr4) agonists
PCT/EP2014/059905 WO2014184275A1 (en) 2013-05-17 2014-05-15 New somatostatin receptor subtype 4 (sstr4) agonists

Publications (1)

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PL2997021T3 true PL2997021T3 (pl) 2018-05-30

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PL14724085T PL2997021T3 (pl) 2013-05-17 2014-05-15 Nowi agoniści receptora somatostatyny podtypu 4 (SSTR4)

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BR112015028452B1 (pt) 2023-04-11

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