PL2800565T3 - Związki karbaminianowe i sposoby ich wytwarzania oraz zastosowanie - Google Patents

Związki karbaminianowe i sposoby ich wytwarzania oraz zastosowanie

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Publication number
PL2800565T3
PL2800565T3 PL13733636T PL13733636T PL2800565T3 PL 2800565 T3 PL2800565 T3 PL 2800565T3 PL 13733636 T PL13733636 T PL 13733636T PL 13733636 T PL13733636 T PL 13733636T PL 2800565 T3 PL2800565 T3 PL 2800565T3
Authority
PL
Poland
Prior art keywords
making
methods
same
carbamate compounds
carbamate
Prior art date
Application number
PL13733636T
Other languages
English (en)
Inventor
Justin S. Cisar
Cheryl A. Grice
Todd K. Jones
Micah J. Niphakis
Jae Won Chang
Kenneth M. Lum
Benjamin F. Cravatt
Original Assignee
Lundbeck La Jolla Research Center, Inc.
The Scripps Research Institute
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lundbeck La Jolla Research Center, Inc., The Scripps Research Institute filed Critical Lundbeck La Jolla Research Center, Inc.
Publication of PL2800565T3 publication Critical patent/PL2800565T3/pl

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    • C07D295/16—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms
    • C07D295/20—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms by radicals derived from carbonic acid, or sulfur or nitrogen analogues thereof
    • C07D295/205—Radicals derived from carbonic acid
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    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
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    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
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    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
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