PL116228B1 - Process for preparing novel derivatives of 4"-desoxyaminoerythromycin a" - Google Patents

Process for preparing novel derivatives of 4"-desoxyaminoerythromycin a" Download PDF

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Publication number
PL116228B1
PL116228B1 PL1978204428A PL20442878A PL116228B1 PL 116228 B1 PL116228 B1 PL 116228B1 PL 1978204428 A PL1978204428 A PL 1978204428A PL 20442878 A PL20442878 A PL 20442878A PL 116228 B1 PL116228 B1 PL 116228B1
Authority
PL
Poland
Prior art keywords
deoxy
aminoerythromycin
product
formula
compounds
Prior art date
Application number
PL1978204428A
Other languages
English (en)
Polish (pl)
Other versions
PL204428A1 (pl
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US05/856,479 external-priority patent/US4150220A/en
Application filed by Pfizer filed Critical Pfizer
Publication of PL204428A1 publication Critical patent/PL204428A1/xx
Publication of PL116228B1 publication Critical patent/PL116228B1/pl

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08Hetero rings containing eight or more ring members, e.g. erythromycins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Communicable Diseases (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
PL1978204428A 1977-02-04 1978-02-03 Process for preparing novel derivatives of 4"-desoxyaminoerythromycin a" PL116228B1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US76548077A 1977-02-04 1977-02-04
US05/856,479 US4150220A (en) 1977-02-04 1977-12-01 Semi-synthetic 4"-erythromycin A derivatives

Publications (2)

Publication Number Publication Date
PL204428A1 PL204428A1 (pl) 1979-06-04
PL116228B1 true PL116228B1 (en) 1981-05-30

Family

ID=27117613

Family Applications (1)

Application Number Title Priority Date Filing Date
PL1978204428A PL116228B1 (en) 1977-02-04 1978-02-03 Process for preparing novel derivatives of 4"-desoxyaminoerythromycin a"

Country Status (30)

Country Link
JP (1) JPS5827798B2 (cs)
AR (1) AR222147A1 (cs)
AU (1) AU501298B1 (cs)
BG (2) BG32718A3 (cs)
CA (1) CA1106367A (cs)
CH (1) CH628906A5 (cs)
CS (1) CS221801B2 (cs)
DD (1) DD140048A5 (cs)
DE (1) DE2804507C2 (cs)
DK (1) DK148036C (cs)
ES (2) ES466057A1 (cs)
FI (1) FI780354A7 (cs)
FR (2) FR2379550A1 (cs)
GB (2) GB1585315A (cs)
GR (1) GR68691B (cs)
HU (1) HU182559B (cs)
IE (1) IE46661B1 (cs)
IL (2) IL53968A0 (cs)
IT (1) IT1094209B (cs)
LU (1) LU79004A1 (cs)
NL (1) NL176174C (cs)
NO (2) NO146472C (cs)
NZ (1) NZ186385A (cs)
PH (2) PH14421A (cs)
PL (1) PL116228B1 (cs)
PT (1) PT67568B (cs)
RO (4) RO79686A7 (cs)
SE (2) SE445223B (cs)
SU (1) SU927122A3 (cs)
YU (3) YU40913B (cs)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4133950A (en) * 1978-01-03 1979-01-09 Pfizer Inc. 4"-Deoxy-4"-carbamate and dithiocarbamate derivatives of oleandomycin and its esters
US4124755A (en) * 1978-01-03 1978-11-07 Pfizer Inc. 11-Alkanoyl-4"-deoxy-4"-isonitrilo-oleandomycin derivatives
US4382085A (en) * 1982-03-01 1983-05-03 Pfizer Inc. 4"-Epi erythromycin A and derivatives thereof as useful antibacterial agents
US4518590A (en) * 1984-04-13 1985-05-21 Pfizer Inc. 9α-Aza-9α-homoerythromycin compounds, pharmaceutical compositions and therapeutic method
HN1998000074A (es) * 1997-06-11 1999-01-08 Pfizer Prod Inc Derivados de macrolidos c-4 sustituidos
US6407074B1 (en) 1997-06-11 2002-06-18 Pfizer Inc C-4″-substituted macrolide derivatives

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3836519A (en) * 1973-05-04 1974-09-17 Abbott Lab Sulfonyl derivatives of erythromycin
US3884903A (en) * 1973-06-21 1975-05-20 Abbott Lab 4{41 -Deoxy-4{41 -oxoerythromycin B derivatives

Also Published As

Publication number Publication date
PH16675A (en) 1983-12-13
CA1106367A (en) 1981-08-04
DE2804507A1 (de) 1978-08-10
IL53968A0 (en) 1978-04-30
YU40799B (en) 1986-06-30
IE780239L (en) 1978-08-04
FR2379550A1 (fr) 1978-09-01
IE46661B1 (en) 1983-08-24
IT1094209B (it) 1985-07-26
BG32718A3 (bg) 1982-09-15
RO81622A (ro) 1983-04-29
RO79686A7 (ro) 1982-08-17
YU40798B (en) 1986-06-30
PT67568B (en) 1979-06-18
CH628906A5 (en) 1982-03-31
JPS53101337A (en) 1978-09-04
IL61997A0 (en) 1981-02-27
NZ186385A (en) 1980-10-08
GR68691B (cs) 1982-02-01
FR2379550B1 (cs) 1980-07-04
YU227983A (en) 1984-04-30
YU7378A (en) 1983-04-30
IT7820005A0 (it) 1978-02-03
NL7801262A (nl) 1978-08-08
DD140048A5 (de) 1980-02-06
NO780389L (no) 1978-08-07
NO811913L (no) 1978-08-07
FR2385735B1 (cs) 1980-10-24
ES472429A1 (es) 1979-04-01
CS221801B2 (en) 1983-04-29
SE8300870D0 (sv) 1983-02-16
RO79687A7 (ro) 1982-08-17
YU26583A (en) 1984-02-29
FR2385735A1 (fr) 1978-10-27
SU927122A3 (ru) 1982-05-07
JPS5827798B2 (ja) 1983-06-11
NL176174B (nl) 1984-10-01
NO150484B (no) 1984-07-16
RO77345A (ro) 1981-08-17
BG33159A3 (bg) 1982-12-15
DK51878A (da) 1978-08-05
NO146472B (no) 1982-06-28
AU501298B1 (en) 1979-06-14
SE457086B (sv) 1988-11-28
PT67568A (en) 1978-02-01
PH14421A (en) 1981-07-10
GB1585315A (en) 1981-02-25
DK148036B (da) 1985-02-11
HU182559B (en) 1984-02-28
NL176174C (nl) 1985-03-01
SE445223B (sv) 1986-06-09
NO150484C (no) 1984-10-24
PL204428A1 (pl) 1979-06-04
DK148036C (da) 1985-07-15
SE7800270L (sv) 1978-08-05
NO146472C (no) 1982-10-06
LU79004A1 (fr) 1979-09-06
AR222147A1 (es) 1981-04-30
RO81622B (ro) 1983-04-30
SE8300870L (sv) 1983-02-16
ES466057A1 (es) 1978-10-01
FI780354A7 (fi) 1978-08-05
DE2804507C2 (de) 1982-11-04
YU40913B (en) 1986-08-31
GB1585316A (en) 1981-02-25

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