PL115756B1 - Process for preparing novel 1,1-dioxid-4-hydroxy-2h-1,2-benzothiazin-3-carboxyamides - Google Patents

Process for preparing novel 1,1-dioxid-4-hydroxy-2h-1,2-benzothiazin-3-carboxyamides Download PDF

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Publication number
PL115756B1
PL115756B1 PL1978211753A PL21175378A PL115756B1 PL 115756 B1 PL115756 B1 PL 115756B1 PL 1978211753 A PL1978211753 A PL 1978211753A PL 21175378 A PL21175378 A PL 21175378A PL 115756 B1 PL115756 B1 PL 115756B1
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PL
Poland
Prior art keywords
methyl
hydroxy
benzothiazine
dioxide
group
Prior art date
Application number
PL1978211753A
Other languages
English (en)
Polish (pl)
Other versions
PL211753A1 (pl
Original Assignee
Thomae Gmbh Dr K
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Thomae Gmbh Dr K filed Critical Thomae Gmbh Dr K
Publication of PL211753A1 publication Critical patent/PL211753A1/xx
Publication of PL115756B1 publication Critical patent/PL115756B1/pl

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D275/00—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings
    • C07D275/04—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings condensed with carbocyclic rings or ring systems
    • C07D275/06—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings condensed with carbocyclic rings or ring systems with hetero atoms directly attached to the ring sulfur atom
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D279/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one sulfur atom as the only ring hetero atoms
    • C07D279/02—1,2-Thiazines; Hydrogenated 1,2-thiazines
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains three hetero rings
    • C07D513/14—Ortho-condensed systems

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Rheumatology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Pain & Pain Management (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
PL1978211753A 1977-12-16 1978-12-14 Process for preparing novel 1,1-dioxid-4-hydroxy-2h-1,2-benzothiazin-3-carboxyamides PL115756B1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19772756113 DE2756113A1 (de) 1977-12-16 1977-12-16 Neue 4-hydroxy-2h-1,2-benzothiazin- 3-carboxamid-1,1-dioxide, verfahren zu ihrer herstellung und diese enthaltende arzneimittel

Publications (2)

Publication Number Publication Date
PL211753A1 PL211753A1 (pl) 1979-08-13
PL115756B1 true PL115756B1 (en) 1981-04-30

Family

ID=6026297

Family Applications (1)

Application Number Title Priority Date Filing Date
PL1978211753A PL115756B1 (en) 1977-12-16 1978-12-14 Process for preparing novel 1,1-dioxid-4-hydroxy-2h-1,2-benzothiazin-3-carboxyamides

Country Status (27)

Country Link
US (1) US4233299A (OSRAM)
EP (1) EP0002482B1 (OSRAM)
JP (1) JPS5492976A (OSRAM)
AT (1) AT365589B (OSRAM)
AU (1) AU522538B2 (OSRAM)
BG (2) BG33286A3 (OSRAM)
CA (1) CA1102802A (OSRAM)
CS (2) CS202515B2 (OSRAM)
DD (1) DD140354A5 (OSRAM)
DE (2) DE2756113A1 (OSRAM)
DK (1) DK149344C (OSRAM)
ES (2) ES475677A1 (OSRAM)
FI (1) FI61896C (OSRAM)
GR (1) GR65626B (OSRAM)
HU (1) HU175846B (OSRAM)
IE (1) IE48042B1 (OSRAM)
IL (1) IL56206A (OSRAM)
LU (1) LU88557I2 (OSRAM)
MX (1) MX9202949A (OSRAM)
NL (1) NL940002I2 (OSRAM)
NO (2) NO150203C (OSRAM)
NZ (1) NZ189186A (OSRAM)
PL (1) PL115756B1 (OSRAM)
PT (1) PT68915A (OSRAM)
RO (1) RO75792A (OSRAM)
SU (1) SU841588A3 (OSRAM)
YU (1) YU294978A (OSRAM)

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US3892740A (en) * 1974-10-15 1975-07-01 Pfizer Process for the production of carboxamides of oxo-1,2-benzothiazine-1,1-dioxides
US4074048A (en) * 1976-05-10 1978-02-14 Warner-Lambert Company Process for the preparation of 4-hydroxy-2H-1,2-benzothiazine-3-carboxamide 1,1-dioxides
US4100347A (en) * 1976-06-10 1978-07-11 Pfizer Inc. 3,4-Dihydro-2-methyl-4-oxo-2H-1,2-benzothiazine-3-carboxylic acid-1,1-dioxide

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SU841588A3 (ru) 1981-06-23
ATA863078A (de) 1981-06-15
IL56206A (en) 1982-04-30
PT68915A (de) 1979-01-01
RO75792A (ro) 1981-02-28
EP0002482B1 (de) 1981-01-07
AU522538B2 (en) 1982-06-10
NO150203C (no) 1984-09-05
BG60475B2 (bg) 1995-04-28
PL211753A1 (pl) 1979-08-13
LU88557I2 (fr) 1995-03-21
DE2756113A1 (de) 1979-06-21
FI61896B (fi) 1982-06-30
FI61896C (fi) 1982-10-11
EP0002482A1 (de) 1979-06-27
YU294978A (en) 1982-10-31
AU4253078A (en) 1979-06-21
CS410091A3 (en) 1992-06-17
ES475677A1 (es) 1979-04-16
FI783867A7 (fi) 1979-06-17
IE782482L (en) 1979-06-16
GR65626B (en) 1980-10-15
DK562078A (da) 1979-06-17
CS202515B2 (en) 1981-01-30
NO784231L (no) 1979-06-19
ES8802454A3 (es) 1988-06-16
JPS6324997B2 (OSRAM) 1988-05-23
CA1102802A (en) 1981-06-09
NL940002I2 (nl) 1997-05-01
DK149344B (da) 1986-05-12
NL940002I1 (nl) 1994-03-16
IL56206A0 (en) 1979-03-12
DK149344C (da) 1986-10-13
ES550377A0 (es) 1988-06-16
HU175846B (hu) 1980-10-28
NO1997002I1 (no) 1997-01-14
JPS5492976A (en) 1979-07-23
NO150203B (no) 1984-05-28
IE48042B1 (en) 1984-09-05
NZ189186A (en) 1981-03-16
BG33286A3 (bg) 1983-01-14
DD140354A5 (de) 1980-02-27
AT365589B (de) 1982-01-25
US4233299A (en) 1980-11-11
MX9202949A (es) 1992-07-01
DE2860445D1 (en) 1981-02-26

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