PH31291A - Process for the preparation of chlorosulfate and sulfate derivatives of 2,3,4,5-bis-o-(1-methylidene)-b-d-fructopyranose and 91-cyclohexyl methanol. - Google Patents
Process for the preparation of chlorosulfate and sulfate derivatives of 2,3,4,5-bis-o-(1-methylidene)-b-d-fructopyranose and 91-cyclohexyl methanol.Info
- Publication number
- PH31291A PH31291A PH44955A PH44955A PH31291A PH 31291 A PH31291 A PH 31291A PH 44955 A PH44955 A PH 44955A PH 44955 A PH44955 A PH 44955A PH 31291 A PH31291 A PH 31291A
- Authority
- PH
- Philippines
- Prior art keywords
- chlorosulfate
- fructopyranose
- bis
- methylidene
- preparation
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D493/00—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system
- C07D493/02—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system in which the condensed system contains two hetero rings
- C07D493/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C303/00—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides
- C07C303/34—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides of amides of sulfuric acids
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D309/00—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings
- C07D309/02—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
- C07D309/04—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having no double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
- C07D309/06—Radicals substituted by oxygen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D493/00—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system
- C07D493/12—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system in which the condensed system contains three hetero rings
- C07D493/14—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H9/00—Compounds containing a hetero ring sharing at least two hetero atoms with a saccharide radical
- C07H9/02—Compounds containing a hetero ring sharing at least two hetero atoms with a saccharide radical the hetero ring containing only oxygen as ring hetero atoms
- C07H9/04—Cyclic acetals
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Health & Medical Sciences (AREA)
- Biochemistry (AREA)
- Biotechnology (AREA)
- General Health & Medical Sciences (AREA)
- Genetics & Genomics (AREA)
- Molecular Biology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Saccharide Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US76272091A | 1991-09-19 | 1991-09-19 | |
US92626992A | 1992-08-05 | 1992-08-05 |
Publications (1)
Publication Number | Publication Date |
---|---|
PH31291A true PH31291A (en) | 1998-07-06 |
Family
ID=27117178
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
PH44955A PH31291A (en) | 1991-09-19 | 1992-09-18 | Process for the preparation of chlorosulfate and sulfate derivatives of 2,3,4,5-bis-o-(1-methylidene)-b-d-fructopyranose and 91-cyclohexyl methanol. |
Country Status (23)
Country | Link |
---|---|
US (1) | US5387700A (fi) |
EP (1) | EP0533483B1 (fi) |
JP (1) | JP3174410B2 (fi) |
KR (1) | KR100229180B1 (fi) |
CN (1) | CN1035820C (fi) |
AT (1) | ATE163937T1 (fi) |
AU (1) | AU651244B2 (fi) |
CA (1) | CA2078519C (fi) |
DE (1) | DE69224691T2 (fi) |
DK (1) | DK0533483T3 (fi) |
EG (1) | EG20164A (fi) |
ES (1) | ES2114917T3 (fi) |
FI (1) | FI107731B (fi) |
GR (1) | GR3026618T3 (fi) |
HU (1) | HU212634B (fi) |
IL (1) | IL103172A (fi) |
MX (1) | MX9205305A (fi) |
MY (1) | MY113564A (fi) |
NO (1) | NO179284C (fi) |
NZ (1) | NZ244409A (fi) |
PH (1) | PH31291A (fi) |
TW (1) | TW217413B (fi) |
ZW (1) | ZW14792A1 (fi) |
Families Citing this family (64)
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JP3250777B2 (ja) * | 1995-02-13 | 2002-01-28 | セントラル硝子株式会社 | イミド類、その塩類およびそれらの製造法 |
UA65607C2 (uk) * | 1998-03-04 | 2004-04-15 | Орто-Макнейл Фармацевтикал, Інк. | Фармацевтична композиція (варіанти) та спосіб її приготування |
EP1158950B1 (en) * | 1999-02-17 | 2006-01-25 | Ortho-Mcneil Pharmaceutical, Inc. | Anticonvulsant derivatives useful in treating essential tremor |
US6420369B1 (en) | 1999-05-24 | 2002-07-16 | Ortho-Mcneil Pharmaceutical, Inc. | Anticonvulsant derivatives useful in treating dementia |
BR0112519A (pt) * | 2000-07-07 | 2004-03-30 | Ortho Mcneil Pharm Inc | Derivados anticonvulsivantes úteis para prevenir o desenvolvimento de diabetes melito do tipo ii e sìndrome x |
EP1309325A1 (en) | 2000-08-02 | 2003-05-14 | Ortho-McNeil Pharmaceutical, Inc. | Anticonvulsant derivatives useful for the treatment of depression |
ATE334718T1 (de) * | 2000-10-30 | 2006-08-15 | Ortho Mcneil Pharm Inc | Kombinationstherapie mit antidiabetischen und antikonvulsiven mitteln |
US7041650B2 (en) * | 2001-07-09 | 2006-05-09 | Ortho-Mcneil Pharmaceutical, Inc. | Anticonvulsant derivative salts |
UA78211C2 (en) * | 2001-07-09 | 2007-03-15 | Ortho Mcneil Pharm Inc | Salts of fructopyranose derivatives as anticonvulsant |
JP2005508373A (ja) * | 2001-11-06 | 2005-03-31 | オーソ−マクニール・フアーマシユーチカル・インコーポレーテツド | 抗痙攣剤誘導体およびカリウムを用いる共同療法を含んでなる感覚異常の処置および予防 |
US20030224006A1 (en) | 2002-03-01 | 2003-12-04 | Zaworotko Michael J. | Multiple-component solid phases containing at least one active pharmaceutical ingredient |
US20030225002A1 (en) * | 2002-02-26 | 2003-12-04 | Livingstone Ian R. | Co-therapy for the treatment of migraine comprising anticonvulsant derivatives and anti-migraine agents |
US7060725B2 (en) | 2002-05-13 | 2006-06-13 | Janssen Pharmaceutica N.V. | Substituted sulfamate anticonvulsant derivatives |
AR039744A1 (es) * | 2002-06-26 | 2005-03-09 | Alza Corp | Metodos y formas de dosificacion para aumentar la solubilidad de las composiciones de farmacos para la administracion controlada |
MXPA05001184A (es) * | 2002-07-29 | 2005-09-12 | Johnson & Johnson | Formulaciones y formas de dosificacion para administracion controlada de topiramato. |
US7196209B2 (en) * | 2002-10-31 | 2007-03-27 | Ortho-Mcneil Pharmaceutical, Inc. | Continuous process for the preparation of fructopyranose sulfamate derivatives |
CN100430408C (zh) * | 2002-10-31 | 2008-11-05 | 奥索-麦克尼尔药品公司 | 制备吡喃果糖氨基磺酸酯衍生物的连续法 |
UA81657C2 (ru) * | 2003-03-04 | 2008-01-25 | Орто-Макнейл Фармасьютикел, Инк. | Способ получения противосудорожных производных топирамата |
WO2004108732A1 (en) * | 2003-05-12 | 2004-12-16 | Sun Pharmaceutical Industries Limited | PROCESS FOR THE PREPARATION OF 2,3:4,5-BIS-O(1-METHYLETHYLIDENE)-ß-D-FRUCTOPYRANOSE SULFAMATE |
AU2004264316A1 (en) * | 2003-08-06 | 2005-02-24 | Alza Corporation | Uniform delivery of topiramate over prolonged period of time with enhanced dispersion formulation |
AU2004268549A1 (en) * | 2003-08-22 | 2005-03-10 | Alza Corporation | Stepwise delivery of topiramate over prolonged period of time |
AU2004268661A1 (en) * | 2003-09-02 | 2005-03-10 | Alza Corporation | Novel drug compositions and dosage forms of topiramate |
TW200528144A (en) * | 2003-11-14 | 2005-09-01 | Alza Corp | Controlled release of topiramate in liquid dosage forms |
KR20050062976A (ko) * | 2003-12-19 | 2005-06-28 | 일동제약주식회사 | 2,3:4,5-비스-오-(1-메틸에틸리덴)-베타-디-프럭토피라노즈설파메이트의 새로운 개량된 제조방법 |
US20050175696A1 (en) * | 2003-12-29 | 2005-08-11 | David Edgren | Drug granule coatings that impart smear resistance during mechanical compression |
CA2550699A1 (en) * | 2003-12-29 | 2005-07-21 | Alza Corporation, Inc. | Novel drug compositions and dosage forms of topiramate |
JP2007517061A (ja) * | 2003-12-29 | 2007-06-28 | アルザ・コーポレーシヨン | 新規薬剤組成物及び投与形態物 |
US20050203287A1 (en) * | 2004-03-11 | 2005-09-15 | Chandrasekhar Batchu | Process for the preparation of sulfamate derivatives |
AR049646A1 (es) * | 2004-06-16 | 2006-08-23 | Janssen Pharmaceutica Nv | Derivados de sulfamato y sulfamida utiles para el tratamiento de la epilepsia y trastornos relacionados |
MY147767A (en) * | 2004-06-16 | 2013-01-31 | Janssen Pharmaceutica Nv | Novel sulfamate and sulfamide derivatives useful for the treatment of epilepsy and related disorders |
AU2005277134A1 (en) * | 2004-08-24 | 2006-03-02 | Janssen Pharmaceutica N.V. | Novel benzo-fused heteroaryl sulfamide derivatives useful as anticonvulsant agents |
WO2006041718A2 (en) * | 2004-10-05 | 2006-04-20 | Fallbrook Technologies, Inc. | Continuously variable transmission |
EA200702558A1 (ru) * | 2005-05-20 | 2008-06-30 | Янссен Фармацевтика Н. В. | Способ получения производных сульфамида |
CN101257889A (zh) * | 2005-05-25 | 2008-09-03 | 詹森药业有限公司 | 托吡酯的儿科制剂 |
US8937096B2 (en) * | 2005-12-19 | 2015-01-20 | Janssen Pharmaceutica Nv | Use of benzo-fused heterocyle sulfamide derivatives for the treatment of mania and bipolar disorder |
US8497298B2 (en) * | 2005-12-19 | 2013-07-30 | Janssen Pharmaceutica Nv | Use of benzo-fused heterocycle sulfamide derivatives for lowering lipids and lowering blood glucose levels |
US8716231B2 (en) * | 2005-12-19 | 2014-05-06 | Janssen Pharmaceutica Nv | Use of benzo-fused heterocycle sulfamide derivatives for the treatment of pain |
US8492431B2 (en) * | 2005-12-19 | 2013-07-23 | Janssen Pharmaceutica, N.V. | Use of benzo-fused heterocycle sulfamide derivatives for the treatment of obesity |
US20070155823A1 (en) * | 2005-12-19 | 2007-07-05 | Smith-Swintosky Virginia L | Use of benzo-fused heterocycle sulfamide derivatives as neuroprotective agents |
US8691867B2 (en) * | 2005-12-19 | 2014-04-08 | Janssen Pharmaceutica Nv | Use of benzo-fused heterocycle sulfamide derivatives for the treatment of substance abuse and addiction |
US20070155827A1 (en) * | 2005-12-19 | 2007-07-05 | Smith-Swintosky Virginia L | Use of benzo-fused heterocycle sulfamide derivatives for the treatment of depression |
US20070191461A1 (en) * | 2006-02-15 | 2007-08-16 | Smith-Swintosky Virginia L | Use of benzo-heteroaryl sulfamide derivatives for the treatment of migraine |
US20070191453A1 (en) * | 2006-02-15 | 2007-08-16 | Smith-Swintosky Virginia L | Use of benzo-heteroaryl sulfamide derivatives for the treatment of substance abuse and addiction |
US20070191459A1 (en) * | 2006-02-15 | 2007-08-16 | Smith-Swintosky Virginia L | Use of Benzo-Heteroaryl Sulfamide Derivatives for Lowering Lipids and Lowering Blood Glucose Levels |
US20070191449A1 (en) * | 2006-02-15 | 2007-08-16 | Smith-Swintosky Virginia L | Use of Benzo-Heteroaryl Sulfamide Derivatives for the Treatment of Depression |
US20070191474A1 (en) * | 2006-02-15 | 2007-08-16 | Smith-Swintosky Virginia L | Use of benzo-fused heterocyle sulfamide derivatives for the treatment of migraine |
WO2007099388A1 (en) * | 2006-03-01 | 2007-09-07 | Glade Organics Private Limited | An improved process for the manufacture of topiramate |
WO2007108009A1 (en) * | 2006-03-17 | 2007-09-27 | Alembic Limited | A process for purification of topiramate |
AU2007253814A1 (en) * | 2006-05-19 | 2007-11-29 | Janssen Pharmaceutica N.V. | Co-therapy for the treatment of epilepsy |
JP5424571B2 (ja) * | 2007-04-12 | 2014-02-26 | 協和発酵キリン株式会社 | トピラマート含有固形製剤 |
EP2573424A3 (en) * | 2007-04-24 | 2017-07-26 | Fallbrook Intellectual Property Company LLC | Electric traction drives |
CN101450951B (zh) * | 2007-11-30 | 2012-10-10 | 重庆凯林制药有限公司 | 托吡酯的制备方法 |
US20090247617A1 (en) * | 2008-03-26 | 2009-10-01 | Abdel-Magid Ahmed F | Process for the preparation of benzo-fused heteroaryl sulfamates |
US20090247616A1 (en) * | 2008-03-26 | 2009-10-01 | Smith-Swintosky Virginia L | Use of benzo-fused heterocyle sulfamide derivatives for the treatment of anxiety |
EA018567B1 (ru) | 2008-06-23 | 2013-08-30 | Янссен Фармацевтика Нв | Кристаллическая форма (2s)-(-)-n-(6-хлор-2,3-дигидробензо[1,4]диоксин-2-илметил)сульфамида |
US8815939B2 (en) * | 2008-07-22 | 2014-08-26 | Janssen Pharmaceutica Nv | Substituted sulfamide derivatives |
EP2367836B8 (en) * | 2010-02-05 | 2015-09-02 | Scinopharm Taiwan Ltd. | Process for the preparation and purification of topiramate |
CN102936268A (zh) * | 2012-11-13 | 2013-02-20 | 江苏吉贝尔药业有限公司 | 一种托吡酯中间体丙酮叉的制备方法 |
CN106397502A (zh) * | 2016-08-31 | 2017-02-15 | 安徽省润生医药股份有限公司 | 一种托吡酯的合成工艺 |
CN108341844A (zh) * | 2018-04-25 | 2018-07-31 | 广州小桔生物科技有限公司 | 一种高纯度托吡酯的制备方法 |
CN110655542A (zh) * | 2018-06-29 | 2020-01-07 | 鲁南制药集团股份有限公司 | 一种2,3:4,5-双-O-(1-甲基亚乙基)-β-D-吡喃果糖氯磺酸酯的晶型 |
CN110655541A (zh) * | 2018-06-29 | 2020-01-07 | 鲁南制药集团股份有限公司 | 一种2,3:4,5-双-O-(1-甲基亚乙基)-β-D-吡喃果糖氯磺酸酯晶型 |
WO2020104837A1 (en) | 2018-11-21 | 2020-05-28 | Rosemont Pharmaceuticals Limited | Oral topiramate suspension formulations with extended shelf stability and enhanced bioavailability |
CN114350340B (zh) * | 2022-01-13 | 2023-01-17 | 陕西科技大学 | 一种压裂用增渗剂及其制备方法和应用 |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4513006A (en) * | 1983-09-26 | 1985-04-23 | Mcneil Lab., Inc. | Anticonvulsant sulfamate derivatives |
US4582916A (en) * | 1983-09-26 | 1986-04-15 | Mcneilab, Inc. | Chlorosulfate and azidosulfate esters of tetrahydro-2H-pyran-2-yl-methanol |
-
1992
- 1992-09-15 AU AU24518/92A patent/AU651244B2/en not_active Expired
- 1992-09-15 IL IL10317292A patent/IL103172A/xx not_active IP Right Cessation
- 1992-09-17 CA CA002078519A patent/CA2078519C/en not_active Expired - Lifetime
- 1992-09-17 MY MYPI92001667A patent/MY113564A/en unknown
- 1992-09-17 EG EG54692A patent/EG20164A/xx active
- 1992-09-18 KR KR1019920017043A patent/KR100229180B1/ko not_active IP Right Cessation
- 1992-09-18 MX MX9205305A patent/MX9205305A/es unknown
- 1992-09-18 AT AT92308509T patent/ATE163937T1/de active
- 1992-09-18 PH PH44955A patent/PH31291A/en unknown
- 1992-09-18 HU HU9202974A patent/HU212634B/hu unknown
- 1992-09-18 EP EP92308509A patent/EP0533483B1/en not_active Expired - Lifetime
- 1992-09-18 FI FI924189A patent/FI107731B/fi not_active IP Right Cessation
- 1992-09-18 DE DE69224691T patent/DE69224691T2/de not_active Expired - Lifetime
- 1992-09-18 JP JP27351092A patent/JP3174410B2/ja not_active Expired - Lifetime
- 1992-09-18 DK DK92308509T patent/DK0533483T3/da active
- 1992-09-18 ZW ZW14792A patent/ZW14792A1/xx unknown
- 1992-09-18 NZ NZ244409A patent/NZ244409A/en not_active IP Right Cessation
- 1992-09-18 ES ES92308509T patent/ES2114917T3/es not_active Expired - Lifetime
- 1992-09-18 NO NO923637A patent/NO179284C/no not_active IP Right Cessation
- 1992-09-19 CN CN92111591A patent/CN1035820C/zh not_active Expired - Lifetime
- 1992-11-10 TW TW081108966A patent/TW217413B/zh not_active IP Right Cessation
-
1993
- 1993-08-12 US US08/106,470 patent/US5387700A/en not_active Expired - Lifetime
-
1998
- 1998-04-10 GR GR980400814T patent/GR3026618T3/el unknown
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