PH26408A - Sustained release isuprofen composition - Google Patents
Sustained release isuprofen composition Download PDFInfo
- Publication number
- PH26408A PH26408A PH34733A PH34733A PH26408A PH 26408 A PH26408 A PH 26408A PH 34733 A PH34733 A PH 34733A PH 34733 A PH34733 A PH 34733A PH 26408 A PH26408 A PH 26408A
- Authority
- PH
- Philippines
- Prior art keywords
- sustained release
- weight
- xanthan gum
- formulation
- active ingredient
- Prior art date
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- HEFNNWSXXWATRW-UHFFFAOYSA-N Ibuprofen Chemical compound CC(C)CC1=CC=C(C(C)C(O)=O)C=C1 HEFNNWSXXWATRW-UHFFFAOYSA-N 0.000 claims description 37
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- 239000010346 polypectate Substances 0.000 description 1
- 229920001282 polysaccharide Polymers 0.000 description 1
- 239000005017 polysaccharide Substances 0.000 description 1
- 229920000136 polysorbate Polymers 0.000 description 1
- 229940068965 polysorbates Drugs 0.000 description 1
- 239000011148 porous material Substances 0.000 description 1
- 229920003133 pregelled starch Polymers 0.000 description 1
- 230000002028 premature Effects 0.000 description 1
- 230000001072 progestational effect Effects 0.000 description 1
- 108090000623 proteins and genes Proteins 0.000 description 1
- 102000004169 proteins and genes Human genes 0.000 description 1
- 230000003236 psychic effect Effects 0.000 description 1
- 230000009467 reduction Effects 0.000 description 1
- 239000011347 resin Substances 0.000 description 1
- 229920005989 resin Polymers 0.000 description 1
- 229940125723 sedative agent Drugs 0.000 description 1
- 239000000932 sedative agent Substances 0.000 description 1
- 229910052710 silicon Inorganic materials 0.000 description 1
- 239000010703 silicon Substances 0.000 description 1
- 239000000377 silicon dioxide Substances 0.000 description 1
- 235000012239 silicon dioxide Nutrition 0.000 description 1
- 235000015424 sodium Nutrition 0.000 description 1
- 235000019333 sodium laurylsulphate Nutrition 0.000 description 1
- 239000008247 solid mixture Substances 0.000 description 1
- 239000007892 solid unit dosage form Substances 0.000 description 1
- 235000019698 starch Nutrition 0.000 description 1
- 239000008107 starch Substances 0.000 description 1
- 230000003637 steroidlike Effects 0.000 description 1
- 239000000021 stimulant Substances 0.000 description 1
- 210000002784 stomach Anatomy 0.000 description 1
- 238000003860 storage Methods 0.000 description 1
- 239000005720 sucrose Substances 0.000 description 1
- 235000000346 sugar Nutrition 0.000 description 1
- 150000005846 sugar alcohols Chemical class 0.000 description 1
- 238000009495 sugar coating Methods 0.000 description 1
- 239000000829 suppository Substances 0.000 description 1
- 239000004094 surface-active agent Substances 0.000 description 1
- 230000002195 synergetic effect Effects 0.000 description 1
- 239000007885 tablet disintegrant Substances 0.000 description 1
- 239000000454 talc Substances 0.000 description 1
- 229910052623 talc Inorganic materials 0.000 description 1
- IMCGHZIGRANKHV-AJNGGQMLSA-N tert-butyl (3s,5s)-2-oxo-5-[(2s,4s)-5-oxo-4-propan-2-yloxolan-2-yl]-3-propan-2-ylpyrrolidine-1-carboxylate Chemical compound O1C(=O)[C@H](C(C)C)C[C@H]1[C@H]1N(C(=O)OC(C)(C)C)C(=O)[C@H](C(C)C)C1 IMCGHZIGRANKHV-AJNGGQMLSA-N 0.000 description 1
- 239000002562 thickening agent Substances 0.000 description 1
- QORWJWZARLRLPR-UHFFFAOYSA-H tricalcium bis(phosphate) Chemical compound [Ca+2].[Ca+2].[Ca+2].[O-]P([O-])([O-])=O.[O-]P([O-])([O-])=O QORWJWZARLRLPR-UHFFFAOYSA-H 0.000 description 1
- -1 various gums Substances 0.000 description 1
- 229920003169 water-soluble polymer Polymers 0.000 description 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
Landscapes
- Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Medicinal Preparation (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Steroid Compounds (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB868601204A GB8601204D0 (en) | 1986-01-18 | 1986-01-18 | Therapeutic agents |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| PH26408A true PH26408A (en) | 1992-07-02 |
Family
ID=10591589
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| PH34733A PH26408A (en) | 1986-01-18 | 1987-01-16 | Sustained release isuprofen composition |
Country Status (23)
| Country | Link |
|---|---|
| US (1) | US5415871A (h) |
| EP (1) | EP0234670B1 (h) |
| JP (1) | JPH0669965B2 (h) |
| KR (1) | KR940011242B1 (h) |
| AT (1) | ATE77548T1 (h) |
| AU (2) | AU608208B2 (h) |
| CA (1) | CA1313133C (h) |
| DE (1) | DE3779933T2 (h) |
| DK (1) | DK175215B1 (h) |
| ES (1) | ES2042541T4 (h) |
| FI (1) | FI93608C (h) |
| GB (1) | GB8601204D0 (h) |
| GR (1) | GR3005796T3 (h) |
| IE (1) | IE59333B1 (h) |
| IL (1) | IL81281A (h) |
| IN (1) | IN164250B (h) |
| MX (1) | MX4949A (h) |
| MY (1) | MY100721A (h) |
| NO (1) | NO173317C (h) |
| NZ (1) | NZ218907A (h) |
| PH (1) | PH26408A (h) |
| PT (1) | PT84133B (h) |
| ZA (1) | ZA87173B (h) |
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| US5169639A (en) * | 1988-09-19 | 1992-12-08 | Edward Mendell Co., Inc. | Controlled release verapamil tablets |
| US5128143A (en) * | 1988-09-19 | 1992-07-07 | Edward Mendell Co., Inc. | Sustained release excipient and tablet formulation |
| US5009895A (en) * | 1990-02-02 | 1991-04-23 | Merck & Co., Inc. | Sustained release with high and low viscosity HPMC |
| IT1250483B (it) * | 1990-08-30 | 1995-04-07 | Eurand Int | Sistema di ritardo a matrice multipla |
| DE4140179C2 (de) * | 1991-12-05 | 1995-12-21 | Alfatec Pharma Gmbh | Akutform für ein Ibuprofen enthaltendes Arzneimittel |
| DE4140172C2 (de) * | 1991-12-05 | 1995-12-21 | Alfatec Pharma Gmbh | Retardform für ein Ibuprofen enthaltendes Arzneimittel |
| DE4140192C2 (de) * | 1991-12-05 | 1996-02-29 | Alfatec Pharma Gmbh | Sol-gesteuerte Thermokolloidmatrix auf Gelatinebasis für perorale Retardformen |
| DE4140183C2 (de) * | 1991-12-05 | 1995-12-21 | Alfatec Pharma Gmbh | Retardform für ein Flurbiprofen enthaltendes Arzneimittel |
| DE4140184C2 (de) * | 1991-12-05 | 1995-12-21 | Alfatec Pharma Gmbh | Akutform für ein Flurbiprofen enthaltendes Arzneimittel |
| US5478577A (en) * | 1993-11-23 | 1995-12-26 | Euroceltique, S.A. | Method of treating pain by administering 24 hour oral opioid formulations exhibiting rapid rate of initial rise of plasma drug level |
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1986
- 1986-01-18 GB GB868601204A patent/GB8601204D0/en active Pending
- 1986-12-31 IE IE342086A patent/IE59333B1/en not_active IP Right Cessation
-
1987
- 1987-01-06 DE DE8787300035T patent/DE3779933T2/de not_active Expired - Lifetime
- 1987-01-06 AT AT87300035T patent/ATE77548T1/de not_active IP Right Cessation
- 1987-01-06 EP EP87300035A patent/EP0234670B1/en not_active Expired - Lifetime
- 1987-01-06 ES ES87300035T patent/ES2042541T4/es not_active Expired - Lifetime
- 1987-01-07 IN IN9/MAS/87A patent/IN164250B/en unknown
- 1987-01-12 ZA ZA87173A patent/ZA87173B/xx unknown
- 1987-01-13 NZ NZ218907A patent/NZ218907A/xx unknown
- 1987-01-13 DK DK198700148A patent/DK175215B1/da not_active IP Right Cessation
- 1987-01-14 MY MYPI87000032A patent/MY100721A/en unknown
- 1987-01-15 FI FI870155A patent/FI93608C/fi not_active IP Right Cessation
- 1987-01-15 MX MX494987A patent/MX4949A/es unknown
- 1987-01-16 PT PT84133A patent/PT84133B/pt unknown
- 1987-01-16 CA CA000527498A patent/CA1313133C/en not_active Expired - Fee Related
- 1987-01-16 PH PH34733A patent/PH26408A/en unknown
- 1987-01-16 NO NO870181A patent/NO173317C/no not_active IP Right Cessation
- 1987-01-16 AU AU67625/87A patent/AU608208B2/en not_active Ceased
- 1987-01-16 JP JP62006312A patent/JPH0669965B2/ja not_active Expired - Lifetime
- 1987-01-16 IL IL81281A patent/IL81281A/xx not_active IP Right Cessation
- 1987-01-17 KR KR1019870000334A patent/KR940011242B1/ko not_active Expired - Fee Related
-
1991
- 1991-04-19 US US07/687,090 patent/US5415871A/en not_active Expired - Lifetime
- 1991-06-28 AU AU79462/91A patent/AU628754B2/en not_active Ceased
-
1992
- 1992-09-24 GR GR920402118T patent/GR3005796T3/el unknown
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