PH22672A - Imidazolylmethyltetrahydrocarbazolone derivatives, composition and method of use thereof - Google Patents

Imidazolylmethyltetrahydrocarbazolone derivatives, composition and method of use thereof

Info

Publication number
PH22672A
PH22672A PH31770A PH31770A PH22672A PH 22672 A PH22672 A PH 22672A PH 31770 A PH31770 A PH 31770A PH 31770 A PH31770 A PH 31770A PH 22672 A PH22672 A PH 22672A
Authority
PH
Philippines
Prior art keywords
imidazolylmethyltetrahydrocarbazolone
derivatives
composition
imidazolylmethyltetrahydrocarbazolone derivatives
Prior art date
Application number
PH31770A
Other languages
English (en)
Inventor
Coates Ian Harold
Bell James Angus
Humber David Cedric
Ewan George Blanch
Original Assignee
Glaxo Group Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB848401888A external-priority patent/GB8401888D0/en
Priority claimed from GB848425959A external-priority patent/GB8425959D0/en
Application filed by Glaxo Group Ltd filed Critical Glaxo Group Ltd
Publication of PH22672A publication Critical patent/PH22672A/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/56—Ring systems containing three or more rings
    • C07D209/80—[b, c]- or [b, d]-condensed
    • C07D209/82—Carbazoles; Hydrogenated carbazoles
    • C07D209/88—Carbazoles; Hydrogenated carbazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the ring system
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
PH31770A 1984-01-25 1985-01-25 Imidazolylmethyltetrahydrocarbazolone derivatives, composition and method of use thereof PH22672A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB848401888A GB8401888D0 (en) 1984-01-25 1984-01-25 Heterocyclic compounds
GB848425959A GB8425959D0 (en) 1984-10-15 1984-10-15 Heterocyclic compounds

Publications (1)

Publication Number Publication Date
PH22672A true PH22672A (en) 1988-11-14

Family

ID=26287221

Family Applications (1)

Application Number Title Priority Date Filing Date
PH31770A PH22672A (en) 1984-01-25 1985-01-25 Imidazolylmethyltetrahydrocarbazolone derivatives, composition and method of use thereof

Country Status (29)

Country Link
KR (1) KR920003064B1 (el)
AT (1) AT392276B (el)
AU (1) AU579132B2 (el)
BE (1) BE901576A (el)
CA (1) CA1252793A (el)
CH (1) CH664152A5 (el)
CY (1) CY1479A (el)
CZ (1) CZ404391A3 (el)
DE (2) DE3502508A1 (el)
DK (1) DK169521B1 (el)
ES (3) ES8609309A1 (el)
FI (1) FI84349C (el)
FR (1) FR2561244B1 (el)
GB (1) GB2153821B (el)
GR (1) GR850219B (el)
HK (1) HK33189A (el)
HU (1) HU193592B (el)
IE (1) IE57809B1 (el)
IL (1) IL74165A (el)
IT (1) IT1182150B (el)
LU (2) LU85743A1 (el)
NL (2) NL190373C (el)
NO (2) NO164025C (el)
NZ (1) NZ210940A (el)
PH (1) PH22672A (el)
PT (1) PT79890B (el)
SE (1) SE460359B (el)
SG (1) SG7089G (el)
SK (1) SK404391A3 (el)

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JPH0249772A (ja) * 1988-04-07 1990-02-20 Glaxo Group Ltd イミダゾール誘導体
DK185489A (da) * 1988-04-22 1989-10-23 Duphar Int Res Imidazolylmethyl-cycloalkanoebaaindoloner, deres fremstilling og anvendelse
JPH0256485A (ja) * 1988-04-27 1990-02-26 Glaxo Group Ltd ラクタム誘導体
GB8812636D0 (en) * 1988-05-27 1988-06-29 Glaxo Group Ltd Chemical compounds
AU627221B2 (en) * 1988-09-27 1992-08-20 Fujisawa Pharmaceutical Co., Ltd. Pyridoindole derivatives and processes for preparation thereof
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FR2639944B1 (fr) * 1988-12-06 1991-01-18 Adir Nouveaux derives de l'indole, leur procede de preparation et les compositions pharmaceutiques qui les contiennent
CA2004911A1 (en) * 1988-12-22 1990-06-22 Mitsuaki Ohta 4,5,6,7-tetrahydrobenzimidazole derivatives
US5223625A (en) * 1988-12-22 1993-06-29 Duphar International Research B.V. Annelated indolo [3,2,-C]lactams
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DK0422154T3 (da) * 1989-04-21 1994-03-07 Sandoz Ag Terapeutisk anvendelse af 5-HT3-receptorantagonister
GB8914804D0 (en) * 1989-06-28 1989-08-16 Glaxo Group Ltd Process
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US5276050A (en) * 1989-08-01 1994-01-04 Glaxo Group Limited Medicaments
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GB2236751B (en) 1989-10-14 1993-04-28 Wyeth John & Brother Ltd Heterocyclic compounds
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US5187166A (en) * 1990-07-31 1993-02-16 Nisshin Flour Milling Co., Ltd. Azabicyclo derivatives and their use as antiemetics
EP1022025A3 (en) * 1991-06-26 2002-06-05 Sepracor, Inc. Method and compositions for treating emesis nausea and other disorders using optically pure R(+) ondansetron
JPH05310732A (ja) * 1992-03-12 1993-11-22 Mitsubishi Kasei Corp シンノリン−３−カルボン酸誘導体
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CA2106642C (en) * 1992-10-14 2005-08-16 Peter Bod Carbazolone derivatives and process for preparing the same
HU212934B (en) 1992-10-14 1996-12-30 Richter Gedeon Vegyeszet Process for producing novel alkoxalylated carbazolone derivatives
KR960700711A (ko) * 1993-03-08 1996-02-24 후지야마 아키라 뇌혈관성 질환의 치료 또는 예방용 약제(Medicament for treating or preventing cerebrovascular diseases)
GB9310756D0 (en) * 1993-05-25 1993-07-14 Glaxo Lab Sa Compositions
GB2325408B (en) * 1994-06-28 1999-01-27 Kenneth Francis Prendergast Chewing gum formulation comprising ondansetron
GB9423588D0 (en) * 1994-11-22 1995-01-11 Glaxo Wellcome Inc Compositions
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US5969137A (en) * 1996-09-19 1999-10-19 Virginia Commonwealth University Benzylamidine derivatives with serotonin receptor binding activity
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FI6164U1 (fi) * 2003-01-09 2004-03-15 Synthon Bv Ondansetronmuotoja
GB2398071B (en) * 2003-01-24 2006-06-07 Synthon Bv Process for making ondansetron and intermediate thereof
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US20090170872A1 (en) * 2005-07-05 2009-07-02 Orchid Research Laboratories Limited Compounds and Their Pharmaceutical Use
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US3634420A (en) * 1969-05-09 1972-01-11 American Cyanamid Co 3(morpholinomethyl)-2 3-dihydro-carbazol-4(1h)-ones
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Also Published As

Publication number Publication date
FI850323A0 (fi) 1985-01-25
ES8801247A1 (es) 1987-12-16
IT8547600A0 (it) 1985-01-25
IE57809B1 (en) 1993-04-21
ES539852A0 (es) 1986-07-16
ES556101A0 (es) 1987-12-16
NL190373B (nl) 1993-09-01
GB2153821B (en) 1988-01-20
CY1479A (en) 1989-07-21
HUT37784A (en) 1986-02-28
SK277923B6 (en) 1995-08-09
DE3502508C2 (el) 1990-05-03
LU85743A1 (fr) 1986-08-04
GR850219B (el) 1985-05-23
SE460359B (sv) 1989-10-02
NL940009I2 (nl) 1999-05-03
SE8500368L (sv) 1985-07-26
NL190373C (nl) 1994-02-01
ATA20485A (de) 1990-08-15
AU579132B2 (en) 1988-11-17
CH664152A5 (fr) 1988-02-15
SE8500368D0 (sv) 1985-01-25
ES8708224A1 (es) 1987-10-01
NZ210940A (en) 1989-08-29
DE19375046I2 (de) 2002-10-10
GB2153821A (en) 1985-08-29
DE3502508A1 (de) 1985-08-14
IL74165A (en) 1988-11-15
AU3809785A (en) 1985-08-01
PT79890A (en) 1985-02-01
NO164025C (no) 1990-08-22
FI84349C (fi) 1991-11-25
NL8500202A (nl) 1985-08-16
SK404391A3 (en) 1995-08-09
IT1182150B (it) 1987-09-30
DK35785A (da) 1985-07-26
NO164025B (no) 1990-05-14
KR920003064B1 (ko) 1992-04-13
DK35785D0 (da) 1985-01-25
FI84349B (fi) 1991-08-15
NO1994022I1 (no) 1994-11-09
NL940009I1 (nl) 1994-07-18
ES548430A0 (es) 1987-10-01
HU193592B (en) 1987-11-30
GB8501889D0 (en) 1985-02-27
BE901576A (fr) 1985-07-25
FI850323L (fi) 1985-07-26
KR850005439A (ko) 1985-08-26
NO850300L (no) 1985-07-26
DK169521B1 (da) 1994-11-21
FR2561244B1 (fr) 1988-03-04
HK33189A (en) 1989-04-28
FR2561244A1 (fr) 1985-09-20
AT392276B (de) 1991-02-25
CA1252793A (en) 1989-04-18
SG7089G (en) 1989-06-09
LU88268I2 (el) 1994-02-03
IE850187L (en) 1985-07-25
ES8609309A1 (es) 1986-07-16
CZ404391A3 (en) 1993-04-14
PT79890B (en) 1987-02-03

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