PH12012500809A1 - Methods and compositions for treating cancer - Google Patents

Methods and compositions for treating cancer

Info

Publication number
PH12012500809A1
PH12012500809A1 PH1/2012/500809A PH12012500809A PH12012500809A1 PH 12012500809 A1 PH12012500809 A1 PH 12012500809A1 PH 12012500809 A PH12012500809 A PH 12012500809A PH 12012500809 A1 PH12012500809 A1 PH 12012500809A1
Authority
PH
Philippines
Prior art keywords
compositions
thyl
treating cancer
methods
pyridazin
Prior art date
Application number
PH1/2012/500809A
Other languages
English (en)
Inventor
William C Shakespeare
Timothy P Clackson
Victor M Rivera
Wei-Sheng Huang
Joseph M Gozgit
Rachel M Squillace
Original Assignee
Ariad Pharma Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=43922622&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=PH12012500809(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Ariad Pharma Inc filed Critical Ariad Pharma Inc
Publication of PH12012500809A1 publication Critical patent/PH12012500809A1/en

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/50—Pyridazines; Hydrogenated pyridazines
    • A61K31/5025—Pyridazines; Hydrogenated pyridazines ortho- or peri-condensed with heterocyclic ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/02—Antineoplastic agents specific for leukemia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Epidemiology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Hematology (AREA)
  • Oncology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicinal Preparation (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
PH1/2012/500809A 2009-10-30 2010-11-01 Methods and compositions for treating cancer PH12012500809A1 (en)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US25669009P 2009-10-30 2009-10-30
US25666909P 2009-10-30 2009-10-30
US26101409P 2009-11-13 2009-11-13
PCT/US2010/055016 WO2011053938A1 (en) 2009-10-30 2010-11-01 Methods and compositions for treating cancer

Publications (1)

Publication Number Publication Date
PH12012500809A1 true PH12012500809A1 (en) 2012-11-26

Family

ID=43922622

Family Applications (1)

Application Number Title Priority Date Filing Date
PH1/2012/500809A PH12012500809A1 (en) 2009-10-30 2010-11-01 Methods and compositions for treating cancer

Country Status (16)

Country Link
US (2) US20120316137A1 (enExample)
EP (2) EP2493460A4 (enExample)
JP (1) JP2013509444A (enExample)
KR (1) KR20120115237A (enExample)
CN (1) CN102770129A (enExample)
AU (1) AU2010313152A1 (enExample)
CA (1) CA2777128A1 (enExample)
CL (1) CL2012001133A1 (enExample)
CR (1) CR20120202A (enExample)
EA (1) EA201290255A1 (enExample)
IL (1) IL218987A0 (enExample)
MX (1) MX2012005023A (enExample)
NI (1) NI201200072A (enExample)
PH (1) PH12012500809A1 (enExample)
WO (1) WO2011053938A1 (enExample)
ZA (1) ZA201202256B (enExample)

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CN106236732A (zh) * 2016-08-31 2016-12-21 佛山市弘泰药物研发有限公司 一种依维莫司软胶囊的制备方法
CN110291081B (zh) * 2016-12-15 2023-01-31 阿瑞雅德制药公司 作为c-kit抑制剂的苯并咪唑化合物
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CN109875999B (zh) * 2018-05-29 2022-07-12 上海交通大学医学院附属第九人民医院 泊那替尼在kit突变型恶性黑色素瘤中的应用
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Also Published As

Publication number Publication date
EP2493460A4 (en) 2013-04-24
EP2762142A1 (en) 2014-08-06
CL2012001133A1 (es) 2013-08-02
CN102770129A (zh) 2012-11-07
MX2012005023A (es) 2012-06-19
WO2011053938A1 (en) 2011-05-05
EP2493460A1 (en) 2012-09-05
WO2011053938A8 (en) 2011-08-11
JP2013509444A (ja) 2013-03-14
ZA201202256B (en) 2012-12-27
IL218987A0 (en) 2012-06-28
NI201200072A (es) 2012-08-20
KR20120115237A (ko) 2012-10-17
CR20120202A (es) 2012-06-12
US20130178622A1 (en) 2013-07-11
AU2010313152A1 (en) 2012-04-19
US20120316137A1 (en) 2012-12-13
EA201290255A1 (ru) 2013-04-30
CA2777128A1 (en) 2011-05-05

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